Paliperidone Palmitate

Product Name: Paliperidone Palmitate
CAS No.: 199739-10-1
Chemical Name: Paliperidone Palmitate
Synonyms: Invega Sustenna;RO 92670;Paliperidone Palmitate;Paliperidone Palmitate-d31;Paliperidone Palmitate [USAN];9-Hydroxyrisperidone palmitate;Paliperidone Palmitate USP/EP/BP;Paliperidone Palmitate Benzisoxazole Impurity;Paliperidone Impurity 39 (Paliperidone Palmitate);3-(2-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethyl)-2-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-9-yl palmitate
CBNumber: CB82519012
Molecular Formula: C39H57FN4O4
Formula Weight: 664.89
MOL File: 199739-10-1.mol

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Paliperidone Palmitate Property

Melting point:: 110-115°C
Boiling point:: 736.3±70.0 °C(Predicted)
Density: 1.19
storage temp.: Sealed in dry,Store in freezer, under -20°C
solubility: Chloroform (Slightly), Ethyl Acetate (Slightly, Heated, Sonicated), Methanol (Slightly)
form: Solid
pka: 8.07±0.10(Predicted)
color: Off-White to Light Beige

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Hazard and Precautionary Statements (GHS)

Symbol(GHS)

Signal word

Danger

Hazard statements

H301Toxic if swalloed

Precautionary statements

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P301+P310IF SWALLOWED: Immediately call a POISON CENTER or doctor/physician.

P321Specific treatment (see … on this label).

P330Rinse mouth.

P405Store locked up.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

TRC

Product number: P141020
Product name: PaliperidonePalmitate
Packaging: 500mg
Price: $210
Updated: 2021/12/16

Activate Scientific

Product number: AS148096
Product name: PaliperidonePalmitate
Purity: 98%
Packaging: 250mg
Price: $233
Updated: 2021/12/16

American Custom Chemicals Corporation

Product number: API0027470
Product name: PALIPERIDONE PALMITATE
Purity: 95.00%
Packaging: 25MG
Price: $750.75
Updated: 2021/12/16

American Custom Chemicals Corporation

Product number: API0027470
Product name: PALIPERIDONE PALMITATE
Purity: 95.00%
Packaging: 250MG
Price: $1963.5
Updated: 2021/12/16

ChemScene

Product number: CS-0016387
Product name: Paliperidonepalmitate
Purity: 98.16%
Packaging: 10mg
Price: $70
Updated: 2021/12/16

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Paliperidone Palmitate Chemical Properties,Usage,Production

Description

Paliperidone palmitate is an atypical long acting antipsychotics，which can fast onset in acute phase and continuously improve the symptoms in maintenance phase． It has the solid efficacy and convenient ad[1]ministration，which offer a new option for schizophrenia treatment and will help patients to adhere the treatment and prevent relapse． As the sole long acting antipsychotics with monthly injection，it was approved by CFDA in 2011 and indicated for the acute and maintenance treatment of schizophrenia．

Uses

Paliperidone Palmitate is a long-acting injectable atypical antipsychotic used in the treatment of schizophrenia.

Definition

ChEBI: 3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl}-2-methyl-4-oxo-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-9-yl hexadecanoate is a fatty acid ester obtained by the formal condensation of the carboxy group of hexadecanoic acid with the hydroxy group of 3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl}-9-hydroxy-2-methyl-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-4-one. It is a member of 1,2-benzoxazoles, a heteroarylpiperidine, an organofluorine compound, a pyridopyrimidine and a fatty acid ester.

Side effects

The review of the literature also underlined that paliperidone palmitate is well tolerated, compared with placebo. Frequency and severity of side-effects such as extrapyramidal symptoms, hyperprolactinemia and weight gain, was similar or less than those found in treatment with other atypical antipsychotics, including long-acting ones.

Paliperidone Palmitate Preparation Products And Raw materials

Raw materials

Preparation Products

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Paliperidone Palmitate Suppliers

Austria 1 Canada 1 China 182 India 17 Mexico 1 United Kingdom 1 United States 11 Global 214

Zhuzhou focus pharmaceutical technology co., LTD

Tel: +86-13776644403
Email: robert@focuspharma.cc
Country: China
ProdList: 1957
Advantage: 58

Wuhan Wiseman Bioengineering Co.,Ltd

Tel: 027-59506022 13419526507
Fax: 027-59506022
Email: 13419526507@163.com
Country: China
ProdList: 2935
Advantage: 58

Jiangxi ravel Biotechnology Co.,Ltd

Tel: 18502762009
Email: 721846333@qq.com
Country: China
ProdList: 2446
Advantage: 58

Jewim Pharmaceutical (Shandong) Co., Ltd.

Tel: 15621883869
Email: 172688504@qq.com
Country: China
ProdList: 111
Advantage: 58

Henan Dongyao Pharmaceutical Technology Co., Ltd

Tel: 18519331287
Email: 1751713684@qq.com
Country: China
ProdList: 172
Advantage: 58

Jilin Lianben Technology Development Co., Ltd

Tel: 15688981295
Fax: 0432-62601618
Email: wangyifei@lianben.com
Country: China
ProdList: 46
Advantage: 58

Shanghai Boyle Chemical Co., Ltd.

Tel
Fax: 86-21-57758967
Email: sales@boylechem.com
Country: China
ProdList: 2923
Advantage: 55

J & K SCIENTIFIC LTD.

Tel: 010-82848833 400-666-7788
Fax: 86-10-82849933
Email: jkinfo@jkchemical.com
Country: China
ProdList: 96815
Advantage: 76

Chemvon Biotechnology Co., Ltd

Tel: 021-50790412
Fax: +86-21-50790419
Email: info@chemvon.com
Country: China
ProdList: 371
Advantage: 57

Chembest Research Laboratories Limited

Tel: 021-20908456
Fax: 021-58180499
Email: sales@BioChemBest.com
Country: China
ProdList: 6011
Advantage: 61

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View Lastest Price from Paliperidone Palmitate manufacturers

Sinoway Industrial co., ltd.

Product: Paliperidone Palmitate 199739-10-1
Price: US $175.00-85.00/Kg/Bag
Min. Order: 1Kg/Bag
Purity: 0.99
Supply Ability: 20 tons
Release date: 2023-12-05

Ouhuang Engineering Materials (Hubei) Co., Ltd

Product: Paliperidone Palmitate 199739-10-1
Price: US $50.00/kg
Min. Order: 1kg
Purity: 99.10%
Supply Ability: 50000kg
Release date: 2024-04-22

Zibo Hangyu Biotechnology Development Co., Ltd

Product: Paliperidone Palmitate 199739-10-1
Price: US $70.00-700.00/kg
Min. Order: 10kg
Purity: 0.99
Supply Ability: 20tons
Release date: 2023-11-20

199739-10-1, Paliperidone PalmitateRelated Search:

3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-9-hydroxy-2-methylpyrido[1,2-a]pyrimidin-4-one Paliperidone E-Oxime Isooctyl palmitate Clindamycin palmitate hydrochloride Paliperidone Paliperidone Impurity 4 2,4-Difluorophenyl-(4-piperidinyl)methanone oxime hydrochloride Isopropyl palmitate Ethylhexyl Palmitate Clindamycin palmitate hydrochloride Vitamin A palmitate PALMITELAIDIC ACID Paliperidone N-Oxide 9-hydroxy-2-methyl-3-vinyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-one (R)-9-Hydroxy Risperidone (S)-9-Hydroxy Risperidone 3-(2-Chloroethyl)-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one RAC 9-HYDROXYRISPERIDONE-D4

(9RS)-3-(2-(4-(6-Fluoro-1,2-benzisoxazol-3-yl)piperidin-1-yl)et hyl)-2-Methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido(1,2-a)pyriMi din-9-yl hexadecanoate

Hexadecanoic acid 3-[2-[4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl]-ethyl]-6,7,8,9-tetrahydro-2-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl ester

Paliperidone Palmitate

Paliperidone Palmitate [USAN]

Invega Sustenna

RO 92670

9-Hydroxyrisperidone palmitate

Hexadecanoic acid 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl ester

Paliperidone Palmitate-d31

Paliperidone Impurity 39 (Paliperidone Palmitate)

3-(2-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethyl)-2-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-9-yl palmitate

Paliperidone Palmitate USP/EP/BP

Paliperidone palmitateQ: What is Paliperidone palmitate Q: What is the CAS Number of Paliperidone palmitate Q: What is the storage condition of Paliperidone palmitate Q: What are the applications of Paliperidone palmitate

Paliperidone Palmitate Benzisoxazole Impurity

199739-10-1

C39H57FN4O4

Heterocycles

Intermediates & Fine Chemicals

Pharmaceuticals

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