ChemicalBook > CAS DataBase List > MK-4827 (R-enantioMer)

MK-4827 (R-enantioMer)

Product Name
MK-4827 (R-enantioMer)
CAS No.
1038915-58-0
Chemical Name
MK-4827 (R-enantioMer)
Synonyms
(R)-Niraparib;ent-Niraparib;ent-Nirapanib;Niraparib Impurity;Niraparib Impurity 13;Niraparib Impurity 51;MK-4827 (R-enantioMer);Niraparib R-enantiomer;R isomer of MK-4827, Niraparib;(R)-2-(4-(PIPERIDIN-3-YL)PHENYL)-2H-INDAZOLE-7-CARBOXAMIDE
CBNumber
CB42716288
Molecular Formula
C19H20N4O
Formula Weight
320.39
MOL File
1038915-58-0.mol
More
Less

MK-4827 (R-enantioMer) Property

Boiling point:
463.6±45.0 °C(Predicted)
Density 
1.34±0.1 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
DMSO : ≥ 32 mg/mL (99.88 mM)
pka
15.36±0.30(Predicted)
form 
Solid
color 
Light yellow to yellow
More
Less

Hazard and Precautionary Statements (GHS)

More
Less

N-Bromosuccinimide Price

TRC
Product number
N481410
Product name
ent-Niraparib
Packaging
500mg
Price
$2230
Updated
2021/12/16
ChemScene
Product number
CS-3085
Product name
NiraparibR-enantiomer
Purity
99.50%
Packaging
5mg
Price
$220
Updated
2021/12/16
ChemScene
Product number
CS-3085
Product name
NiraparibR-enantiomer
Purity
99.50%
Packaging
10mg
Price
$380
Updated
2021/12/16
ChemScene
Product number
CS-3085
Product name
NiraparibR-enantiomer
Purity
99.50%
Packaging
50mg
Price
$990
Updated
2021/12/16
Crysdot
Product number
CD00013477
Product name
(R)-2-(4-(Piperidin-3-yl)phenyl)-2H-indazole-7-carboxamide
Purity
97%
Packaging
1g
Price
$3294
Updated
2021/12/16
More
Less

MK-4827 (R-enantioMer) Chemical Properties,Usage,Production

Uses

ent-Niraparib is an isomer of Niraparib (N481400), a novel oral poly(ADP-ribose)polymerase (PARP) inhibitor efficacious in BRCA-1 and -2 mutant tumors.

Definition

ChEBI: 2-{4-[(3R)-piperidin-3-yl]phenyl}-2H-indazole-7-carboxamide is a 2-[4-(piperidin-3-yl)phenyl]-2H-indazole-7-carboxamide that has R-configuration. It is a potent PARP1 inhibitor with IC50 of 2.4 nM. It has a role as an EC 2.4.2.30 (NAD(+) ADP-ribosyltransferase) inhibitor and an antineoplastic agent.

MK-4827 (R-enantioMer) Preparation Products And Raw materials

Raw materials

Preparation Products

More
Less

MK-4827 (R-enantioMer) Suppliers

Pharmaffiliates Analytics and Synthetics P. Ltd
Tel
--
Fax
--
Email
mktg@pharmaffiliates.com
Country
India
ProdList
6739
Advantage
58
More
Less

View Lastest Price from MK-4827 (R-enantioMer) manufacturers

ShenZhen H&D Pharmaceutical Technology Co., LTD
Product
(R)-Niraparib 1038915-58-0
Price
US $0.00-0.00/mg
Min. Order
10mg
Purity
0.98
Supply Ability
10g
Release date
2024-05-07

1038915-58-0, MK-4827 (R-enantioMer)Related Search:


  • MK-4827 (R-enantioMer)
  • Niraparib Impurity
  • R isomer of MK-4827, Niraparib
  • (R)-2-(4-(PIPERIDIN-3-YL)PHENYL)-2H-INDAZOLE-7-CARBOXAMIDE
  • Niraparib R-enantiomer
  • 2-{4-[(3S)-piperidin-3-yl]phenyl}-2H-indazole-7-carboxamide
  • ent-Niraparib
  • 2H-Indazole-7-carboxamide, 2-[4-(3R)-3-piperidinylphenyl]-
  • poly ADP ribose polymerase,Inhibitor,Niraparib (R enantiomer),PARP,Niraparib (Renantiomer),Niraparib (R-enantiomer),inhibit
  • (R)-Niraparib
  • Niraparib Impurity 13
  • ent-Nirapanib
  • Niraparib Impurity 51
  • 1038915-58-0