ChemicalBook > CAS DataBase List > SGC2085
SGC2085
- Product Name
- SGC2085
- CAS No.
- 1821908-48-8
- Chemical Name
- SGC2085
- Synonyms
- CS-2688;CS-2529;SGC-2085; SGC 2085;SGC2085, 10 mM in DMSO;(S)-2-Amino-N-(4-(3,5-dimethylphenoxy)-3-methylbenzyl)propanamide;SGC2085,SGC 2085,Inhibitor,inhibit,SGC-2085,Histone Methyltransferase;(2S)-2-Amino-N-[[4-(3,5-dimethylphenoxy)-3-methylphenyl]methyl]Propanamide;Propanamide, 2-amino-N-[[4-(3,5-dimethylphenoxy)-3-methylphenyl]methyl]-, (2S)-
- CBNumber
- CB73160081
- Molecular Formula
- C19H24N2O2
- Formula Weight
- 312.41
- MOL File
- 1821908-48-8.mol
More
Less
SGC2085 Property
- Boiling point:
- 498.3±45.0 °C(Predicted)
- Density
- 1.097±0.06 g/cm3(Predicted)
- storage temp.
- Keep in dark place,Inert atmosphere,Store in freezer, under -20°C
- solubility
- DMSO : ≥ 32 mg/mL (102.43 mM)
- pka
- 14.83±0.46(Predicted)
- form
- Solid
- color
- White to off-white
- InChI
- InChI=1S/C19H24N2O2/c1-12-7-13(2)9-17(8-12)23-18-6-5-16(10-14(18)3)11-21-19(22)15(4)20/h5-10,15H,11,20H2,1-4H3,(H,21,22)/t15-/m0/s1
- InChIKey
- GLFOFXKMALJTCZ-HNNXBMFYSA-N
- SMILES
- C(NCC1=CC=C(OC2=CC(C)=CC(C)=C2)C(C)=C1)(=O)[C@@H](N)C
More
Less
N-Bromosuccinimide Price
ChemScene
- Product number
- CS-6152
- Product name
- SGC2085
- Purity
- 99.87%
- Packaging
- 1mg
- Price
- $110
- Updated
- 2021/12/16
ChemScene
- Product number
- CS-6152
- Product name
- SGC2085
- Purity
- 99.87%
- Packaging
- 5mg
- Price
- $330
- Updated
- 2021/12/16
ChemScene
- Product number
- CS-6152
- Product name
- SGC2085
- Purity
- 99.87%
- Packaging
- 10mg
- Price
- $500
- Updated
- 2021/12/16
AK Scientific
- Product number
- 5127EG
- Product name
- (2S)-2-Amino-N-[[4-(3,5-dimethylphenoxy)-3-methylphenyl]methyl]propanamide
- Packaging
- 250mg
- Price
- $439
- Updated
- 2021/12/16
ChemScene
- Product number
- CS-6152
- Product name
- SGC2085
- Purity
- 99.87%
- Packaging
- 50mg
- Price
- $1500
- Updated
- 2021/12/16
More
Less
SGC2085 Chemical Properties,Usage,Production
Uses
SGC2085 is a potent and selective inhibitor of coactivator associated arginine methyltransferase 1 (CARM1) with an IC50 of 50 nM. SGC2085 also selectively inhibits PRMT6 with an IC50 value of 5.2 μM, but not other PRMT proteins[1].
IC 50
PRMT4
References
[1] Ferreira de Freitas R, et al. Discovery of a Potent and Selective Coactivator Associated Arginine Methyltransferase 1 (CARM1) Inhibitor by Virtual Screening. J Med Chem. 2016 Jul 28;59(14):6838-47. DOI:10.1021/acs.jmedchem.6b00668
SGC2085 Preparation Products And Raw materials
Raw materials
Preparation Products
More
Less
SGC2085 Suppliers
- Tel
- --
- Fax
- --
- sales@ajchem.in
- Country
- India
- ProdList
- 6100
- Advantage
- 58
1821908-48-8, SGC2085Related Search:
1-Piperazinecarboxylic acid, 4-[3-amino-6-(2-hydroxyphenyl)-4-pyridazinyl]-, 1,1-dimethylethyl ester
SGC-GAK-1
SGC707
SGC0946