STIRIPENTOL

Product Name: STIRIPENTOL
CAS No.: 49763-96-4
Chemical Name: STIRIPENTOL
Synonyms: Diacomit;bcx2600;RCX-2600;Slipperto;STIRIPENTOL;Stiripentol >BCX2600|||Diacomit;Stiripentol, ≥ 98.0%;Stiripentol(BCX 2600);STIRIPENTOL USP/EP/BP
CBNumber: CB2150457
Molecular Formula: C14H18O3
Formula Weight: 234.29
MOL File: 49763-96-4.mol

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STIRIPENTOL Property

Melting point:: 73-74°C
Boiling point:: 365.4±11.0 °C(Predicted)
Density: 1.139±0.06 g/cm3(Predicted)
storage temp.: -20°C
solubility: DMSO: ≥20mg/mL
pka: 14.45±0.20(Predicted)
form: powder
color: white to beige
InChIKey: IBLNKMRFIPWSOY-FNORWQNLSA-N
CAS DataBase Reference: 49763-96-4

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Safety

Hazard Codes: Xn
Risk Statements: 22
WGK Germany: 3
RTECS: SB3393000
HS Code: 2932.99.7000

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Hazard and Precautionary Statements (GHS)

Symbol(GHS)

Signal word

Warning

Hazard statements

H302Harmful if swallowed

Precautionary statements

P280Wear protective gloves/protective clothing/eye protection/face protection.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

Sigma-Aldrich

Product number: S6826
Product name: Stiripentol
Purity: ≥98% (HPLC)
Packaging: 5mg
Price: $87.5
Updated: 2024/03/01

Sigma-Aldrich

Product number: S6826
Product name: Stiripentol
Purity: ≥98% (HPLC)
Packaging: 25mg
Price: $354
Updated: 2024/03/01

TCI Chemical

Product number: S0905
Product name: Stiripentol
Purity: >98.0%(GC)
Packaging: 1g
Price: $245
Updated: 2024/03/01

TCI Chemical

Product number: S0905
Product name: Stiripentol
Purity: >98.0%(GC)
Packaging: 5g
Price: $846
Updated: 2024/03/01

Cayman Chemical

Product number: 17781
Product name: Stiripentol
Purity: ≥98%
Packaging: 5mg
Price: $68
Updated: 2024/03/01

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STIRIPENTOL Chemical Properties,Usage,Production

Description

Stiripentol is a third-generation antiepileptic compound. It is a positive allosteric modulator of GABA_A receptors, potentiating GABA-mediated activation to a greater extent in receptors expressing α₃ subunits and to a lower extent in those containing β₁ or ε subunits. It also inhibits GABA reuptake in vitro and increases the release of GABA in neonatal rat hippocampal slices. Stiripentol (500 μM) inhibits lactate dehydrogenase (LDH), blocking both lactate-to-pyruvate and pyruvate-to-lactate conversions by human LDH1 and LDH5. Formulations containing stiripentol have been used in the adjunctive treatment of seizures associated with Dravet syndrome.

Chemical Properties

White Solid

Uses

An antiepileptic drug

Uses

Stiripentol has been used in pharmacokinetic analysis and as a reference standard in fluorescence spectra analysis.

Uses

Stiripentol is an epilepsy drug, it has been used as co-therapy for treatment of epilepsy.

Definition

ChEBI: 1-(1,3-benzodioxol-5-yl)-4,4-dimethyl-1-penten-3-ol is a phenylpropanoid.

Biochem/physiol Actions

Anti-convulsant drug

STIRIPENTOL Preparation Products And Raw materials

Raw materials

Preparation Products

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STIRIPENTOL Suppliers

Canada 1 China 143 Europe 2 Germany 1 India 11 Japan 1 United Kingdom 5 United States 25 Global 189

Chemleader Biomedical Co., Limited.

Tel: 021-58180488
Fax: 021-58180499
Email: sales@Medchemleader.com
Country: China
ProdList: 1005
Advantage: 58

J & K SCIENTIFIC LTD.

Tel: 010-82848833 400-666-7788
Fax: 86-10-82849933
Email: jkinfo@jkchemical.com
Country: China
ProdList: 96815
Advantage: 76

3B Pharmachem (Wuhan) International Co.,Ltd.

Tel: 821-50328103-801 18930552037
Fax: 86-21-50328109
Email: 3bsc@sina.com
Country: China
ProdList: 15839
Advantage: 69

Chembest Research Laboratories Limited

Tel: +86-21-20908456
Fax: 021-58180499
Email: sales@BioChemBest.com
Country: China
ProdList: 6005
Advantage: 61

TCI (Shanghai) Development Co., Ltd.

Tel: 021-67121386
Fax: 021-67121385
Email: Sales-CN@TCIchemicals.com
Country: China
ProdList: 24529
Advantage: 81

LGM Pharma

Tel: 1-(800)-881-8210
Fax: 615-250-9817
Email: inquiries@lgmpharma.com
Country: United States
ProdList: 2123
Advantage: 70

Chemsky（shanghai）International Co.,Ltd.

Tel: 021-50135380
Email: shchemsky@sina.com
Country: China
ProdList: 32321
Advantage: 50

China DongFan Chemical Co.,LTD

Tel: 86-0571-85151182
Fax: 86-0571-85151182
Country: China
ProdList: 5691
Advantage: 66

Hunan Hui Bai Shi Biotechnology Co., Ltd.

Tel: 0731-85526065 13308475853
Email: ivy@hnhbsj.com
Country: China
ProdList: 4552
Advantage: 62

ShangHai YuanYe Biotechnology Co., Ltd.

Tel: 021-61312847 13636370518
Fax: 021-55068248
Email: shyysw007@163.com
Country: China
ProdList: 4940
Advantage: 60

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View Lastest Price from STIRIPENTOL manufacturers

Baoji Guokang Healthchem co.,ltd

Product: STIRIPENTOL 49763-96-4
Price: US $714.30/Kg/Bag
Min. Order: 1KG
Purity: 99%
Supply Ability: 500kg
Release date: 2021-06-02

Dideu Industries Group Limited

Product: STIRIPENTOL 49763-96-4
Price: US $1.10/g
Min. Order: 1g
Purity: 99.9%
Supply Ability: 100 Tons min
Release date: 2021-08-17

Zhuozhou Wenxi import and Export Co., Ltd

Product: Stiripentol 49763-96-4
Price: US $15.00-10.00/KG
Min. Order: 1KG
Purity: 99%+ HPLC
Supply Ability: Monthly supply of 1 ton
Release date: 2021-06-26

49763-96-4, STIRIPENTOLRelated Search:

1-Penten-3-ol 4,4-Dimethyl-1-(2-methoxy-3,4-methylenedioxyphenyl)-1-penten-3-ol 3'-hydroxyisosafrole 4-phenyl-3-buten-2-ol STIRIPENTOL

Diacomit

(RS)-(E)-4,4-dimethyl-1-[3,4(methylenedioxy)-phenyl]-1-penten-3-ol

1-(1,3-BENZODIOXOL-5YL)-4,4-DIMETHYL-1-PENTEN-3-OL

STIRIPENTOL

1-(1,3-benzodioxol-5-yl)-4,4-dimethyl-1-penten-3-o

4,4-dimethyl-1-(3,4-methylenedioxyphenyl)-1-penten-3-o

4,4-dimethyl-1-(3,4-methylenedioxyphenyl)-1-penten-3-ol

bcx2600

1-(Benzo[d][1,3]dioxol-5-yl)-4,4-dimethylpent-1-en-3-ol

RCX-2600

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Stiripentol(BCX 2600)

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STIRIPENTOL USP/EP/BP

1-(1,3-benzodioxol-5-yl)-4,4-dimethylpent-1-en-3-ol

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Stiripentol, ≥ 98.0%

BCX2600|||Diacomit

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Slipperto

49763-96-4

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