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ChemicalBook > CAS DataBase List > 5-Bromo-2-methoxybenzonitrile

5-Bromo-2-methoxybenzonitrile

Uses
Product Name
5-Bromo-2-methoxybenzonitrile
CAS No.
144649-99-0
Chemical Name
5-Bromo-2-methoxybenzonitrile
Synonyms
ST5408714;Albb-008949;4-Bromo-2-cyanoanisole;5-Bromo-o-anisyl cyanide;-Bromo-o-anisyl cyanide;2-Methoxy-5-bromobenzonitrile;Benzonitrile, 5-broMo-2-Methoxy-;5-Bromo-2-methoxybenzonitrile 96%;5-Bromo-2-(methyloxy)benzonitrile;5-Bromo-2-methoxybenzonitrile >
CBNumber
CB71106575
Molecular Formula
C8H6BrNO
Formula Weight
212.04
MOL File
144649-99-0.mol
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5-Bromo-2-methoxybenzonitrile Property

Melting point:
91-92 °C
Boiling point:
287.8±20.0 °C(Predicted)
Density 
1.56±0.1 g/cm3(Predicted)
storage temp. 
2-8°C
solubility 
soluble in Methanol
form 
powder to crystal
color 
White to Yellow to Orange
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Safety

Hazard Codes 
Xn
Risk Statements 
20/21/22
Safety Statements 
36/37
RIDADR 
UN3439
WGK Germany 
3
HazardClass 
6.1
PackingGroup 
III
HS Code 
29269090
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
701173
Product name
5-Bromo-2-methoxybenzonitrile
Purity
96%
Packaging
5g
Price
$73
Updated
2023/06/20
Sigma-Aldrich
Product number
701173
Product name
5-Bromo-2-methoxybenzonitrile
Purity
96%
Packaging
25g
Price
$284
Updated
2023/01/07
TCI Chemical
Product number
B3123
Product name
5-Bromo-2-methoxybenzonitrile
Purity
>98.0%(GC)
Packaging
5g
Price
$110
Updated
2025/07/31
TCI Chemical
Product number
B3123
Product name
5-Bromo-2-methoxybenzonitrile
Purity
>98.0%(GC)
Packaging
25g
Price
$424
Updated
2025/07/31
TRC
Product number
B696613
Product name
5-Bromo-2-methoxybenzonitrile
Packaging
250mg
Price
$55
Updated
2021/12/16
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5-Bromo-2-methoxybenzonitrile Chemical Properties,Usage,Production

Uses

5-Bromo-2-methoxybenzonitrile can be used as an organic and pharmaceutical intermediate. Halogenated benzonitrile is an important organic intermediate, mainly used in the preparation of pharmaceuticals and pesticides, and has wide applications in the manufacture of dyes, engineering plastics, and photosensitive materials.

Chemical Properties

off-white crystalline

Synthesis

6609-56-9

144649-99-0

General procedure for the synthesis of 2-methoxy-5-bromobenzonitrile from 2-methoxybenzonitrile: N-bromosuccinimide (NBS, 1.5 eq., 0.3 mmol), catalyst (10 mol%, 0.02 mmol), and acetonitrile (CH3CN, 1.0 mL) were added to the reaction tube, followed by 2-methoxybenzonitrile (0.2 mmol). The reaction mixture was stirred for 12 h at room temperature protected from light. Upon completion of the reaction, the reaction was quenched with saturated sodium thiosulfate (Na2S2O3) aqueous solution (2 mL). The reaction mixture was extracted with ethyl acetate (3.5 mL). The organic phases were combined, washed with brine (10 mL), dried over anhydrous sodium sulfate (Na2SO4) and filtered through a diatomaceous earth pad. The filtrate was concentrated under reduced pressure and the residue was purified by rapid chromatography on a silica gel column using petroleum ether/dichloromethane (5:1) as eluent to afford the target product 2-methoxy-5-bromobenzonitrile.

References

[1] Tetrahedron, 2017, vol. 73, # 50, p. 7105 - 7114
[2] Patent: US2009/203657, 2009, A1. Location in patent: Page/Page column 51
[3] Patent: US2009/203677, 2009, A1. Location in patent: Page/Page column 54
[4] Patent: US2009/197871, 2009, A1. Location in patent: Page/Page column 53-54
[5] Patent: WO2009/100169, 2009, A1. Location in patent: Page/Page column 132-133

5-Bromo-2-methoxybenzonitrile Preparation Products And Raw materials

Raw materials

Preparation Products

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5-Bromo-2-methoxybenzonitrile Suppliers

J & K SCIENTIFIC LTD.
Tel
18210857532; 18210857532
Fax
86-10-82849933
Email
jkinfo@jkchemical.com
Country
China
ProdList
96815
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76
Alfa Aesar
Tel
400-6106006
Fax
021-67582001/03/05
Email
saleschina@alfa-asia.com
Country
China
ProdList
30123
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84
TCI (Shanghai) Development Co., Ltd.
Tel
021-67121386
Fax
021-67121385
Email
Sales-CN@TCIchemicals.com
Country
China
ProdList
24529
Advantage
81
Energy Chemical
Tel
021-021-58432009 400-005-6266
Fax
021-58436166
Email
sales8178@energy-chemical.com
Country
China
ProdList
44801
Advantage
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Shijiazhuang Sdyano Fine Chemical Co., Ltd.
Tel
0311-89250318 031166536426
Fax
4000311741
Email
master@sjzsdyn.com
Country
China
ProdList
2807
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Shanghai Harvest Chemical Industrial Co., Ltd.
Tel
021-31038972,31038973 17321035817
Fax
+86-21-51385350
Email
sales@harvest-chem.com
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China
ProdList
2816
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64
Nanjing Chemlin Chemical Co., Ltd
Tel
025-83697070
Fax
+86-25-83453306
Email
info@chemlin.com.cn
Country
China
ProdList
15883
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64
Shanghai Hanhong Scientific Co.,Ltd.
Tel
021-54306202 13764082696
Email
info@hanhongsci.com
Country
China
ProdList
42934
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64
Shandong Xiya Chemical Co., Ltd
Tel
4009903999 13355009207
Fax
0539-6365991
Email
3007715519@qq.com
Country
China
ProdList
18729
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57
Shanghai Sphchem Co., Ltd.
Tel
021-56491756 13512199871
Fax
021-5649-1756
Email
2819742715@qq.com
Country
China
ProdList
4000
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55
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View Lastest Price from 5-Bromo-2-methoxybenzonitrile manufacturers

Career Henan Chemical Co
Product
5-Bromo-2-methoxybenzonitrile 144649-99-0
Price
US $1.00/KG
Min. Order
1KG
Purity
99%
Supply Ability
200kg
Release date
2019-12-24

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