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PHYSOSTIGMINE SALICYLATE

Product Name
PHYSOSTIGMINE SALICYLATE
CAS No.
57-64-7
Chemical Name
PHYSOSTIGMINE SALICYLATE
Synonyms
ESERINE SALICYLATE;Physostigmine-d3 salicylate;ar-44;tl-1380;CCRIS 3405;Isopto Eserine;EINECS 200-343-8;physostolsalicylate;Physostigminsalicylat;ESERINE MONOSALICYLATE
CBNumber
CB2146890
Molecular Formula
C22H27N3O5
Formula Weight
413.47
MOL File
57-64-7.mol
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PHYSOSTIGMINE SALICYLATE Property

Melting point:
181-183 °C
storage temp. 
-20°C
solubility 
DMF: 30 mg/ml,DMSO: 10 mg/ml,Ethanol: 1 mg/ml,PBS (pH 7.2): 1 mg/ml
pka
pKa 1.96/8.08(H2O,t =15) (Uncertain)
form 
Solid
color 
White to yellow
Merck 
7384
BRN 
3900576
InChI
InChI=1/C15H21N3O2.C7H6O3/c1-15-7-8-17(3)13(15)18(4)12-6-5-10(9-11(12)15)20-14(19)16-2;8-6-4-2-1-3-5(6)7(9)10/h5-6,9,13H,7-8H2,1-4H3,(H,16,19);1-4,8H,(H,9,10)/t13-,15+;/s3
InChIKey
HZOTZTANVBDFOF-DPKVYHSMNA-N
SMILES
C12C=C(C=CC=1N(C)[C@@]1([H])N(CC[C@@]21C)C)OC(=O)NC.C1(C(=O)O)=CC=CC=C1O |&1:8,13,r|
CAS DataBase Reference
57-64-7(CAS DataBase Reference)
EPA Substance Registry System
Physostigmine salicylate (57-64-7)
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Safety

Hazard Codes 
T+
Risk Statements 
26/28
Safety Statements 
25-45
RIDADR 
UN 1544 6.1/PG 1
WGK Germany 
3
RTECS 
TJ2450000
HazardClass 
6.1(a)
PackingGroup 
II
HS Code 
2939800000
Toxicity
LD50 i.p. in mice: 0.64 mg/kg (Sofia, Knabloch)
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Danger
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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
P1600000
Product name
Physostigmine salicylate
Purity
European Pharmacopoeia (EP) Reference Standard
Packaging
p1600000
Price
$220
Updated
2024/03/01
Sigma-Aldrich
Product number
1537003
Product name
Physostigmine salicylate
Purity
United States Pharmacopeia (USP) Reference Standard
Packaging
200mg
Price
$436
Updated
2024/03/01
TRC
Product number
P398510
Product name
Physostigmine salicylate
Packaging
50mg
Price
$765
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
AAA0003349
Product name
ESERINE SALICYLATE SALT
Purity
95.00%
Packaging
1G
Price
$2737.84
Updated
2021/12/16
ChemScene
Product number
CS-0013051
Product name
Physostigmine salicylate
Purity
≥99.00%
Packaging
100mg
Price
$300
Updated
2021/12/16
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PHYSOSTIGMINE SALICYLATE Chemical Properties,Usage,Production

Chemical Properties

solid

Uses

Physostigmine salicylate (Eserine salicylate) is used as bulk pharmaceuticals (parasympathomimetic, cholinergic, ophthalmic, anti-Alzheimer). Product Data Sheet

Uses

cholinergic, anticholinesterase, miotic

Definition

ChEBI: Physostigmine salicylate is an azaheterocycle salicylate salt and a member of salicylates. It contains a physostigmine.

brand name

Antilirium (Forest); Isopto Eserine (Alcon).

General Description

The salicylate ofphysostigmine (eserine salicylate) may be prepared byneutralizing an ethereal solution of the alkaloid with anethereal solution of salicylic acid. Excess salicylic acid isremoved from the precipitated product by washing itwith ether. The salicylate is less deliquescent than thesulfate.
Physostigmine salicylate occurs as a white, shining,odorless crystal or white powder that is soluble in water(1:75), alcohol (1:16), or chloroform (1:6) but much lesssoluble in ether (1:250). On prolonged exposure to air andlight, the crystals turn red. The red may be removed bywashing the crystals with alcohol, although this causes lossof the compound as well. Aqueous solutions are neutral orslightly acidic and take on a red coloration after a period.The coloration may be taken as an index of the loss of activityof physostigmine solutions.

General Description

Crystal form that turns red on exposure to heat or light.

Reactivity Profile

Behaves as a weak acid in solution.

Health Hazard

PHYSOSTIGMINE SALICYLATE is similar to physostigmine. It is classified as super toxic. The probable oral lethal dose (humans) is less than 5 mg/kg or a taste for a 150 lb. person. It is a cholinesterase inhibitor.

Fire Hazard

When heated to decomposition, PHYSOSTIGMINE SALICYLATE emits toxic fumes of nitrogen oxides.

Safety Profile

Poison by ingestion, subcutaneous, intramuscular, intravenous, and intraperitoneal routes. Human systemic effects: arrhythmias, nausea or vomiting. Experimental reproductive effects. When heated to decomposition it emits toxic fumes of NOx See also PHYSOSTIGMINE.

PHYSOSTIGMINE SALICYLATE Preparation Products And Raw materials

Raw materials

Preparation Products

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PHYSOSTIGMINE SALICYLATE Suppliers

Shanghai Leiming Medical Technology Co., LTD
Tel
13761371720
Email
zhangleitao111@sina.com
Country
China
ProdList
475
Advantage
58
Meryer (Shanghai) Chemical Technology Co., Ltd.
Tel
021-61259108 18621169109
Fax
86-21-61259102
Email
market03@meryer.com
Country
China
ProdList
40228
Advantage
62
3B Pharmachem (Wuhan) International Co.,Ltd.
Tel
821-50328103-801 18930552037
Fax
86-21-50328109
Email
3bsc@sina.com
Country
China
ProdList
15839
Advantage
69
Chembest Research Laboratories Limited
Tel
+86-21-20908456
Fax
021-58180499
Email
sales@BioChemBest.com
Country
China
ProdList
6005
Advantage
61
Beijing HwrkChemical Technology Co., Ltd
Tel
010-89508211 18501085097
Fax
010-89508210
Email
sales.bj@hwrkchemical.com
Country
China
ProdList
8415
Advantage
55
Syntechem Co.,Ltd
Tel
Fax
E-Mail Inquiry
Email
info@syntechem.com
Country
China
ProdList
12984
Advantage
57
Spectrum Chemical Manufacturing Corp.
Tel
021-021-021-67601398-809-809-809 15221380277
Fax
021-57711696
Email
marketing_china@spectrumchemical.com
Country
China
ProdList
9658
Advantage
60
Beijing Yisiyan Technology Research Center
Tel
010-56645598 13366904824
Fax
01062230033
Email
bjkaida@163.com
Country
China
ProdList
1637
Advantage
59
UHN Shanghai Research & Development Co., Ltd.
Tel
021-58958002 18930822973
Fax
+86 (21) 5895-8628
Email
SALES@UHNSHANGHAI.COM
Country
China
ProdList
977
Advantage
58
Guangzhou Isun Pharmaceutical Co., Ltd
Tel
020-39119399 18927568969
Fax
020-39119999
Email
isunpharm@qq.com
Country
China
ProdList
4428
Advantage
55
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View Lastest Price from PHYSOSTIGMINE SALICYLATE manufacturers

Dideu Industries Group Limited
Product
PHYSOSTIGMINE SALICYLATE 57-64-7
Price
US $1.10/g
Min. Order
1g
Purity
99.9%
Supply Ability
100 Tons min
Release date
2021-07-27

57-64-7, PHYSOSTIGMINE SALICYLATERelated Search:


  • PHYSOSTIGMINE SALICYLATE SALT
  • 2-hydroxy-,compd.with(3as-cis)-1,2,3,3a,8,8a-hexahydro-1,3a,8-benzoicaci
  • ar-44
  • ESERINE MONOSALICYLATE
  • ESERINE SALICYLATE
  • ESERINE SALICYLATE SALT
  • ESERINE SALICYLATE 99.9%
  • Physostigmine monosalicylate
  • Physostigmine salicylate (Eserine salicylate)
  • Benzoic acid, 2-hydroxy-, compd. with (3aS,8aR)-1,2,3,3a,8,8a-hexahydro-1,3a,8-trimethylpyrrolo2,3-bindol-5-yl methylcarbamate (1:1)
  • PHYSOSTIGMINESALICYLATE,USP
  • ESERINE SALICYLATE(RG)
  • Benzoic acid, 2-hydroxy-, compd. with (3aS,8aR)-1,2,3,3a,8,8a-hexahydro-1,3a,8-trimethylpyrrolo[2,3-b]indol-5-yl methylcarbamate (1:1) (9CI)
  • Benzoic acid, 2-hydroxy-, compd. with (3aS-cis)-1,2,3,3a,8,8a-hexahydro-1,3a,8-trimethylpyrrolo[2,3-b]indol-5-yl methylcarbamate (1:1)
  • Isopto Eserine
  • Physostigmine salicylate (6CI)
  • Physostigmine, monosalicylate (8CI)
  • Pyrrolo[2,3-b]indol-5-ol, 1,2,3,3a,8,8a-hexahydro-1,3a,8-trimethyl-, methylcarbamate (ester), (3aS,8aR)-, mono(2-hydroxybenzoate) (salt) (9CI)
  • Pyrrolo[2,3-b]indol-5-ol, 1,2,3,3a,8,8a-hexahydro-1,3a,8-trimethyl-, methylcarbamate (ester), (3aS-cis)-, mono(2-hydroxybenzoate) (salt)
  • Salicylic acid, compd. with physostigmine (1:1) (8CI)
  • Physostigminsalicylat
  • Benzoicacid,2-hydroxy-,cpmpd,with(3aS-cis)-1,2,3,3a,8,8a-hexahydro-1,3a,8-trimethylpyrrolo[2,3-b]indo1-5-ylmethylcarbamateester(1:1)
  • physostigmine,[salicylate(1:1)]
  • physostigmine,salicylate(1:1)
  • physostolsalicylate
  • salicylicacid,compd.withphysostigmine(1:1)
  • tl-1380
  • trimethylpyrrolo[2,3-b]indol-5-ylmethylcarbamate(1:1)
  • Physostigmine Salicylate (200 mg)
  • Physostigmine-d3 salicylate
  • (3aS,8aR)-1,3a,8-triMethyl-1,2,3,3a,8,8a-hexahydropyrrolo[2,3-b]indol-5-yl MethylcarbaMate 2-hydroxybenzoate
  • Eserine salicylate salt >=97.0% (N)
  • Physostigmine salicylate CRS
  • (?)-Physostigmine (salicylate)
  • PHYSOSTIGMINE SALICYLATE USP/EP/BP
  • PHYSOSTIGMINE SALICYLATE INJECTION
  • Physostigmine Salicylate (1537003)
  • inhibit,Eserine,antidote,Physostigmine,blood-brain,Physostigmine Salicylate,Alzheimer's,Cholinesterase (ChE),Inhibitor,barrier
  • CCRIS 3405
  • EINECS 200-343-8
  • Physostigmine Salicylate
  • 57-64-7
  • C22H27N3O5
  • C15H21N3O2C7H6O3
  • Analytical Standards
  • Analytical Chromatography Product Catalog
  • Alkaloids
  • Indole Alkaloids
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  • Chromatography
  • EQ - EZ
  • Forensic and Veterinary Standards
  • Inhibitors
  • ANTILIRIUM
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