ChemicalBook > CAS DataBase List > GDC-0810(ARN-810)

GDC-0810(ARN-810)

Product Name
GDC-0810(ARN-810)
CAS No.
1365888-06-7
Chemical Name
GDC-0810(ARN-810)
Synonyms
RG6046;RG 6046;ARN-810;CS-2080;RG-6046;GDC-0810;Brilanestrant);GDC-0810(ARN-810);ARN-810;BRILANESTRANT;GDC-0810 (Brilanestrant)
CBNumber
CB93040499
Molecular Formula
C26H20ClFN2O2
Formula Weight
446.9
MOL File
1365888-06-7.mol
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GDC-0810(ARN-810) Property

Boiling point:
622.8±55.0 °C(Predicted)
Density 
1.342±0.06 g/cm3(Predicted)
solubility 
DMSO:89.0(Max Conc. mg/mL);199.15(Max Conc. mM)
Ethanol:89.0(Max Conc. mg/mL);199.15(Max Conc. mM)
form 
A solid
pka
13.94±0.40(Predicted)
color 
White to off-white
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Cayman Chemical
Product number
29595
Product name
ARN810
Packaging
5mg
Price
$120
Updated
2024/03/01
Cayman Chemical
Product number
29595
Product name
ARN810
Packaging
25mg
Price
$510
Updated
2024/03/01
Cayman Chemical
Product number
29595
Product name
ARN810
Packaging
1mg
Price
$36
Updated
2024/03/01
Cayman Chemical
Product number
29595
Product name
ARN810
Packaging
10mg
Price
$223
Updated
2024/03/01
TRC
Product number
B677393
Product name
Brilanestrant
Packaging
10mg
Price
$210
Updated
2021/12/16
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GDC-0810(ARN-810) Chemical Properties,Usage,Production

Uses

Brilanestrant is an orally bioavailable Selective Estrogen Receptor Degrader (SERD) that demonstrates robust activity in tamoxifen-resistant breast cancer xenografts. GDC-0810 functions by binding to the estrogen receptor, inducing a conformational change resulting in the degradation of the receptor. GDC-0810 or ARN-810 demonstrates robust activity in models of tamoxifen-sensitive and tamoxifen-resistant breast cancer, and is currently in clinical trials in women with locally advanced or metastatic estrogen receptor-positive breast cancer.

GDC-0810(ARN-810) Preparation Products And Raw materials

Raw materials

Preparation Products

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GDC-0810(ARN-810) Suppliers

Shanghai Boyle Chemical Co., Ltd.
Tel
Fax
86-21-57758967
Email
sales@boylechem.com
Country
China
ProdList
2923
Advantage
55
Chembest Research Laboratories Limited
Tel
+86-21-20908456
Fax
021-58180499
Email
sales@BioChemBest.com
Country
China
ProdList
6008
Advantage
61
WUHAN SUN-SHINE BIO-TECHNOLOGY Co., Ltd.
Tel
17702719238 17702719238
Email
sales@sun-shinechem.com
Country
China
ProdList
950
Advantage
64
Haoyuan Chemexpress Co., Ltd.
Tel
021-58950125
Fax
(86) 21-58955996
Email
info@chemexpress.com
Country
China
ProdList
7553
Advantage
61
Shanghai Aladdin Bio-Chem Technology Co.,LTD
Tel
400-400-6206333 18521732826
Fax
021-50323701
Email
market@aladdin-e.com
Country
China
ProdList
25009
Advantage
65
Shanghai Lollane Biological Technology Co.,Ltd.
Tel
021-52996696,15000506266 15000506266
Fax
+86-21-52996696
Country
China
ProdList
4335
Advantage
55
Guangzhou QiYun Biotechnology Co., Ltd.
Tel
020-61288194 61288195
Fax
020-61288700
Email
505721671@qq.com
Country
China
ProdList
3868
Advantage
58
ShangHai Biochempartner Co.,Ltd
Tel
17754423994 17754423994
Fax
QQ:2853530913
Email
2853530910@QQ.com
Country
China
ProdList
8014
Advantage
62
Beijing Solarbio Science & Tecnology Co., Ltd.
Tel
010-50973130 4009686088
Email
3193328036@qq.com
Country
China
ProdList
29786
Advantage
68
Amadis Chemical Company Limited
Tel
571-89925085
Fax
0086-571-89925065
Email
sales@amadischem.com
Country
China
ProdList
131980
Advantage
58

1365888-06-7, GDC-0810(ARN-810)Related Search:


  • (E)-3-(4-((E)-2-(2-CHLORO-4-FLUOROPHENYL)-1-(1H-INDAZOL-5-YL)BUT-1-EN-1-YL)PHENYL)ACRYLIC ACID
  • GDC-0810 (Brilanestrant)
  • GDC-0810(ARN-810)
  • GDC-0810
  • (E)-3-[4-[(E)-2-(2-Chloro-4-fluorophenyl)-1-(1H-indazol-5-yl)but-1-en-1-yl]phenyl]-2-propenoic acid
  • ARN-810
  • ARN-810;BRILANESTRANT
  • CS-2080
  • Brilanestrant)
  • GDC0810; GDC 0810; GDC-0810; ARN810; ARN 810; ARN-810; RG6046; RG-6046; RG 6046; BRILANESTRANT
  • RG 6046
  • RG6046
  • RG-6046
  • Brilanestrant (GDC-0810, ARN-810)
  • 2-Propenoic acid, 3-[4-[(1E)-2-(2-chloro-4-fluorophenyl)-1-(1H-indazol-5-yl)-1-buten-1-yl]phenyl]-, (2E)-
  • ARN810,inhibit,Estrogen Receptor/ERR,ARN 810,Brilanestrant,Inhibitor
  • Brilanestrant (GDC-0810)
  • 1365888-06-7
  • C26H20ClFN2O2