ChemicalBook > CAS DataBase List > Docarpamine

Docarpamine

Product Name
Docarpamine
CAS No.
74639-40-0
Chemical Name
Docarpamine
Synonyms
TA 870;TA-8704;Tanadopa;Docarpamine;3,4-Bis[(ethoxycarbonyl)oxy]-N-(N-acetyl-L-methionyl)benzeneethanamine;4-{2-[(N-Acetyl-L-methionyl)amino]ethyl}-1,2-phenylenediethylbiscarbonate;(S)-2-(Acetylamino)-N-[3,4-bis(ethoxycarbonyloxy)phenethyl]-4-(methylthio)butanamide;Carbonic acid, 4-[2-[[(2S)-2-(acetylamino)-4-(methylthio)-1-oxobutyl]amino]ethyl]-1,2-phenylene diethyl ester;Carbonic acid, 4-[2-[[2-(acetylamino)-4-(methylthio)-1-oxobutyl]amino]ethyl]-1,2-phenylene diethyl ester, (S)-;Carbonic acid, C,C'-[4-[2-[[2-(acetylamino)-4-(methylthio)-1-oxobutyl]amino]ethyl]-1,2-phenylene] C,C'-diethyl ester
CBNumber
CB21178560
Molecular Formula
C21H30N2O8S
Formula Weight
470.54
MOL File
74639-40-0.mol
More
Less

Docarpamine Property

Melting point:
85-90°; mp 105-108° (Nishiyama, 1992)
alpha 
D20 -15.6° (c = 2 in methanol)
Boiling point:
731.0±60.0 °C(Predicted)
Density 
1.222±0.06 g/cm3(Predicted)
pka
14.51±0.46(Predicted)
More
Less

Safety

Toxicity
LD50 in male, female rats (mg/kg): 1000-1400, ~1000 s.c.; in rats, dogs (mg/kg): _>2000 orally (Nishiyama, 1992)
More
Less

Hazard and Precautionary Statements (GHS)

More
Less

N-Bromosuccinimide Price

American Custom Chemicals Corporation
Product number
API0002463
Product name
DOCARPAMINE
Purity
95.00%
Packaging
5MG
Price
$497.54
Updated
2021/12/16
More
Less

Docarpamine Chemical Properties,Usage,Production

Description

Docarpamine is a cardiostimulant with diuretic activity launched in Japan for the treatment of circulatory insufficiency. It is an orally effective peripheral dopamine prodrug that is well absorbed from the gastrointestinal tract and converted to dopamine in vivo, which exerts renal vasodilatory and natriuretic effects by activating renal dopamine (DA1) receptors, and a positive inotropic effect by activating cardiac β1-receptors. It has been reported to be effective in treating patients with acute heart failure, shock and acute renal failure.

Originator

Tanabe Seiyaku (Japan)

Uses

Docarpamine maybe a usefule alternative to intravenous dopamine after cardiac surgery.

Definition

ChEBI: Docarpamine is an organic molecular entity.

brand name

Tanadopa

Docarpamine Preparation Products And Raw materials

Raw materials

Preparation Products

More
Less

Docarpamine Suppliers

SHANGHAI HOHANCE CHEMICAL CO.,LTD
Tel
021-31115312 18217084087
Fax
86 021 31115317
Email
mary@hohance.com
Country
China
ProdList
143
Advantage
62
RR Scientific LLC
Tel
+86-13917743231
Email
sales@rrscientific.com
Country
United States
ProdList
878
Advantage
58
BOC Sciences
Tel
+1-631-485-4226
Fax
1-631-614-7828
Email
inquiry@bocsci.com
Country
United States
ProdList
19553
Advantage
58
Hubei Shishun Biotechnology Co. Ltd
Tel
027-59223025 15107168801
Fax
027-59223025
Email
1718480011@qq.com
Country
China
ProdList
9865
Advantage
58
Hubei Guangao Biotechnology Co., Ltd
Tel
027-027-59223056 18162699093
Fax
027-59223056
Email
1208480011@qq.com
Country
China
ProdList
9924
Advantage
58
Hubei Qifei Pharmaceutical Chemical Co., Ltd
Tel
027-027-59322506 18071128681
Fax
027-59322506
Email
1438082200@qq.com
Country
China
ProdList
9976
Advantage
58
R.R Scientific, LLC.
Tel
15010167677
Email
zhiyuu1218@163.com
Country
China
ProdList
876
Advantage
58
Shaanxi Didu New Material Co., Ltd
Tel
029-81145920 15353716720
Email
1046@dideu.com
Country
China
ProdList
9983
Advantage
58
Weifu (Shanghai) Pharmaceutical Technology Co., LTD
Tel
021-57609736 13524092974;
Email
info@shanghaiweifu.cn
Country
China
ProdList
237
Advantage
58
TLC Pharmaceutical Standards Ltd.
Tel
18012923235
Email
chinasales04@tlcstandards.com.cn
Country
China
ProdList
4925
Advantage
58

74639-40-0, DocarpamineRelated Search:


  • Docarpamine
  • Carbonic acid, 4-[2-[[(2S)-2-(acetylamino)-4-(methylthio)-1-oxobutyl]amino]ethyl]-1,2-phenylene diethyl ester
  • Carbonic acid, 4-[2-[[2-(acetylamino)-4-(methylthio)-1-oxobutyl]amino]ethyl]-1,2-phenylene diethyl ester, (S)-
  • TA 870
  • Tanadopa
  • (S)-2-(Acetylamino)-N-[3,4-bis(ethoxycarbonyloxy)phenethyl]-4-(methylthio)butanamide
  • 3,4-Bis[(ethoxycarbonyl)oxy]-N-(N-acetyl-L-methionyl)benzeneethanamine
  • TA-8704
  • Carbonic acid, C,C'-[4-[2-[[2-(acetylamino)-4-(methylthio)-1-oxobutyl]amino]ethyl]-1,2-phenylene] C,C'-diethyl ester
  • 4-{2-[(N-Acetyl-L-methionyl)amino]ethyl}-1,2-phenylenediethylbiscarbonate
  • 74639-40-0
  • C21H30N2O8S