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Cilliobrevin D

Product Name
Cilliobrevin D
CAS No.
1370554-01-0
Chemical Name
Cilliobrevin D
Synonyms
Cilliobrevin D;Ciliobrevin D, 10 mM in DMSO;Cytoplasmic Dynein Inhibitor, Ciliobrevin D;Benzenepropanenitrile, 2,4-dichloro-α-(7-chloro-3,4-dihydro-4-oxo-2(1H)-quinazolinylidene)-β-oxo-;2-(7-Chloro-4-oxo-3,4-dihydroquinazolin-2(1H)-ylidene)-3-(2,4-dichlorophenyl)-3-oxopropanenitrile;inhibit,melanosome,spindles,cytoplasmic,γ-tubulin,Inhibitor,dynein,ATPases,Ciliobrevin D,Hedgehog,peroxisomes,aggregation
CBNumber
CB22714664
Molecular Formula
C17H8Cl3N3O2
Formula Weight
392.62
MOL File
1370554-01-0.mol
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Cilliobrevin D Property

Boiling point:
591.8±50.0 °C(Predicted)
Density 
1.537±0.06 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
DMSO: 5 mg/mL (12.73 mM; ultrasonic and warming and heat to 80°C)
pka
5.99±0.20(Predicted)
form 
Solid
color 
Light yellow to yellow
InChI
InChI=1S/C17H8Cl3N3O2/c18-8-1-3-10(13(20)5-8)15(24)12(7-21)16-22-14-6-9(19)2-4-11(14)17(25)23-16/h1-6,22H,(H,23,25)
InChIKey
JKKSCGHDRHRWOQ-UHFFFAOYSA-N
SMILES
C(=C1NC(=O)C2=CC=C(Cl)C=C2N1)(C#N)C(C1C=CC(Cl)=CC=1Cl)=O
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
250401
Product name
Cytoplasmic Dynein Inhibitor, Ciliobrevin D
Purity
Ciliobrevin D is a cell-permeable, reversible, and specific blocker of AAA+ ATPase motor cytoplasmic dynein. Disrupts spindle pole focusing and kinetochore-microtubule attachment (~10 to 40 µM).
Packaging
10 mg
Price
$252
Updated
2025/07/31
TRC
Product number
C441315
Product name
CiliobrevinD
Packaging
25mg
Price
$1260
Updated
2021/12/16
ChemScene
Product number
CS-0087674
Product name
CiliobrevinD
Purity
98.94%
Packaging
50mg
Price
$1950
Updated
2021/12/16
ChemScene
Product number
CS-0087674
Product name
CiliobrevinD
Purity
98.94%
Packaging
5mg
Price
$350
Updated
2021/12/16
ChemScene
Product number
CS-0087674
Product name
CiliobrevinD
Purity
98.94%
Packaging
10mg
Price
$595
Updated
2021/12/16
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Cilliobrevin D Chemical Properties,Usage,Production

Uses

Ciliobrevin D is an inhibitor of the AAA+ ATPase motor cytoplasmic dynein.

in vivo

Knockdown of Dync1h1 or inactivation of dynein 1 by Ciliobrevin D in the testis in vivo perturbs spermatogenesis. Knockdown of Dync1h1 or the use of Ciliobrevin D to inactivate dynein 1 in the testis in vivo perturbs MT organization through changes in the spatial expression of EB1, perturbs F-actin organization, and perturbs distribution of adhesion protein complexes at the BTB, leading to a loss of BTB integrity. F-actin disorganization in the seminiferous epithelium following Dync1h1 knockdown or dynein 1 inactivation by Ciliobrevin D is mediated by changes in the spatiotemporal expression of actin regulatory proteins Arp3 and Eps8[3].

Cilliobrevin D Preparation Products And Raw materials

Raw materials

Preparation Products

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Cilliobrevin D Suppliers

BOC Sciences
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1-631-485-4226; 16314854226
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MedChemExpress
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1370554-01-0, Cilliobrevin DRelated Search:


  • Cilliobrevin D
  • Cytoplasmic Dynein Inhibitor, Ciliobrevin D
  • Benzenepropanenitrile, 2,4-dichloro-α-(7-chloro-3,4-dihydro-4-oxo-2(1H)-quinazolinylidene)-β-oxo-
  • inhibit,melanosome,spindles,cytoplasmic,γ-tubulin,Inhibitor,dynein,ATPases,Ciliobrevin D,Hedgehog,peroxisomes,aggregation
  • 2-(7-Chloro-4-oxo-3,4-dihydroquinazolin-2(1H)-ylidene)-3-(2,4-dichlorophenyl)-3-oxopropanenitrile
  • Ciliobrevin D, 10 mM in DMSO
  • 1370554-01-0