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R-(+)-LISURIDE HYDROGEN MALEATE

Product Name
R-(+)-LISURIDE HYDROGEN MALEATE
CAS No.
19875-60-6
Chemical Name
R-(+)-LISURIDE HYDROGEN MALEATE
Synonyms
Apodel;cuvalit;lysenyl;Revanil;Dopergin;lisuridemaleate;lysenylbimaleate;Lysuride maleate;lysenylhydrogenmaleate;lisuridehydrogenmaleate
CBNumber
CB7338975
Molecular Formula
C24H30N4O5
Formula Weight
454.52
MOL File
19875-60-6.mol
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R-(+)-LISURIDE HYDROGEN MALEATE Property

Melting point:
200° (dec)
alpha 
D20 +288° (c = 0.5 in methanol)
storage temp. 
Desiccate at RT
solubility 
DMSO:34.83(Max Conc. mg/mL);76.63(Max Conc. mM)
form 
Solid
color 
Off-White to Light Yellow
Stability:
Hygroscopic
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Safety

Toxicity
LD50 i.v. in mice: 14.4 mg/kg (Votava, Lamplova)
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Danger
Hazard statements

H300Fatal if swallowed

Precautionary statements

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P301+P310IF SWALLOWED: Immediately call a POISON CENTER or doctor/physician.

P321Specific treatment (see … on this label).

P330Rinse mouth.

P405Store locked up.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

Tocris
Product number
4052
Product name
Lisuridemaleate
Purity
≥99%(HPLC)
Packaging
10
Price
$233
Updated
2021/12/16
Tocris
Product number
4052
Product name
Lisuridemaleate
Purity
≥99%(HPLC)
Packaging
50
Price
$980
Updated
2021/12/16
Usbiological
Product number
255690
Product name
Lisuride maleate
Packaging
10mg
Price
$480
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0003189
Product name
R-(+)-LISURIDE HYDROGEN MALEATE
Purity
95.00%
Packaging
5MG
Price
$599.68
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0003189
Product name
R-(+)-LISURIDE HYDROGEN MALEATE
Purity
95.00%
Packaging
25MG
Price
$652.46
Updated
2021/12/16
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R-(+)-LISURIDE HYDROGEN MALEATE Chemical Properties,Usage,Production

Uses

Lisuride Maleate is a dopamine receptor agonist with additionally serotoninergic, adrenergic, and glutamate antagonistic properties. Treatment of Parkinsonism and other diseases associated with high level of prolactin.

in vivo

Lisuride (maleate) (0.78 and 3.13 mg/kg; i.p.; p.o.) is 3-4 times more potent on i.p. than on p.o. [2].
Lisuride (maleate) (0.78-3.13 mg/kg; i.p.) antagonizes the motor depression and hypothermia induced by reserpine[2].
Lisuride (maleate) (0.78-3.13 mg/kg; i.p.) is about as effective as apomorphine and D-amphetamine and causes significant hypothermia measured after dosages as low as 0.10 mg/kg i.p.[2].

Animal Model:NMRI mice (18-25 g)[2]
Dosage:0.78 and 3.13 mg/kg
Administration:i.p., p.o.
Result:Been 3-4 times more potent on i.p. than on p.o..

storage

Store at RT

R-(+)-LISURIDE HYDROGEN MALEATE Preparation Products And Raw materials

Raw materials

Preparation Products

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R-(+)-LISURIDE HYDROGEN MALEATE Suppliers

China 24 Germany 1 United Kingdom 1 United States 6 Global 32
3B Pharmachem (Wuhan) International Co.,Ltd.
Tel
821-50328103-801 18930552037
Fax
86-21-50328109
Email
3bsc@sina.com
Country
China
ProdList
15838
Advantage
69
EMMX Biotechnology LLC
Tel
888-539-0666
Fax
888-539-0666
Email
info@emmx.com
Country
United States
ProdList
8447
Advantage
60
INTERCHEMIE NANJING PHARMATECH CO., LTD
Tel
13656237714 13656237714;
Fax
0512-65852853
Email
xiaokunfu@kyyykj.com
Country
China
ProdList
295
Advantage
55
Shanghai Zhibang Biological Medicine Co., LTD
Tel
021-54285032 18116461626
Fax
021-54285032
Email
25493162@qq.com
Country
China
ProdList
148
Advantage
58
Zhengzhou Acme Chemical Co., Ltd.
Tel
0371-037163312495,13303845143 13303845143
Fax
QQ3001379618
Email
3001379618@qq.com
Country
China
ProdList
10267
Advantage
58
Energy Chemical
Tel
021-58432009 400-005-6266
Fax
021-58436166
Email
marketing@energy-chemical.com
Country
China
ProdList
44918
Advantage
58
Cdreamlab (Hubei) Technology Co., LTD
Tel
0717-6300888 18062399888
Email
service@cdreamlab.com
Country
China
ProdList
299
Advantage
58
Shanghai Tachizaki Biomedical Research Center
Tel
18014399201
Email
sales@chemlab-tachizaki.com
Country
China
ProdList
2742
Advantage
58
Shaanxi Xihua Chemical Industry Co., Ltd
Tel
029-81136151 17392212881
Email
1095@dideu.com
Country
China
ProdList
10001
Advantage
58
R&D Systems, Inc
Tel
18003437475
Fax
1-612-656-4400
Email
rdname@qq.com
Country
China
ProdList
6960
Advantage
58

19875-60-6, R-(+)-LISURIDE HYDROGEN MALEATERelated Search:

R-(+)-LISURIDE HYDROGEN MALEATE S-(-)-LISURIDE 1H-INDOLE-4-ETHANAMINE

  • 3-(9,10-didehydro-6-methylergolin-8-alpha-yl)-1,1-diethylureamaleate(1:1)
  • 3-(9,10-didehydro-6-methylergolin-8-alpha-yl)-1,1-diethyl-uremaleate(1:1)
  • 3-(9,10-didehydro-6-methylergolin-8-yl)-1,1-diethylureahydrogenmaleate
  • cuvalit
  • lisuridehydrogenmaleate
  • lisuridemaleate
  • lysenyl
  • lysenylbimaleate
  • 1-((5r,8s)-6-methyl-9,10-didehydro-8-ergolinyl)-3,3-diethylureahydrogenmale
  • lysenylhydrogenmaleate
  • R-(+)-LISURIDE HYDROGEN MALEATE
  • Apodel
  • Dopergin
  • Revanil
  • Urea, 3-(9,10-didehydro-6-methylergolin-8a-yl)-1,1-diethyl-, maleate (1:1) (8CI)
  • Urea, N'-[(8a)-9,10-didehydro-6-methylergolin-8-yl]-N,N-diethyl-, (2Z)-2-butenedioate (1:1) (9CI)
  • Urea, N'-[(8a)-9,10-didehydro-6-methylergolin-8-yl]-N,N-diethyl-, (Z)-2-butenedioate (1:1)
  • Lysuride maleate
  • N'-(9,10-Didehydro-6-methylergoline-8α-yl)-N,N-diethylurea·(Z)-2-butenedioic acid
  • N'-[(8α)-9,10-Didehydro-6-methylergolin-8-yl]-N,N-diethylureamaleate
  • Urea, N'-[(8α)-9,10-didehydro-6-methylergolin-8-yl]-N,N-diethyl-, (2Z)-2-butenedioate (1:1)
  • 19875-60-6
  • C25H31N3O5
  • C20H26N4OC4H4O4