1-Boc-5-aminoindole

Product Name: 1-Boc-5-aminoindole
CAS No.: 166104-20-7
Chemical Name: 1-Boc-5-aminoindole
Synonyms: N-Boc-5-Aminoindole;5-AMINOINDOLE-1-BOC;1-BOC-5-AMINOINDOLE;5-Amino-1-Boc-indole;1-BOC-5-AMINOINDOLE, 98+%;5-AMINO-1-BOC-BENZIMIDAZOLE;5-AMINO-1-BOC-BENZOIMIDAZOLE;5-Aminoindole, N1-BOC protected;5-Amino-1H-indole, N1-BOC protected;tert-butyl 5-aminoindole-1-carboxylate
CBNumber: CB4400660
Molecular Formula: C13H16N2O2
Formula Weight: 232.28
MOL File: 166104-20-7.mol

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1-Boc-5-aminoindole Property

Boiling point:: 384.2±34.0 °C(Predicted)
Density: 1.16±0.1 g/cm3(Predicted)
storage temp.: under inert gas (nitrogen or Argon) at 2–8 °C
pka: 4.28±0.10(Predicted)
form: low melting solid
color: Brown
CAS DataBase Reference: 166104-20-7(CAS DataBase Reference)

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Safety

HS Code: 2933998090

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Hazard and Precautionary Statements (GHS)

Symbol(GHS)

Signal word

Warning

Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

Biosynth Carbosynth

Product number: FB51012
Product name: 1-Boc-5-aminoindole
Packaging: 500mg
Price: $95
Updated: 2021/12/16

Matrix Scientific

Product number: 072083
Product name: 1-Boc-5-Aminoindole
Purity: 95+%
Packaging: 1g
Price: $163
Updated: 2021/12/16

AK Scientific

Product number: N061
Product name: 1-Boc-5-Aminoindole
Packaging: 5g
Price: $195
Updated: 2021/12/16

Biosynth Carbosynth

Product number: FB51012
Product name: 1-Boc-5-aminoindole
Packaging: 1g
Price: $197.7
Updated: 2021/12/16

SynQuest Laboratories

Product number: 4H51-1-66
Product name: 5-Amino-1H-indole, N1-Boc protected
Packaging: 1g
Price: $216
Updated: 2021/12/16

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1-Boc-5-aminoindole Chemical Properties,Usage,Production

Synthesis

166104-19-4

166104-20-7

General procedure for the synthesis of N-Boc-5-aminoindole from tert-butyl 5-nitro-1H-indole-1-carboxylate: tert-butyl 5-nitro-1H-indole-1-carboxylate (525 mg, 2.0 mmol) was dissolved in ethyl acetate (8 mL), and 10% palladium-carbon-catalyst (50 mg) was added. The reaction mixture was stirred overnight at room temperature in a hydrogen atmosphere. Upon completion of the reaction, the catalyst was removed by suction filtration and the filtrate was concentrated under reduced pressure to afford the white solid product N-Boc-5-aminoindole (469 mg, 100% yield).

References

[1] Patent: CN104311541, 2017, B. Location in patent: Paragraph 0164; 0165
[2] Patent: US2009/247568, 2009, A1. Location in patent: Page/Page column 36
[3] Journal of Medicinal Chemistry, 2013, vol. 56, # 15, p. 6273 - 6277
[4] Synthetic Communications, 2006, vol. 36, # 14, p. 2069 - 2077
[5] Journal of Medicinal Chemistry, 2011, vol. 54, # 4, p. 1106 - 1110

1-Boc-5-aminoindole Preparation Products And Raw materials

Raw materials

Preparation Products

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1-Boc-5-aminoindole Suppliers

China 116 Germany 2 India 1 United Kingdom 6 United States 24 Global 149

Capot Chemical Co., Ltd

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T&W GROUP

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View Lastest Price from 1-Boc-5-aminoindole manufacturers

Honest Joy Holdings Limited

Product: 1-Boc-5-aminoindole 166104-20-7
Price: US $0.00/KG
Min. Order: 1KG
Purity: 98.7%
Supply Ability: 100 tons
Release date: 2022-02-08

Career Henan Chemical Co

Product: 1-Boc-5-aminoindole 166104-20-7
Price: US $1.00/KG
Min. Order: 1KG
Purity: 99%
Supply Ability: 1kg-1000kg
Release date: 2020-01-02

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1-BOC-5-AMINOINDOLE

5-AMINOINDOLE-1-BOC

N-Boc-5-Aminoindole

tert-butyl 5-amino-1H-indole-1-carboxylate

5-Aminoindole, N1-BOC protected

1-BOC-5-AMINOINDOLE, 98+%

5-Amino-1-Boc-indole

5-amino-1-indolecarboxylic acid tert-butyl ester

5-Amino-1H-indole, N1-BOC protected

1H-Indole-1-carboxylic acid, 5-amino-, 1,1-dimethylethyl ester

tert-butyl 5-aminoindole-1-carboxylate

166104-20-7

15862

pharmacetical