ChemicalBook > CAS DataBase List > PyridiniuM, 4-[2-[[(6R,7R)-2-carboxy-7-[[(2Z)-2-(ethoxyiMino)-2-[5-(phosphonoaMino)-1,2,4-thiadiazol-3-yl]acetyl]aMino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]thio]-4-thiazolyl]-1-Methyl-, inner salt

PyridiniuM, 4-[2-[[(6R,7R)-2-carboxy-7-[[(2Z)-2-(ethoxyiMino)-2-[5-(phosphonoaMino)-1,2,4-thiadiazol-3-yl]acetyl]aMino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]thio]-4-thiazolyl]-1-Methyl-, inner salt

Product Name
PyridiniuM, 4-[2-[[(6R,7R)-2-carboxy-7-[[(2Z)-2-(ethoxyiMino)-2-[5-(phosphonoaMino)-1,2,4-thiadiazol-3-yl]acetyl]aMino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]thio]-4-thiazolyl]-1-Methyl-, inner salt
CAS No.
229016-73-3
Chemical Name
PyridiniuM, 4-[2-[[(6R,7R)-2-carboxy-7-[[(2Z)-2-(ethoxyiMino)-2-[5-(phosphonoaMino)-1,2,4-thiadiazol-3-yl]acetyl]aMino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]thio]-4-thiazolyl]-1-Methyl-, inner salt
Synonyms
TAK 599 HCL;PPI0903freeacid;TAK-599 free acid;ceftoreline fosimil;Ceftaroline Impurity7;Ceftaroline inner salt;Ceftaroline Fosamil Impurity 4;Ceftaroline FosaMil Inner salt;Ceftaroline Fosamil Impurity L;PyridiniuM,4-[2-[[(6R,7R)-2-carboxy-7-[[(2Z)-2-(ethoxyiMino)-2-[5-(phosphonoaMino)-1,2,4-thiadiazol-3Chemicalbook-yl]acetyl]aMino]-8-oxo-5-thia-1-azabicyclo
CBNumber
CB92628317
Molecular Formula
C22H21N8O8PS4
Formula Weight
684.67
MOL File
229016-73-3.mol
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

TRC
Product number
C243970
Product name
CeftarolineFosamilInnersalt
Packaging
10mg
Price
$13750
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
CCH0012998
Product name
4-[2-[[(6R,7R)-2-CARBOXY-7-[[(2Z)-2-(ETHOXYIMINO)-2-[5-(PHOSPHONOAMINO)-1,2,4-THIADIAZOL-3-YL]ACETYL]AMINO]-8-OXO-5-THIA-1-AZABICYCLO-[4.2.0]-OCT-2-EN-3-YL]THIO]-4-THIAZOLYL]-1-METHYL-PYRIDINIUM INNER SALT
Purity
95.00%
Packaging
5MG
Price
$495.2
Updated
2021/12/16
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PyridiniuM, 4-[2-[[(6R,7R)-2-carboxy-7-[[(2Z)-2-(ethoxyiMino)-2-[5-(phosphonoaMino)-1,2,4-thiadiazol-3-yl]acetyl]aMino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]thio]-4-thiazolyl]-1-Methyl-, inner salt Chemical Properties,Usage,Production

Uses

Ceftaroline Fosamil is a cephalosporin antibiotic. It is active against methicillin-resistant Staphylococcus aureus (MRSA) and Gram-positive bacteria.

Definition

ChEBI: A cephalosporin that is the N-phospho prodrug of ceftaroline. A broad-spectrum antibiotic, it is active against methicillin-resistant Staphylococcus aureus (MRSA). It is used for the treatment of adults with acute bacterial kin and skin structure infections.

in vivo

Ceftaroline fosamil inner salt (s.c.) shows protective effects against experimental systemic infection caused by S. aureus N133 in mice, with ED50s of 1.60-2.37 mg/kg[1].
Ceftaroline fosamil inner salt (10 mg/kg; s.c.) disappeares rapidly and converts smoothly into T-91825 in blood of rats and monkeys[1].

IC 50

β-lactam

PyridiniuM, 4-[2-[[(6R,7R)-2-carboxy-7-[[(2Z)-2-(ethoxyiMino)-2-[5-(phosphonoaMino)-1,2,4-thiadiazol-3-yl]acetyl]aMino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]thio]-4-thiazolyl]-1-Methyl-, inner salt Preparation Products And Raw materials

Raw materials

Preparation Products

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PyridiniuM, 4-[2-[[(6R,7R)-2-carboxy-7-[[(2Z)-2-(ethoxyiMino)-2-[5-(phosphonoaMino)-1,2,4-thiadiazol-3-yl]acetyl]aMino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]thio]-4-thiazolyl]-1-Methyl-, inner salt Suppliers

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View Lastest Price from PyridiniuM, 4-[2-[[(6R,7R)-2-carboxy-7-[[(2Z)-2-(ethoxyiMino)-2-[5-(phosphonoaMino)-1,2,4-thiadiazol-3-yl]acetyl]aMino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]thio]-4-thiazolyl]-1-Methyl-, inner salt manufacturers

BOC Sciences
Product
Ceftaroline Fosamil 229016-73-3
Price
US $0.00/g
Min. Order
1g
Purity
≥98%
Supply Ability
1kg
Release date
2020-05-15
Career Henan Chemical Co
Product
PyridiniuM,4-[2-[[(6R,7R)-2-carboxy-7-[[(2Z)-2-(ethoxyiMino)-2-[5-(phosphonoaMino)-1,2,4-thiadiazol-3Chemicalbook-yl]acetyl]aMino]-8-oxo-5-thia-1-azabicyclo 229016-73-3
Price
US $1.00/g
Min. Order
1g
Purity
≥98%
Supply Ability
g/kg/Ton
Release date
2019-12-25

229016-73-3, PyridiniuM, 4-[2-[[(6R,7R)-2-carboxy-7-[[(2Z)-2-(ethoxyiMino)-2-[5-(phosphonoaMino)-1,2,4-thiadiazol-3-yl]acetyl]aMino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]thio]-4-thiazolyl]-1-Methyl-, inner saltRelated Search:

7 β - aMino - 3 - [4 - pyridyl - 2 - thiazole sulfur radical ] - 3 - cepheM - 4 - carboxylic acid Ceftaroline Fosamil Impurity 5 Ceftaroline IMP Ceftaroline Fosamil Impurity 7 Ceftolin Ceftaroline Impurity 2 Ceftaroline Fosamil Impurity 6 TAK 599 (Z)-2-(5-AMino-1,2,4-thiadiazol-3-yl)-2-ethoxyiMinoacetic acid 4-(4-Pyridinyl)thiazole-2-thiol Ceftaroline Fosamil Impurity 1 Ceftaroline Impurity 1 7 β - aMino - 3 - [4 - pyridyl - 2 - thiazole sulfur radical ] - 3 - cepheM - 4 - carboxylic acid ·2HCl Sodium 1-(2-hydroxyethyl)-1H-tetrazol-5-ylthiolate Cefololin 3-position side chain Cefololin 7-position side chain Cefololin 3-position side chain Lorraine cephalosporin side chain ester 7

  • 4-[2-[[(6R,7R)-2-Carboxy-7-[[(2Z)-(ethoxyimino)[5-(phosphonoamino)-1,2,4-thiadiazol-3-yl]acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]thio]-4-thiazolyl]-1-methylpyridinium inner salt
  • 4-[2-[[(6R,7R)-2-Carboxy-7-[[(2Z)-2-(ethoxyimino)-2-[5-(phosphonoamino)-1,2,4-thiadiazol-3-yl]acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]thio]-4-thiazolyl]-1-methyl-pyridinium Inner Salt
  • PyridiniuM, 4-[2-[[(6R,7R)-2-carboxy-7-[[(2Z)-2-(ethoxyiMino)-2-[5-(phosphonoaMino)-1,2,4-thiadiazol-3-yl]acetyl]aMino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]thio]-4-thiazolyl]-1-Methyl-, inner salt
  • Ceftaroline FosaMil Inner salt
  • Ceftaroline Fosamil Impurity 4
  • Ceftaroline Impurity7
  • TAK 599 HCL
  • PyridiniuM,4-[2-[[(6R,7R)-2-carboxy-7-[[(2Z)-2-(ethoxyiMino)-2-[5-(phosphonoaMino)-1,2,4-thiadiazol-3Chemicalbook-yl]acetyl]aMino]-8-oxo-5-thia-1-azabicyclo
  • Ceftaroline Fosamil Impurity 11/ Ceftaroline Fosamil Inner salt/4-[2-[[(6R,7R)-2-Carboxy-7-[[(2Z)-2-(ethoxyimino)-2-[5-(phosphonoamino)-1,2,4-thiadiazol-3-yl]acetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]thio]-4-thiazolyl]-1-methyl-pyridinium Inner Salt
  • Ceftaroline Fosamil Impurity L
  • ceftoreline fosimil
  • PPI0903freeacid
  • TAK-599 free acid
  • Ceftaroline inner salt
  • 229016-73-3
  • C22H21N8O8PS4