ChemicalBook > CAS DataBase List > R-(+)-LISURIDE HYDROGEN MALEATE

R-(+)-LISURIDE HYDROGEN MALEATE

Product Name
R-(+)-LISURIDE HYDROGEN MALEATE
CAS No.
19875-60-6
Chemical Name
R-(+)-LISURIDE HYDROGEN MALEATE
Synonyms
Apodel;cuvalit;lysenyl;Revanil;Dopergin;lisuridemaleate;lysenylbimaleate;Lysuride maleate;lysenylhydrogenmaleate;lisuridehydrogenmaleate
CBNumber
CB7338975
Molecular Formula
C24H30N4O5
Formula Weight
454.52
MOL File
19875-60-6.mol
More
Less

R-(+)-LISURIDE HYDROGEN MALEATE Property

Melting point:
200° (dec)
alpha 
D20 +288° (c = 0.5 in methanol)
storage temp. 
Desiccate at RT
solubility 
DMSO:34.83(Max Conc. mg/mL);76.63(Max Conc. mM)
form 
Solid
color 
Off-White to Light Yellow
Stability:
Hygroscopic
More
Less

Safety

Toxicity
LD50 i.v. in mice: 14.4 mg/kg (Votava, Lamplova)
More
Less

Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Danger
Hazard statements

H300Fatal if swallowed

Precautionary statements

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P301+P310IF SWALLOWED: Immediately call a POISON CENTER or doctor/physician.

P321Specific treatment (see … on this label).

P330Rinse mouth.

P405Store locked up.

P501Dispose of contents/container to..…

More
Less

N-Bromosuccinimide Price

Tocris
Product number
4052
Product name
Lisuridemaleate
Purity
≥99%(HPLC)
Packaging
10
Price
$233
Updated
2021/12/16
Tocris
Product number
4052
Product name
Lisuridemaleate
Purity
≥99%(HPLC)
Packaging
50
Price
$980
Updated
2021/12/16
Usbiological
Product number
255690
Product name
Lisuride maleate
Packaging
10mg
Price
$480
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0003189
Product name
R-(+)-LISURIDE HYDROGEN MALEATE
Purity
95.00%
Packaging
5MG
Price
$599.68
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0003189
Product name
R-(+)-LISURIDE HYDROGEN MALEATE
Purity
95.00%
Packaging
25MG
Price
$652.46
Updated
2021/12/16
More
Less

R-(+)-LISURIDE HYDROGEN MALEATE Chemical Properties,Usage,Production

Uses

Lisuride Maleate is a dopamine receptor agonist with additionally serotoninergic, adrenergic, and glutamate antagonistic properties. Treatment of Parkinsonism and other diseases associated with high level of prolactin.

in vivo

Lisuride (maleate) (0.78 and 3.13 mg/kg; i.p.; p.o.) is 3-4 times more potent on i.p. than on p.o. [2].
Lisuride (maleate) (0.78-3.13 mg/kg; i.p.) antagonizes the motor depression and hypothermia induced by reserpine[2].
Lisuride (maleate) (0.78-3.13 mg/kg; i.p.) is about as effective as apomorphine and D-amphetamine and causes significant hypothermia measured after dosages as low as 0.10 mg/kg i.p.[2].

Animal Model:NMRI mice (18-25 g)[2]
Dosage:0.78 and 3.13 mg/kg
Administration:i.p., p.o.
Result:Been 3-4 times more potent on i.p. than on p.o..

storage

Store at RT

R-(+)-LISURIDE HYDROGEN MALEATE Preparation Products And Raw materials

Raw materials

Preparation Products

More
Less

R-(+)-LISURIDE HYDROGEN MALEATE Suppliers

China 24 Germany 1 United Kingdom 1 United States 6 Global 32
3B Pharmachem (Wuhan) International Co.,Ltd.
Tel
821-50328103-801 18930552037
Fax
86-21-50328109
Email
3bsc@sina.com
Country
China
ProdList
15838
Advantage
69
INTERCHEMIE NANJING PHARMATECH CO., LTD
Tel
13656237714 13656237714;
Fax
0512-65852853
Email
xiaokunfu@kyyykj.com
Country
China
ProdList
295
Advantage
55
Shanghai Zhibang Biological Medicine Co., LTD
Tel
021-54285032 18116461626
Fax
021-54285032
Email
25493162@qq.com
Country
China
ProdList
148
Advantage
58
Zhengzhou Acme Chemical Co., Ltd.
Tel
0371-037163312495,13303845143 13303845143
Fax
QQ3001379618
Email
3001379618@qq.com
Country
China
ProdList
10267
Advantage
58
Energy Chemical
Tel
021-58432009 400-005-6266
Fax
021-58436166
Email
marketing@energy-chemical.com
Country
China
ProdList
44918
Advantage
58
Cdreamlab (Hubei) Technology Co., LTD
Tel
0717-6300888 18062399888
Email
service@cdreamlab.com
Country
China
ProdList
299
Advantage
58
Shanghai Tachizaki Biomedical Research Center
Tel
18014399201
Email
sales@chemlab-tachizaki.com
Country
China
ProdList
2742
Advantage
58
Shaanxi Xihua Chemical Industry Co., Ltd
Tel
029-81136151 17392212881
Email
1095@dideu.com
Country
China
ProdList
10001
Advantage
58
R&D Systems, Inc
Tel
18003437475
Fax
1-612-656-4400
Email
rdname@qq.com
Country
China
ProdList
6960
Advantage
58
Cayman Chemical Company
Tel
800-364-9897
Email
sales@caymanchem.com
Country
China
ProdList
6838
Advantage
58
Biosynth Biological Technology (Suzhou) Co Ltd
Tel
51288865780
Email
sales@biosynth.com
Country
China
ProdList
6051
Advantage
58
Santa Cruz Biotechnology Inc
Tel
021-60936350
Email
scbt@scbt.com
Country
China
ProdList
6594
Advantage
58
Shandong Quadristar Material Technology Co., Ltd
Tel
18016441705
Email
yufei.sun@quadristar.com.cn
Country
China
ProdList
175
Advantage
58
Shanghai meikai technology co., ltd
Tel
021-68689288 15300790979
Fax
wechat 18721550091
Email
info@mkbio.com.cn
Country
China
ProdList
5000
Advantage
58
DAYANG CHEM (HANGZHOU) CO.,LTD
Tel
+86-88938639 +86-17705817739
Email
info@dycnchem.com
Country
China
ProdList
53899
Advantage
58
Shanghai Haoyang Biological Technology Co., Ltd.
Tel
--
Fax
--
Email
596799915@QQ.COM
Country
CHINA
ProdList
2905
Advantage
58
Beijing Baiao Innovation Technology Co., Ltd.
Tel
--
Fax
--
Email
3007606172@qq.com
Country
CHINA
ProdList
6002
Advantage
58
Beijing Bolide Biotechnology Co., Ltd.
Tel
--
Fax
--
Email
1985563437@qq.com
Country
CHINA
ProdList
6525
Advantage
58
Absin Bioscience Inc.
Tel
--
Fax
--
Email
chenjw@absin.cn
Country
CHINA
ProdList
6208
Advantage
58
Shanghai Chaoyan Biotechnology Co., Ltd.
Tel
--
Fax
--
Email
471161314@qq.com
Country
CHINA
ProdList
6210
Advantage
58
Shanghai Hao Zhun Biological Technology Co., Ltd.
Tel
--
Fax
--
Email
info@zzsrm.com
Country
CHINA
ProdList
6650
Advantage
58
Yick-Vic Chemicals & Pharmaceuticals (HK) Ltd
Tel
--
Fax
--
Email
sales@yickvic.com
Country
China
ProdList
6206
Advantage
58
A.T.CHEMICAL
Tel
--
Fax
--
Email
Jeffreyxu@atchem.net
Country
China
ProdList
6589
Advantage
51
Advanced Technology & Industrial Co., Ltd.
Tel
--
Fax
--
Email
sales@advtechind.com
Country
China
ProdList
6523
Advantage
75

19875-60-6, R-(+)-LISURIDE HYDROGEN MALEATERelated Search:

R-(+)-LISURIDE HYDROGEN MALEATE S-(-)-LISURIDE 1H-INDOLE-4-ETHANAMINE

  • 3-(9,10-didehydro-6-methylergolin-8-alpha-yl)-1,1-diethylureamaleate(1:1)
  • 3-(9,10-didehydro-6-methylergolin-8-alpha-yl)-1,1-diethyl-uremaleate(1:1)
  • 3-(9,10-didehydro-6-methylergolin-8-yl)-1,1-diethylureahydrogenmaleate
  • cuvalit
  • lisuridehydrogenmaleate
  • lisuridemaleate
  • lysenyl
  • lysenylbimaleate
  • 1-((5r,8s)-6-methyl-9,10-didehydro-8-ergolinyl)-3,3-diethylureahydrogenmale
  • lysenylhydrogenmaleate
  • R-(+)-LISURIDE HYDROGEN MALEATE
  • Apodel
  • Dopergin
  • Revanil
  • Urea, 3-(9,10-didehydro-6-methylergolin-8a-yl)-1,1-diethyl-, maleate (1:1) (8CI)
  • Urea, N'-[(8a)-9,10-didehydro-6-methylergolin-8-yl]-N,N-diethyl-, (2Z)-2-butenedioate (1:1) (9CI)
  • Urea, N'-[(8a)-9,10-didehydro-6-methylergolin-8-yl]-N,N-diethyl-, (Z)-2-butenedioate (1:1)
  • Lysuride maleate
  • N'-(9,10-Didehydro-6-methylergoline-8α-yl)-N,N-diethylurea·(Z)-2-butenedioic acid
  • N'-[(8α)-9,10-Didehydro-6-methylergolin-8-yl]-N,N-diethylureamaleate
  • Urea, N'-[(8α)-9,10-didehydro-6-methylergolin-8-yl]-N,N-diethyl-, (2Z)-2-butenedioate (1:1)
  • 19875-60-6
  • C25H31N3O5
  • C20H26N4OC4H4O4