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Tadalafil-d3

Product Name
Tadalafil-d3
CAS No.
960226-55-5
Chemical Name
Tadalafil-d3
Synonyms
Tadalafil-d3;[2H3]-Tadalafil;PubChem ID: 46782966;Pyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4-dione, 6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydro-2-(methyl-d3)-, (6R,12aR)-;(2R,8R)-2-(2H-1,3-benzodioxol-5-yl)-6-(2H?)methyl-3,6,17-triazatetracyclo[8.7.0.03,?.011,1?]heptadeca-1(10),11(16),12,14-tetraene-4,7-dione;Tadalafil D3Q: What is Tadalafil D3 Q: What is the CAS Number of Tadalafil D3 Q: What is the storage condition of Tadalafil D3 Q: What are the applications of Tadalafil D3
CBNumber
CB32104260
Molecular Formula
C22H18N3O4
Formula Weight
388.39602
MOL File
960226-55-5.mol
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Tadalafil-d3 Property

Melting point:
281-283°C
storage temp. 
-20°C Freezer
solubility 
Chloroform (Slightly), DMSO (Slightly)
form 
Solid
color 
White to Off-White
Stability:
Unstable in Methanol
InChI
InChI=1/C22H19N3O4/c1-24-10-19(26)25-16(22(24)27)9-14-13-4-2-3-5-15(13)23-20(14)21(25)12-6-7-17-18(8-12)29-11-28-17/h2-8,16,21,23H,9-11H2,1H3/t16-,21+/s3
InChIKey
WOXKDUGGOYFFRN-PDIFIXMTNA-N
SMILES
c12c3ccccc3nc1[C@H](c1cc3OCOc3cc1)N1C(=O)CN(C)C(=O)[C@H]1C2 |&1:9,27,r|
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P271Use only outdoors or in a well-ventilated area.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P304+P340IF INHALED: Remove victim to fresh air and Keep at rest in a position comfortable for breathing.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

P312Call a POISON CENTER or doctor/physician if you feel unwell.

P321Specific treatment (see … on this label).

P332+P313IF SKIN irritation occurs: Get medical advice/attention.

P337+P313IF eye irritation persists: Get medical advice/attention.

P403+P233Store in a well-ventilated place. Keep container tightly closed.

P405Store locked up.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

Cayman Chemical
Product number
25030
Product name
Tadalafil-d3
Purity
≥99% deuterated forms (d1-d3)
Packaging
1mg
Price
$178
Updated
2024/03/01
Cayman Chemical
Product number
25030
Product name
Tadalafil-d3
Purity
≥99% deuterated forms (d1-d3)
Packaging
5mg
Price
$704
Updated
2024/03/01
TRC
Product number
T004510
Product name
Tadalafil-d3
Packaging
10mg
Price
$1390
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
RDL0005317
Product name
TADALAFIL-D3
Purity
95.00%
Packaging
10MG
Price
$1963.5
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
RDL0005317
Product name
TADALAFIL-D3
Purity
95.00%
Packaging
1MG
Price
$750.75
Updated
2021/12/16
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Tadalafil-d3 Chemical Properties,Usage,Production

Description

Tadalafil-d3 is intended for use as an internal standard for the quantification of tadalafil by GC- or LC-MS. Tadalafil is a potent inhibitor of phosphodiesterase 5 (PDE5; IC50 = 1.2 nM). It is selective for PDE5 over PDE1-4 and 7-10 (IC50s = 9.2-280 μM), however, it does also inhibit PDE11 (IC50 = 11 nM). In vivo, tadalafil (10 mg/kg) decreases production of the proinflammatory cytokines TNF-α, IL-1β, and IL-6 and improves renal function in a rat model of ischemia/reperfusion injury. It also reduces development of tobacco smoke-induced emphysema and pulmonary hypertension in mice. Formulations containing tadalafil have been used to treat erectile dysfunction, pulmonary arterial hypertension, and lower urinary tract dysfunction.

Chemical Properties

Tadalafil-d3 is White Solid

Uses

Tadalafil-d3 is used for the treatment of erectile dysfunction. A phosphodiesterase 5 inhibitor. Intended for use as an internal standard for the quantification of Tadalafil by GC- or LC-mass spectrometry.

Uses

Tadalafil is used for the treatment of erectile dysfunction. A phosphodiesterase 5 inhibitor.

Tadalafil-d3 Preparation Products And Raw materials

Raw materials

Preparation Products

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Tadalafil-d3 Suppliers

J & K SCIENTIFIC LTD.
Tel
010-82848833 400-666-7788
Fax
86-10-82849933
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jkinfo@jkchemical.com
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China
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94657
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Chemsky(shanghai)International Co.,Ltd.
Tel
021-50135380
Email
shchemsky@sina.com
Country
China
ProdList
32321
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50
Daicel Chiral Technologies (China)CO.,LTD
Tel
021-50460086-9 15921403865
Fax
+86-21-50462321
Email
han_yajun@dctc.daicel.com
Country
China
ProdList
7195
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Cato Research Chemicals Inc.
Tel
020-81960175
Fax
+1-541-2553641
Email
min.he@cato-chem.com
Country
China
ProdList
1955
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ChemStrong Scientific Co.,Ltd
Tel
0755-0755-66853366 13670046396
Fax
0755-28363542
Email
sales@chem-strong.com
Country
China
ProdList
18070
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Artis Biotech Co. Ltd.
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0575-18780151478 18582380095
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0575-89298961
Email
sales@artisbio.com
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China
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Clearsynth Canada Inc.
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+1.415.685.4395
Fax
+1.415.685.4395
Email
enquiry@clearsynth.com
Country
Canada
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912
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Shanghai Champ Biopharmaceuticals Co., Ltd.
Tel
021-61537865 13585780846
Email
sales@champchem.com
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China
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360
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Shenzhen SUNGENING Bio-Medical Co., Ltd.
Tel
0755-28967200 13631290199
Fax
0755-28967200
Email
wxf@sungening.com
Country
China
ProdList
9578
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Nanjing Haolv Biotechnology Co.,Ltd
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025-84622273 17361806303
Email
3004208264@qq.com
Country
China
ProdList
3021
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58

960226-55-5, Tadalafil-d3Related Search:


  • Tadalafil-d3
  • Pyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4-dione, 6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydro-2-(methyl-d3)-, (6R,12aR)-
  • PubChem ID: 46782966
  • [2H3]-Tadalafil
  • Tadalafil D3Q: What is Tadalafil D3 Q: What is the CAS Number of Tadalafil D3 Q: What is the storage condition of Tadalafil D3 Q: What are the applications of Tadalafil D3
  • (2R,8R)-2-(2H-1,3-benzodioxol-5-yl)-6-(2H?)methyl-3,6,17-triazatetracyclo[8.7.0.03,?.011,1?]heptadeca-1(10),11(16),12,14-tetraene-4,7-dione
  • 960226-55-5
  • C22H16N3O4D3
  • Chiral Reagents
  • Inhibitors
  • Intermediates & Fine Chemicals
  • Isotope Labelled Compounds
  • Pharmaceuticals
  • Intermediates & Fine Chemicals,Chiral Reagents