ChemicalBook > CAS DataBase List > 4-(5-ETHOXY-3-PYRIDINYL)-N-METHYL-(3E)-3-BUTEN-1-AMINE DIFUMARATE

4-(5-ETHOXY-3-PYRIDINYL)-N-METHYL-(3E)-3-BUTEN-1-AMINE DIFUMARATE

Product Name
4-(5-ETHOXY-3-PYRIDINYL)-N-METHYL-(3E)-3-BUTEN-1-AMINE DIFUMARATE
CAS No.
212332-35-9
Chemical Name
4-(5-ETHOXY-3-PYRIDINYL)-N-METHYL-(3E)-3-BUTEN-1-AMINE DIFUMARATE
Synonyms
TC 2559 (fumarate);TC 2559 DIFUMARATE;4-(5-ETHOXY-3-PYRIDINYL)-N-METHYL-(3E)-3-BUTEN-1-AMINE DIFUMARATE
CBNumber
CB52453441
Molecular Formula
C20H26N2O9
Formula Weight
0
MOL File
212332-35-9.mol
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4-(5-ETHOXY-3-PYRIDINYL)-N-METHYL-(3E)-3-BUTEN-1-AMINE DIFUMARATE Property

Melting point:
123-125°C
storage temp. 
Desiccate at RT
solubility 
DMSO (Slightly), Methanol (Slightly)
form 
Solid
color 
White to Off-White
Water Solubility 
Soluble to 100 mM in water
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Cayman Chemical
Product number
25600
Product name
TC 2559 (fumarate)
Packaging
1mg
Price
$32
Updated
2024/03/01
Cayman Chemical
Product number
25600
Product name
TC 2559 (fumarate)
Packaging
25mg
Price
$533
Updated
2024/03/01
Cayman Chemical
Product number
25600
Product name
TC 2559 (fumarate)
Packaging
5mg
Price
$139
Updated
2024/03/01
Cayman Chemical
Product number
25600
Product name
TC 2559 (fumarate)
Packaging
10mg
Price
$230
Updated
2024/03/01
Tocris
Product number
2737
Product name
TC2559difumarate
Purity
≥98%(HPLC)
Packaging
10
Price
$217
Updated
2021/12/16
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4-(5-ETHOXY-3-PYRIDINYL)-N-METHYL-(3E)-3-BUTEN-1-AMINE DIFUMARATE Chemical Properties,Usage,Production

Uses

TC 2559 Fumarate is a partial agonist for AChR α4β2.

Biological Activity

Subtype-selective partial agonist for α 4 β 2 nicotinic acetylcholine receptors (EC 50 values are 0.18, 12.5, 14.0, > 30, > 100 and > 100 μ M for α 4 β 2, α 4 β 4, α 2 β 4, α 3 β 4, α 3 β 2 and α 7 receptor subtypes respectively). Displays selectivity for ( α 4) 2 ( β 2) 3 receptor stoichiometry and enhanced CNS-PNS selectivity ratio. Attenuates scopolamine-induced cognitive deficits in a step-through passive avoidance task.

4-(5-ETHOXY-3-PYRIDINYL)-N-METHYL-(3E)-3-BUTEN-1-AMINE DIFUMARATE Preparation Products And Raw materials

Raw materials

Preparation Products

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4-(5-ETHOXY-3-PYRIDINYL)-N-METHYL-(3E)-3-BUTEN-1-AMINE DIFUMARATE Suppliers

212332-35-9, 4-(5-ETHOXY-3-PYRIDINYL)-N-METHYL-(3E)-3-BUTEN-1-AMINE DIFUMARATERelated Search:


  • 4-(5-ETHOXY-3-PYRIDINYL)-N-METHYL-(3E)-3-BUTEN-1-AMINE DIFUMARATE
  • TC 2559 DIFUMARATE
  • TC 2559 (fumarate)
  • 212332-35-9
  • C20H26N2O9
  • C12H18N2O2C4H4O4