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MRS 2279

Product Name
MRS 2279
CAS No.
367909-40-8
Chemical Name
MRS 2279
Synonyms
MRS 2279;MRS2279,MRS-2279;MRS 2279, CID: 5311301;[(1S,2R,4R)-4-[(2-chloro-6-methylaminopurin-9-yl)methyl]-2-(phosphonooxymethyl)cyclopentyl] dihydrogen phosphate;Bicyclo[3.1.0]hexane-1-methanol, 4-[2-chloro-6-(methylamino)-9H-purin-9-yl]-2-(phosphonooxy)-, 1-(dihydrogen phosphate), (1R,2S,4S,5S)-;(1R*,2S*)-4-[2-Chloro-6-(methylamino)-9H-purin-9-yl]-2-(phosphonooxy)bicyclo[3.1.0]hexane-1-methanoldihydrogenphosphateesterdiammoniumsalt
CBNumber
CB3848748
Molecular Formula
C13H18ClN5O8P2
Formula Weight
469.71
MOL File
367909-40-8.mol
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MRS 2279 Property

storage temp. 
Desiccate at -20°C
form 
Powder
Water Solubility 
Soluble to 100 mM in water
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Tocris
Product number
2158
Product name
MRS2279
Purity
≥98%(HPLC)
Packaging
1
Price
$400
Updated
2021/12/16
TRC
Product number
M750250
Product name
MRS2279
Packaging
1mg
Price
$355
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
BRS0000600
Product name
MRS-2279
Purity
95.00%
Packaging
5MG
Price
$500.42
Updated
2021/12/16
ApexBio Technology
Product number
B5265
Product name
MRS2279
Packaging
1mg
Price
$581
Updated
2021/12/16
ChemScene
Product number
CS-0029414
Product name
MRS2279
Packaging
1mg
Price
$880
Updated
2021/12/16
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MRS 2279 Chemical Properties,Usage,Production

Uses

MRS 2279 is a selective P2Y1 antagonist with high affinity and results in modulation of aggregation of blood platelets induced by ADP.

Biological Activity

Selective, high affinity competitive antagonist of the P2Y 1 receptor (K i = 2.5 nM; IC 50 = 51.6 nM). Fails to block nucleotide signaling at most other P2Y receptors (P2Y 2 , P2Y 4 , P2Y 6 , P2Y 11 and P2Y 12 ) and potently inhibits ADP-induced aggregation of human blood platelets in vitro (pK B = 8.05).

MRS 2279 Preparation Products And Raw materials

Raw materials

Preparation Products

367909-40-8, MRS 2279Related Search:


  • MRS 2279
  • [(1S,2R,4R)-4-[(2-chloro-6-methylaminopurin-9-yl)methyl]-2-(phosphonooxymethyl)cyclopentyl] dihydrogen phosphate
  • MRS 2279, CID: 5311301
  • (1R*,2S*)-4-[2-Chloro-6-(methylamino)-9H-purin-9-yl]-2-(phosphonooxy)bicyclo[3.1.0]hexane-1-methanoldihydrogenphosphateesterdiammoniumsalt
  • Bicyclo[3.1.0]hexane-1-methanol, 4-[2-chloro-6-(methylamino)-9H-purin-9-yl]-2-(phosphonooxy)-, 1-(dihydrogen phosphate), (1R,2S,4S,5S)-
  • MRS2279,MRS-2279
  • 367909-40-8
  • C13H18ClN5O8P22NH3
  • C13H18ClN5O8P2