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Ocaperidone

Product Name
Ocaperidone
CAS No.
129029-23-8
Chemical Name
Ocaperidone
Synonyms
R79598;Ocaperidona;Ocaperidone;Ocaperidone (R79598);Ocaperidone USP/EP/BP;Ocaperidone, 10 mM in DMSO;3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-2,9-dimethylpyrido[1,2-a]pyrimidin-4-one;3-(2-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethyl)-2,9-dimethyl-4H-pyrido[1,2-a]pyrimidin-4-one;4H-Pyrido[1,2-a]pyrimidin-4-one, 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-2,9-dimethyl-;5-hydroxytryptamine Receptor,Ocaperidone,inhibit,Serotonin Receptor,R 79598,Inhibitor,Dopamine Receptor,5-HT Receptor,R-79598
CBNumber
CB21179370
Molecular Formula
C24H25FN4O2
Formula Weight
420.48
MOL File
129029-23-8.mol
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Ocaperidone Property

Melting point:
180.0 to 184.0 °C
Boiling point:
588.0±60.0 °C(Predicted)
Density 
1.32 g/cm3
storage temp. 
2-8°C
solubility 
DMSO:16.0(Max Conc. mg/mL);38.1(Max Conc. mM)
pka
7.97±0.10(Predicted)
form 
powder to crystal
color 
White to Light yellow
CAS DataBase Reference
129029-23-8
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Safety

HS Code 
2934.99.3000
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

TCI Chemical
Product number
O0498
Product name
Ocaperidone
Purity
>98.0%(HPLC)
Packaging
25mg
Price
$138
Updated
2025/07/31
TCI Chemical
Product number
O0498
Product name
Ocaperidone
Purity
>98.0%(HPLC)
Packaging
100mg
Price
$415
Updated
2025/07/31
TRC
Product number
O234005
Product name
Ocaperidone
Packaging
1mg
Price
$50
Updated
2021/12/16
ChemScene
Product number
CS-0020804
Product name
Ocaperidone
Purity
99.63%
Packaging
5mg
Price
$110
Updated
2021/12/16
ChemScene
Product number
CS-0020804
Product name
Ocaperidone
Purity
99.63%
Packaging
10mg
Price
$150
Updated
2021/12/16
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Ocaperidone Chemical Properties,Usage,Production

Uses

Antipsychotic.

Definition

ChEBI: Ocaperidone is a pyridopyrimidine.

in vivo

Ocaperidone shows a potent occupation of 5HT2 receptor via in vivo binding in the frontal cortex of rats with an ED50 of 0.04 mg/kg, and 0.1 4-0.1 6 mg/kg for D2 receptor in the striatum and the nucleus accumbens[1]. Ocaperidone (R 79598) antagonizes dopamine D2 and 5-HT2, and shows a a partial generalization to buspirone with an ED50 of 0.163 mg/kg[3].

IC 50

5-HT2 Receptor: 0.14 nM (Ki); a1-adrenergic receptor: 0.46 nM (Ki); D2 Receptor: 0.75 nM (Ki); Histamine H1: 1.6 nM (Ki); a2-adrenergic receptor: 5.4 nM (Ki); 5-HT1A Receptor: 7.6 (pEC50, h5-HT1A); 5-HT1A Receptor: 8.08 (pKi, h5-HT1A)

Ocaperidone Preparation Products And Raw materials

Raw materials

Preparation Products

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Ocaperidone Suppliers

Americas 1 China 45 Europe 1 India 2 Japan 1 United States 6 Global 56
Jiangsu Aikon Biopharmaceutical R&D co.,Ltd.
Tel
025-66113011 17798518460
Fax
(1)02557626880
Email
cfzhang@aikonchem.com
Country
China
ProdList
19913
Advantage
55
TOKYO CHEMICAL INDUSTRY CO., LTD.
Tel
03-36680489
Fax
03-3668-0520
Email
Sales-JP@TCIchemicals.com
Country
Japan
ProdList
28387
Advantage
80
TCI Europe
Tel
320-37350700
Fax
+32 (0)37350701
Email
sales@tcieurope.eu
Country
Europe
ProdList
23671
Advantage
75
TCI AMERICA
Tel
800-4238616
Fax
+1-888-520-1075 / +1-503-283-1987
Email
sales@tciamerica.com
Country
Americas
ProdList
23653
Advantage
75
Shanghai EFE Biological Technology Co., Ltd.
Tel
021-65675885 18964387627
Fax
021-65675885
Email
info@efebio.com
Country
China
ProdList
9803
Advantage
58
Shanghai YuanYe Biotechnology Co., Ltd.
Tel
021-61312847; 18021002903
Fax
QQ:3008007432
Email
3008007409@qq.com
Country
China
ProdList
71826
Advantage
60
ShangHai Biochempartner Co.,Ltd
Tel
177-54423994 17754423994
Fax
QQ:2853530913
Email
2853530910@QQ.com
Country
China
ProdList
8000
Advantage
62
Shanghai SuperLan Chemcial Technique Centre
Tel
0-2022843681 15618226720
Fax
+86-21-51601218
Email
chaolaichem@foxmail.com
Country
China
ProdList
12475
Advantage
58
Amadis Chemical Company Limited
Tel
571-89925085
Fax
0086-571-89925065
Email
sales@amadischem.com
Country
China
ProdList
131957
Advantage
58
Angel Pharmatech, Ltd.
Tel
17317130613
Fax
QQ3358272972
Email
3358272972@qq.com
Country
China
ProdList
3276
Advantage
58
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View Lastest Price from Ocaperidone manufacturers

Dideu Industries Group Limited
Product
Ocaperidone 129029-23-8
Price
US $1.10/g
Min. Order
1g
Purity
99.9%
Supply Ability
100 Tons min
Release date
2021-07-23

129029-23-8, OcaperidoneRelated Search:

Carbamazepine Risperidone Capecitabine Sorafenib Cefoperazone Cefoperazone sodium +sulbactam sodium(1:1/2:1) 3-METHYL-1,2-BENZISOXAZOLE Dimethallylamine 6-FLUORO-3-METHYLBENZODISOXAZOLE 3-Piperidin-4-ylbenzo[d]isoxazole 6-Fluoro-3-(4-piperidinyl)-1,2-benzisoxazole hydrochloride 1,2-BENZISOXAZOLE Ocaperidone

  • Ocaperidone
  • Ocaperidona
  • 3-(2-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethyl)-2,9-dimethyl-4H-pyrido[1,2-a]pyrimidin-4-one
  • 3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-2,9-dimethylpyrido[1,2-a]pyrimidin-4-one
  • R79598
  • 4H-Pyrido[1,2-a]pyrimidin-4-one, 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-2,9-dimethyl-
  • Ocaperidone USP/EP/BP
  • Ocaperidone (R79598)
  • 5-hydroxytryptamine Receptor,Ocaperidone,inhibit,Serotonin Receptor,R 79598,Inhibitor,Dopamine Receptor,5-HT Receptor,R-79598
  • Ocaperidone, 10 mM in DMSO
  • 129029-23-8