ChemicalBook > CAS DataBase List > 5-(2-BENZOTHIAZOLYL)-3-ETHYL-2-(-(METHY

5-(2-BENZOTHIAZOLYL)-3-ETHYL-2-(-(METHY

Product Name
5-(2-BENZOTHIAZOLYL)-3-ETHYL-2-(-(METHY
CAS No.
681281-88-9
Chemical Name
5-(2-BENZOTHIAZOLYL)-3-ETHYL-2-(-(METHY
Synonyms
5-(2-BENZOTHIAZOLYL)-3-ETHYL-2-(-(METHY;Akt Inhibitor IV - CAS 681281-88-9 - Calbiochem;6-(2-Benzothiazolyl)-1-ethyl-2-[2-(methylphenylamino)ethenyl]-3-phenyl-1H-benzimidazolium iodide;6-benzothiazol-2-yl-1-ethyl-2-[2-(methyl-phenyl-amino)-vinyl]-3-phenyl-3H-benzoimidazol-1-ium iodide;5-(Benzo[d]thiazol-2-yl)-3-ethyl-2-(2-(methyl(phenyl)amino)vinyl)-1-phenyl-1H-benzo[d]imidazol-3-ium iodide;(E)-5-(benzo[d]thiazol-2-yl)-3-ethyl-2-(2-(methyl(phenyl)amino)vinyl)-1-phenyl-1H-benzo[d]imidazol-3-ium iodide
CBNumber
CB5497911
Molecular Formula
C31H27N4S.I
Formula Weight
614.548
MOL File
681281-88-9.mol
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5-(2-BENZOTHIAZOLYL)-3-ETHYL-2-(-(METHY Property

storage temp. 
2-8°C
solubility 
DMSO: ≥10 mg/mL
form 
solid
color 
orange
InChIKey
NAYRELMNTQSBIN-UHFFFAOYSA-M
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Safety

Hazard Codes 
Xi
Risk Statements 
36/37/38
Safety Statements 
26-36
WGK Germany 
3
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

P321Specific treatment (see … on this label).

P332+P313IF SKIN irritation occurs: Get medical advice/attention.

P362Take off contaminated clothing and wash before reuse.

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
124011
Product name
Akt Inhibitor IV
Packaging
1mg
Price
$172
Updated
2024/03/01
Sigma-Aldrich
Product number
124011
Product name
Akt Inhibitor IV
Packaging
5mg
Price
$619
Updated
2024/03/01
Cayman Chemical
Product number
15569
Product name
Akt Inhibitor IV
Purity
≥95%
Packaging
1mg
Price
$40
Updated
2024/03/01
Cayman Chemical
Product number
15569
Product name
Akt Inhibitor IV
Purity
≥95%
Packaging
5mg
Price
$177
Updated
2024/03/01
Sigma-Aldrich
Product number
B2311
Product name
5-(2-Benzothiazolyl)-3-ethyl-2-[2-(methylphenylamino)ethenyl]-1-phenyl-1H-benzimidazolium iodide
Purity
≥98% (HPLC)
Packaging
5mg
Price
$205
Updated
2024/03/01
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5-(2-BENZOTHIAZOLYL)-3-ETHYL-2-(-(METHY Chemical Properties,Usage,Production

Uses

Akt Inhibitor IV is an Inhibitor of Akt protein kinase

Biological Activity

akt inhibitor iv is an inhibitor of akt activation that inhibits akt-mediated nuclear export of forkhead box class o transcription factor 1a (foxo1a; ic50 = 625 nm) and reduces phosphorylation of akt at ser473 and thr308 in a dose-dependent manner. akt inhibitor iv inhibits replication of parainfluenza virus 5 (piv5) in hela cells (ic50 = 520 nm). it also reduces the growth of cancer cells (ic50 = 0.3 μm for both jurkat and hela cells) via a reduction in mitochondrial polarization and increased production of reactive oxygen species (ros).

5-(2-BENZOTHIAZOLYL)-3-ETHYL-2-(-(METHY Preparation Products And Raw materials

Raw materials

Preparation Products

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5-(2-BENZOTHIAZOLYL)-3-ETHYL-2-(-(METHY Suppliers

Carbosynth
Tel
--
Fax
--
Email
sales@carbosynth.com
Country
United Kingdom
ProdList
6005
Advantage
58

681281-88-9, 5-(2-BENZOTHIAZOLYL)-3-ETHYL-2-(-(METHYRelated Search:


  • Akt Inhibitor IV - CAS 681281-88-9 - Calbiochem
  • (E)-5-(benzo[d]thiazol-2-yl)-3-ethyl-2-(2-(methyl(phenyl)amino)vinyl)-1-phenyl-1H-benzo[d]imidazol-3-ium iodide
  • 6-benzothiazol-2-yl-1-ethyl-2-[2-(methyl-phenyl-amino)-vinyl]-3-phenyl-3H-benzoimidazol-1-ium iodide
  • 5-(Benzo[d]thiazol-2-yl)-3-ethyl-2-(2-(methyl(phenyl)amino)vinyl)-1-phenyl-1H-benzo[d]imidazol-3-ium iodide
  • 6-(2-Benzothiazolyl)-1-ethyl-2-[2-(methylphenylamino)ethenyl]-3-phenyl-1H-benzimidazolium iodide
  • 5-(2-BENZOTHIAZOLYL)-3-ETHYL-2-(-(METHY
  • 681281-88-9
  • C31H27N4SI