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GUANABENZ

Product Name
GUANABENZ
CAS No.
5051-62-7
Chemical Name
GUANABENZ
Synonyms
Rexitene;GUANABENZ;nsc-68982;Callosum benzyl;GUANABENZ USP/EP/BP;Guanabenz (WY 8678);1-(2,6-DICHLOROBENZYLIDENEAMINO)GUANIDINE;n-(2,6-dichlorobenzylidene)amino]guanidine;n-(2,6-dichlorobenzylidene)-n’-amidinohydrazine;2-(2,6-Dichlorobenzylidene)hydrazine-1-carboximidamide
CBNumber
CB3263851
Molecular Formula
C8H8Cl2N4
Formula Weight
231.08
MOL File
5051-62-7.mol
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GUANABENZ Property

Melting point:
227-229° (dec)
Boiling point:
353.9±52.0 °C(Predicted)
Density 
1.49±0.1 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
DMSO: 12 mg/mL (51.93 mM);Ethanol: 15 mg/mL (64.91 mM)
pka
pKa 8.1 (Uncertain)
Water Solubility 
Water: Insoluble
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Safety

Hazard Codes 
Xn
Risk Statements 
20/21/22-62
Safety Statements 
22-36/37/39
RIDADR 
3249
WGK Germany 
3
HazardClass 
6.1(b)
PackingGroup 
III
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

H312Harmful in contact with skin

H332Harmful if inhaled

H361Suspected of damaging fertility or the unborn child

Precautionary statements

P201Obtain special instructions before use.

P202Do not handle until all safety precautions have been read and understood.

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P271Use only outdoors or in a well-ventilated area.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P281Use personal protective equipment as required.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P304+P340IF INHALED: Remove victim to fresh air and Keep at rest in a position comfortable for breathing.

P308+P313IF exposed or concerned: Get medical advice/attention.

P312Call a POISON CENTER or doctor/physician if you feel unwell.

P322Specific measures (see …on this label).

P330Rinse mouth.

P363Wash contaminated clothing before reuse.

P405Store locked up.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
S762091
Product name
N-(2,6-DICHLOROBENZYLIDENEAMINO)GUANIDINE
Purity
Aldrich
Packaging
50mg
Price
$179
Updated
2024/03/01
American Custom Chemicals Corporation
Product number
API0006231
Product name
GUANABENZ
Purity
95.00%
Packaging
5MG
Price
$502.68
Updated
2021/12/16
Medical Isotopes, Inc.
Product number
75138
Product name
Guanabenz
Packaging
5mg
Price
$1545
Updated
2021/12/16
CSNpharm
Product number
CSN23785
Product name
GUANABENZ
Packaging
100mg
Price
$237
Updated
2021/12/16
AHH
Product number
MT-08425
Product name
1-(2,6-Dichlorobenzylideneamino)guanidine
Purity
98%
Packaging
0.1g
Price
$306
Updated
2021/12/16
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GUANABENZ Chemical Properties,Usage,Production

Description

Guanabenz is an α2-adrenergic agonist that exhibits pronounced hypotensive action, and that is associated with a reduction of overall peripheral vascular resistance, decline in frequency of cardiac contractions, and reduced cardiac output.

Originator

Wytensin,Wyeth,US,1982

Uses

alpha agonists

Uses

It is used both independently and in combination with oral diuretics for treating various degrees of hypertension.

Definition

ChEBI: Guanabenz is a dichlorobenzene.

Manufacturing Process

A mixture of 14.0 g of 2,6-dichlorobenzaldehyde, 10.8 g of aminoguanidine bicarbonate and 100 ml of pyridine was refluxed for 3 hours. The reaction mixture was poured into water and the crystalline precipitate filtered off; MP 225°C to 227°C.

Therapeutic Function

Antihypertensive

Synthesis

Guanabenz, [(2,6-dichlorobenzyliden) amino] guanidine (22.3.1), is synthesized in one step by reacting 2,6-dichlorobenzaldehyde with amino guanidine.

Purification Methods

Crystallise the guanidine from MeCN and store it in a CO2–free atmosphere. The monoHCl [23256-5-0] has m 178o(dec) [solubility w% at 25o is 1.1(H2O), 5(EtOH), 0.1(EtOAc), 0.06(CHCl3)]. It is an antihypertensive drug. [Holmes et al. Drugs 26 212 1983.]

GUANABENZ Preparation Products And Raw materials

Raw materials

Preparation Products

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GUANABENZ Suppliers

Guangdong Qianjin Chemical Reagent Co., Ltd.
Tel
0751-2818792 13435114148
Email
3128240096@qq.com
Country
China
ProdList
2994
Advantage
58
LGM Pharma
Tel
1-(800)-881-8210
Fax
615-250-9817
Email
inquiries@lgmpharma.com
Country
United States
ProdList
2123
Advantage
70
Hangzhou Sage Chemical Co., Ltd.
Tel
+86057186818502 13588463833
Fax
Pls mail us for more information!
Email
info@sagechem.com
Country
China
ProdList
10266
Advantage
58
Beijing HuaMeiHuLiBiological Chemical
Tel
010-56205725
Fax
010-65763397
Email
waley188@sohu.com
Country
China
ProdList
12335
Advantage
58
Shanghai TaoSu Biochemical Technology Co., Ltd.
Tel
021-33632979
Fax
021-34692979
Email
info@tsbiochem.com
Country
China
ProdList
8065
Advantage
58
ShangHai Caerulum Pharma Discovery Co., Ltd.
Tel
18149758185 18149758185
Email
sales-cpd@caerulumpharma.com
Country
China
ProdList
3466
Advantage
58
Finetech Industry Limited
Tel
027-87465837 19945049750
Fax
027-8777-2287
Email
sales@finetechnology-ind.com
Country
China
ProdList
9648
Advantage
58
Shanghai HuanChuan Industry Co.,Ltd.
Tel
021-61478794
Fax
021-61478794
Email
sales@hcshhai.com
Country
China
ProdList
9793
Advantage
50
Shanghai JiYi Biotechnology Co. Ltd.
Tel
13621943973
Fax
-
Email
sales@shjiyipharmatech.com
Country
China
ProdList
1166
Advantage
55
ShangHai Biochempartner Co.,Ltd
Tel
177-54423994 17754423994
Fax
QQ:2853530913
Email
2853530910@QQ.com
Country
China
ProdList
8010
Advantage
62
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View Lastest Price from GUANABENZ manufacturers

Dideu Industries Group Limited
Product
GUANABENZ 5051-62-7
Price
US $1.10/g
Min. Order
1g
Purity
99.9%
Supply Ability
100 Tons min
Release date
2021-08-10
Shaanxi Dideu Medichem Co. Ltd
Product
Guanabenz 5051-62-7
Price
US $0.00-0.00/Kg
Min. Order
1KG
Purity
99.0%
Supply Ability
500 MT
Release date
2020-05-09

5051-62-7, GUANABENZRelated Search:


  • GUANABENZ
  • 2-[(2,6-dichlorophenyl)methylene]-hydrazinecarboximidamide
  • n-(2,6-dichlorobenzylidene)amino]guanidine
  • n-(2,6-dichlorobenzylidene)-n’-amidinohydrazine
  • nsc-68982
  • Rexitene
  • HydrazinecarboxiMidaMide, 2-[(2,6-dichlorophenyl)Methylene]-
  • 1-(2,6-DICHLOROBENZYLIDENEAMINO)GUANIDINE
  • 2-(2,6-Dichlorobenzylidene)hydrazine-1-carboximidamide
  • Guanabenz (WY 8678)
  • GUANABENZ USP/EP/BP
  • Callosum benzyl
  • GUANABENZ,inhibit,Adrenergic Receptor,high blood pressure,Beta Receptor,antiparasitic,Inhibitor,antihypertensive,Parasite
  • 5051-62-7
  • C8H8Cl2N4
  • Analytical Standards
  • Analytical Chromatography Product Catalog
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