azafenidin

Product Name: azafenidin
CAS No.: 68049-83-2
Chemical Name: azafenidin
Synonyms: C10895;R 6447;Evolus;Milestone;IN-R 6447;DPX-R 6447;azafenidin;2-(2,4-dichloro-5-prop-2-ynyloxyphenyl)-5,6,7,8-tetrahydro-1,2,4-triazole(4,3-a)pyridin-3(2H)-one;2-(2,4-dichloro-5-prop-2-ynyloxypnenyl)-5,6,7,8-tetrahy-dro-1,2,4-trizolo [4,3-α] pyridin-3-(2H)-one;1,2,4-Triazolo[4,3-a]pyridin-3(2H)-one, 2-[2,4-dichloro-5-(2-propyn-1-yloxy)phenyl]-5,6,7,8-tetrahydro-
CBNumber: CB5945861
Molecular Formula: C15H13Cl2N3O2
Formula Weight: 338.19
MOL File: 68049-83-2.mol

More

Less

azafenidin Property

Melting point:: 168-168.5°
Boiling point:: 468.9±55.0 °C(Predicted)
Density: 1.43±0.1 g/cm3(Predicted)
solubility: DMSO (Slightly), Methanol (Slightly)
form: Solid
pka: 2.45±0.20(Predicted)
color: Brown to Dark Brown
EPA Substance Registry System: Azafeniden (68049-83-2)

More

Less

Safety

Hazard Codes: T,N
Risk Statements: 61-48/22-62-50/53
Safety Statements: 53-45-60-61
Toxicity: LD50 in rats, mice, bobwhite quail, mallard duck (mg/kg): >5000, >5000, >2500, >2500 orally; in rabbits (mg/kg): >2000 dermally.; LC50 in rats, rainbow trout, blue gill sunfish (mg/l): >5.3, 33, 48 (Amuti)

More

Less

Hazard and Precautionary Statements (GHS)

Symbol(GHS)

Signal word

Danger

Hazard statements

H373May cause damage to organs through prolonged or repeated exposure

H410Very toxic to aquatic life with long lasting effects

Precautionary statements

P260Do not breathe dust/fume/gas/mist/vapours/spray.

P273Avoid release to the environment.

P314Get medical advice/attention if you feel unwell.

P391Collect spillage. Hazardous to the aquatic environment

P501Dispose of contents/container to..…

More

Less

N-Bromosuccinimide Price

TRC

Product number: A797400
Product name: Azafenidin
Packaging: 0.5mg
Price: $195
Updated: 2021/12/16

American Custom Chemicals Corporation

Product number: AGR0000375
Product name: AZAFENIDIN
Purity: 95.00%
Packaging: 5MG
Price: $496.14
Updated: 2021/12/16

Medical Isotopes, Inc.

Product number: 38782
Product name: Azafenidin
Packaging: 5mg
Price: $990
Updated: 2021/12/16

More

Less

azafenidin Chemical Properties,Usage,Production

Uses

Azafenidin is a weed controlling herbicide used in various crops.

Uses

Herbicide.

Definition

ChEBI: Azafenidin is a triazolopyridine that is 5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one which is substituted at position 2 by a 2,4-dichloro-5-(prop-2-yn-1-yloxy)phenyl group. A protoporphyrinogen oxidase inhibitor, it is used as a herbicide to control weeds in fruit crops such as pineapple, citrus, melons, and grapes. Not approved for use within the European Union. It has a role as an EC 1.3.3.4 (protoporphyrinogen oxidase) inhibitor. It is a triazolopyridine, a terminal acetylenic compound and a dichlorobenzene.

Metabolic pathway

A common degradation reaction of azafenidin in light, plants and soil is O-dealkylation, and interesting minor reactions in soil are the subsequent methylation of the O-dealkylated degradation product and the reduction of the propynyl group under anaerobic conditions. In soil and light, azafenidin is also readily split to form the triazolinone heterocycle. Azafenidin is readily metabolized in rats and lactating goats through O-dealkylation, hydroxylation of the triazolinone ring in several positions, and glucuronide and sulfate conjugation.

azafenidin Preparation Products And Raw materials

Raw materials

Erythromycin Estolate 2,4-Dichlorophenol (-)-MENTHYL CHLOROFORMATE

Preparation Products

More

Less

azafenidin Suppliers

China 10 India 1 United States 2 Global 13

J & K SCIENTIFIC LTD.

Tel: 010-82848833 400-666-7788
Fax: 86-10-82849933
Email: jkinfo@jkchemical.com
Country: China
ProdList: 96815
Advantage: 76

Shanghai TaoSu Biochemical Technology Co., Ltd.

Tel: 021-33632979
Fax: 021-34692979
Email: info@tsbiochem.com
Country: China
ProdList: 8073
Advantage: 58

Shenzhen SUNGENING Bio-Medical Co., Ltd.

Tel: 0755-28967200 13631290199
Fax: 0755-28967200
Email: wxf@sungening.com
Country: China
ProdList: 9506
Advantage: 60

Shenzhen Polymeri Biochemical Technology Co., Ltd.

Tel: +86-400-002-6226 13028896684
Email: sales@rrkchem.com
Country: China
ProdList: 55827
Advantage: 58

Hubei Jusheng Technology Co.,Ltd.

Tel: 18871490254
Fax: 027-59599243
Email: linda@hubeijusheng.com
Country: CHINA
ProdList: 28180
Advantage: 58

Huansheng Meisen Pharmaceutical Technology (Shandong) Co., Ltd

Tel: 0531-88762217 18301471076
Email: sales@acespharma.com
Country: China
ProdList: 3863
Advantage: 58

Shandong Mopai Biotechnology Co., Ltd

Tel: 13053322091 13053322091
Email: admin@mopaikeji.com
Country: China
ProdList: 10969
Advantage: 58

Nantong Zhonghe Chemical New Materials Co., Ltd

Tel: 13003551299 13003551299
Email: 2369399482@qq.com
Country: China
ProdList: 7568
Advantage: 58

Zibo Hangyu Biotechnology Development Co., Ltd

Tel: +86-0533-2185556 +8617865335152
Email: Mandy@hangyubiotech.com
Country: China
ProdList: 11013
Advantage: 58

68049-83-2, azafenidinRelated Search:

(3-ETHYL-PHENYL)-HYDRAZINE HYDROCHLORIDE (4-CHLORO-3-METHYL-PHENYL)-HYDRAZINE HYDROCHLORIDE 2-IMINOPIPERIDINE HYDROCHLORIDE 4,5-DIETHYL-2,4-DIHYDRO 1,2,4-TRIAZOL-3 ONE azafenidin 2-(2,4-DICHLORO-PHENYL)-5-METHYL-2,4-DIHYDRO-[1,2,4]TRIAZOL-3-ONE Azafenidin-13C6

2-(2,4-dichloro-5-prop-2-ynyloxyphenyl)-5,6,7,8-tetrahydro-1,2,4-triazole(4,3-a)pyridin-3(2H)-one

azafenidin

Evolus

Milestone

2-(2,4-dichloro-5-prop-2-ynyloxypnenyl)-5,6,7,8-tetrahy-dro-1,2,4-trizolo [4,3-α] pyridin-3-(2H)-one

DPX-R 6447

IN-R 6447

R 6447

C10895

1,2,4-Triazolo[4,3-a]pyridin-3(2H)-one, 2-[2,4-dichloro-5-(2-propyn-1-yloxy)phenyl]-5,6,7,8-tetrahydro-

68049-83-2

Agro-Products, Aromatics, Heterocycles