ChemicalBook > CAS DataBase List > Fananserin
Fananserin
- Product Name
- Fananserin
- CAS No.
- 127625-29-0
- Chemical Name
- Fananserin
- Synonyms
- RP-62203;Fananserin;2-[3-[4-(4-Fluorophenyl)piperazino]propyl]-2H-naphth[1,8-cd]isothiazole 1,1-dioxide;2-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl)-2H-naphtho[1,8-cd]isothiazole 1,1-dioxide;2-[3-[4-(4-Fluorophenyl)-1-piperazinyl]propyl]-2H-naphthyl[1,8-cd]isothiazole-1,1-dioxide;2H-Naphth[1,8-cd]isothiazole, 2-[3-[4-(4-fluorophenyl)-1-piperazinyl]propyl]-, 1,1-dioxide;Fananserin,Inhibitor,5-HT Receptor,inhibit,5-HT2,RP62203,RP-62203,dopamine,Dopamine Receptor,Serotonin Receptor,5-hydroxytryptamine Receptor
- CBNumber
- CB71073778
- Molecular Formula
- C23H24FN3O2S
- Formula Weight
- 425.52
- MOL File
- 127625-29-0.mol
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Fananserin Property
- Melting point:
- 95-97 °C(Solv: acetonitrile (75-05-8))
- Boiling point:
- 641.1±65.0 °C(Predicted)
- Density
- 1.331±0.06 g/cm3(Predicted)
- storage temp.
- Store at RT
- solubility
- Soluble to 100 mM in DMSO
- form
- Powder
- pka
- 7.31±0.10(Predicted)
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N-Bromosuccinimide Price
Tocris
- Product number
- 2645
- Product name
- Fananserin
- Purity
- ≥99%(HPLC)
- Packaging
- 10
- Price
- $155
- Updated
- 2021/12/16
Tocris
- Product number
- 2645
- Product name
- Fananserin
- Purity
- ≥99%(HPLC)
- Packaging
- 50
- Price
- $558
- Updated
- 2021/12/16
Usbiological
- Product number
- 255281
- Product name
- Fananserin
- Packaging
- 10mg
- Price
- $403
- Updated
- 2021/12/16
TRC
- Product number
- F102368
- Product name
- Fananserin
- Packaging
- 2.5mg
- Price
- $165
- Updated
- 2021/12/16
ChemScene
- Product number
- CS-0024310
- Product name
- Fananserin
- Purity
- 99.83%
- Packaging
- 5mg
- Price
- $188
- Updated
- 2021/12/16
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Fananserin Chemical Properties,Usage,Production
Uses
Antipsychotic.
Uses
Fananserin is an antagonist of 5-HT2A.
Definition
ChEBI: LSM-2183 is a sulfonic acid derivative and a member of naphthalenes.
Biological Activity
5-HT 2A receptor antagonist that also displays high affinity at D 4 receptors (K i values are 0.26, 2.93, 25, 38, 70 and 726 nM for 5-HT 2A , D 4 , H 1 , α 1 , 5-HT 1A and D 2 receptors respectively). Inhibits inositol phosphate formation evoked by 5-HT in vitro (IC 50 = 7.76 nM) and antagonizes mescaline-induced head twitches in vivo .
Fananserin Preparation Products And Raw materials
Raw materials
Preparation Products
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