Mirogabalin

Product Name: Mirogabalin
CAS No.: 1138245-13-2
Chemical Name: Mirogabalin
Synonyms: Asapiprant;2-((1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)acetic acid;DS5565;A200-0700;Milobarin;mirobalin;Miluobalin;Mirogabalin;Mirogabalin HCl;DS5565;A200-0700
CBNumber: CB23051612
Molecular Formula: C12H19NO2
Formula Weight: 209.28
MOL File: 1138245-13-2.mol

More

Less

Mirogabalin Property

Boiling point:: 357.5±15.0 °C(Predicted)
Density: 1.104±0.06 g/cm3(Predicted)
storage temp.: Store at -20°C
solubility: DMF:0.5(Max Conc. mg/mL);2.39(Max Conc. mM)
Ethanol:1.25(Max Conc. mg/mL);5.97(Max Conc. mM)
PBS (pH 7.2):0.5(Max Conc. mg/mL);2.39(Max Conc. mM)
Water:5.36(Max Conc. mg/mL);25.61(Max Conc. mM)
form: A crystalline solid
pka: 4.65±0.10(Predicted)
InChI: InChI=1S/C12H19NO2/c1-2-8-3-9-5-12(7-13,6-11(14)15)10(9)4-8/h4,9-10H,2-3,5-7,13H2,1H3,(H,14,15)/t9-,10-,12-/m1/s1
InChIKey: FTBQORVNHOIASH-CKYFFXLPSA-N
SMILES: [C@]12([H])[C@]([H])([C@@](CN)(CC(O)=O)C1)C=C(CC)C2

More

Less

Hazard and Precautionary Statements (GHS)

Symbol(GHS)

Signal word

Warning

Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

More

Less

N-Bromosuccinimide Price

Cayman Chemical

Product number: 22475
Product name: Mirogabalin
Purity: ≥98%
Packaging: 1mg
Price: $68
Updated: 2024/03/01

Cayman Chemical

Product number: 22475
Product name: Mirogabalin
Purity: ≥98%
Packaging: 5mg
Price: $152
Updated: 2024/03/01

TRC

Product number: M364940
Product name: Mirogabalin
Packaging: 1mg
Price: $140
Updated: 2021/12/16

TRC

Product number: M364940
Product name: Mirogabalin
Packaging: 2.5mg
Price: $305
Updated: 2021/12/16

ChemScene

Product number: CS-6008
Product name: Mirogabalin
Purity: 99.31%
Packaging: 50mg
Price: $450
Updated: 2021/12/16

More

Less

Mirogabalin Chemical Properties,Usage,Production

Description

Mirogabalin is a calcium channel blocker with analgesic effects. It binds to the α₂δ-1 and α₂δ-2 subunits of voltage-dependent Ca²⁺ channels. Mirogabalin has potent and sustained analgesic effects (ED₅₀ = 2.5 mg/kg) in rats with diabetes induced by streptozotocin (STZ; ). Mirogabalin does not inhibit activities associated with CNS adverse effects of analgesics, such as rotarod performance (ID₅₀ = 9.4 mg/kg) or locomotor activity (ID₅₀ = 43.9 mg/kg), at its effective dose. Formulations containing mirogabalin are in clinical trials for diabetic peripheral neuropathic pain.

Uses

Mirogabalin is a two alpha2delta ligand which is investigated for the treatment of peripheral neuropathic pain, postherpetic neuralgia and fibromyalgia, showing promising results in patients with diabetic peripheral neuropathy.

Mirogabalin Preparation Products And Raw materials

Raw materials

Preparation Products

More

Less

Mirogabalin Suppliers

China 162 India 5 United States 9 Global 176

Hangzhou Kehui Pharmaceutical Co.,Ltd

Tel: 057187359773 18094707759
Email: sales10@hzkehuipharma.com
Country: China
ProdList: 17
Advantage: 58

Nanjing Tianhai Pharmaceutical Technology Co., Ltd.

Tel: 025-58351158 13851454004
Fax: 025-83271564
Email: 3494688757@qq.com
Country: China
ProdList: 116
Advantage: 58

Nanjing Becas pharmatech Ltd.

Tel: 13912903754
Email: info@becaspharma.com
Country: China
ProdList: 2257
Advantage: 58

Nanajing Chenruisheng Biomedical Technology Ltd

Tel: 18805148037
Email: 1277392432@qq.com
Country: China
ProdList: 151
Advantage: 58

Anhui Cheer-Our Medical technology Co.,Ltd

Tel: 13855402841
Email: nicole@cheer-our.com
Country: China
ProdList: 93
Advantage: 58

NANJING ZENJI PHARMACEUTICALS

Tel: 025-58231105-8151
Email: marketing@zenjipharma.com
Country: China
ProdList: 505
Advantage: 58

NANJING ZENJI PHARMACEUTICALS

Tel: 025-58231105-8151
Fax: 025-83172562
Email: marketing@zenjipharma.com
Country: China
ProdList: 237
Advantage: 58

Hangzhou Chemtrue Bio-Tech Co.,Ltd.

Tel: 0571-86828652 18857119830
Fax: 0571-83522824
Email: sales@chemtrue-bio.com
Country: China
ProdList: 314
Advantage: 58

Shandong Xuanshuo Pharmaceutical Technology Co. LTD

Tel: 13335135755
Email: suchangzhou@shiningpharm.com
Country: China
ProdList: 204
Advantage: 58

BeiJing Hwrk Chemicals Limted

Tel: 0757-86329057 18501085097
Fax: 010-89508210
Email: sales3.gd@hwrkchemical.com
Country: China
ProdList: 7639
Advantage: 55

More

Less

View Lastest Price from Mirogabalin manufacturers

ShenZhen H&D Pharmaceutical Technology Co., LTD

Product: Mirogabalin 1138245-13-2
Price: US $0.00-0.00/mg
Min. Order: 10mg
Purity: 0.98
Supply Ability: 10g
Release date: 2024-04-07

Hebei Yanxi Chemical Co., Ltd.

Product: Mirogabalin 1138245-13-2
Price: US $0.00-0.00/kg
Min. Order: 1kg
Purity: 99%
Supply Ability: 100tons
Release date: 2023-08-16

1138245-13-2, MirogabalinRelated Search:

2-((1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)acetic acid

Mirogabalin

Asapiprant

[(1R,5S,6S)-6-(Aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid

A200-0700

DS5565

DS5565;A200-0700

2-[(1R,5S,6S)-6-(aminomethyl)-3-ethyl-6-bicyclo[3.2.0]hept-3-enyl]acetic acid

MIROGABALIN; DS-5565

DS 5565;DS-5565;DS5565

Bicyclo[3.2.0]hept-3-ene-6-acetic acid, 6-(aminomethyl)-3-ethyl-, (1R,5S,6S)-

Miluobalin

Mirogabalin HCl

Milobarin

Mirogabalin Impurity

mirobalin

Mirogabalin free base

1138245-13-2

API

1138245-13-2