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DILEVALOL

Product Name
DILEVALOL
CAS No.
75659-07-3
Chemical Name
DILEVALOL
Synonyms
Levadil;Unicard;Dilevaol;Dilevalon;Sch-19927;DILEVALOL;Dilevalolum;DILEVALOL HCL;(R,R)-Labetalol;Dilevalolum [latin]
CBNumber
CB9773028
Molecular Formula
C19H24N2O3
Formula Weight
328.41
MOL File
75659-07-3.mol
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DILEVALOL Property

Boiling point:
552.7±50.0 °C(Predicted)
Density 
1.200±0.06 g/cm3(Predicted)
pka
8.21±0.31(Predicted)
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Biosynth Carbosynth
Product number
FL24822
Product name
Dilevalol
Packaging
10mg
Price
$145
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0019482
Product name
2-HYDROXY-5-((R)-1-HYDROXY-2-(((R)-4-PHENYLBUTAN-2-YL)AMINO)ETHYL)BENZAMIDE
Purity
95.00%
Packaging
5MG
Price
$498.88
Updated
2021/12/16
Biosynth Carbosynth
Product number
FL24822
Product name
Dilevalol
Packaging
50mg
Price
$507.5
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0019482
Product name
2-HYDROXY-5-((R)-1-HYDROXY-2-(((R)-4-PHENYLBUTAN-2-YL)AMINO)ETHYL)BENZAMIDE
Purity
95.00%
Packaging
1G
Price
$3104.85
Updated
2021/12/16
Crysdot
Product number
CD12036144
Product name
2-Hydroxy-5-((R)-1-hydroxy-2-(((R)-4-phenylbutan-2-yl)amino)ethyl)benzamide
Purity
95+%
Packaging
1g
Price
$1583
Updated
2021/12/16
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DILEVALOL Chemical Properties,Usage,Production

Description

Dilevalol is a "dual-mechanism" antihypertensive reportedly suitable for a wide range of patients. Its partial beta2-agonist action is expected to induce vasodilation, whereas its beta1-antagonist component may protect against stress-induced hemodynamic charges without altering the cardiac output. Dilevalol is the R,R-isomer of labetalol.

Originator

Schering Plough (USA)

Uses

Specific competitive antagonist at both α-and β-adrenergic receptor sites. Antihypertensive.

Uses

(R,R)-Labetalol is a specific competitive antagonist at both α-and β-adrenergic receptor sites. (R,R)-Labetalol is used as an antihypertensive.

Definition

ChEBI: (R,R)-labetalol is a 2-hydroxy-5-{1-hydroxy-2-[(4-phenylbutan-2-yl)amino]ethyl}benzamide that has 1R,2R-configuration. It is a conjugate base of a dilevalol(1+).

brand name

Levadil; Dilevalon

World Health Organization (WHO)

Dilevalol, a beta-adrenoreceptor antagonist, was introduced into medicine in 1989 for the treatment of hypertension. Shortly afterwards, its use became associated with isolated cases of hepatic toxicity. Although few cases were reported, the manufacturer discontinued sales in Japan and Portugal, the only countries where the drug was marketed, and withdrew applications for registration elsewhere.

DILEVALOL Preparation Products And Raw materials

Raw materials

Preparation Products

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DILEVALOL Suppliers

J & K SCIENTIFIC LTD.
Tel
010-82848833 400-666-7788
Fax
86-10-82849933
Email
jkinfo@jkchemical.com
Country
China
ProdList
96815
Advantage
76
LGM Pharma
Tel
1-(800)-881-8210
Fax
615-250-9817
Email
inquiries@lgmpharma.com
Country
United States
ProdList
2123
Advantage
70
Chemsky (shanghai) International Co.,Ltd
Tel
021-50135380
Email
shchemsky@sina.com
Country
China
ProdList
15402
Advantage
60
Shanghai Hekang Biotechnology Co., Ltd.
Tel
18939837085
Fax
2880152141(QQ)
Email
youchemicals@gmail.com
Country
China
ProdList
1830
Advantage
55
Shenzhen Polymeri Biochemical Technology Co., Ltd.
Tel
+86-400-002-6226 +86-13028896684;
Email
sales@rrkchem.com
Country
China
ProdList
57412
Advantage
58
TargetMol Chemicals Inc.
Tel
+1-781-999-5354 +1-00000000000
Email
marketing@targetmol.com
Country
United States
ProdList
32165
Advantage
58
Energy Chemical
Tel
021-58432009 400-005-6266
Fax
021-58436166
Email
marketing@energy-chemical.com
Country
China
ProdList
44918
Advantage
58
QUALITY CONTROL SOLUTIONS LTD.
Tel
0755-66853366; 13670046396
Email
ORDERS@QCSRM.COM
Country
China
ProdList
24326
Advantage
58
TargetMol Chemicals Inc.
Tel
4008200310
Email
marketing@tsbiochem.com
Country
China
ProdList
24647
Advantage
58
Hubei Ruinuo Pharmaceutical Technology Co., Ltd
Tel
13165688766
Fax
0714-5316360
Email
3008058303@qq.com
Country
China
ProdList
3009
Advantage
58

75659-07-3, DILEVALOLRelated Search:


  • 2-Hydroxy-5-[(R)-1-hydroxy-2-[[(R)-1-methyl-3-phenylpropyl]amino]ethyl]benzamide
  • Sch-19927
  • (-)-5-((1R)-1-Hydroxy-2-((1R)-1-methyl-3-phenylpropylamino)ethyl)salicylamid [iupac]
  • (R,R)-Labetalol
  • 2-Hydroxy-5-((1R)-1-hydroxy-2-(((1R)-1-methyl-3-phenylpropyl)amino)ethyl)benzamide
  • Benzamide, 2-hydroxy-5-((1R)-1-hydroxy-2-(((1R)-1-methyl-3-phenylpropyl)amino)ethyl)-
  • DILEVALOL
  • DILEVALOL HCL
  • Dilevaol
  • Dilevalon
  • Levadil
  • Unicard
  • 2-Hydroxy-5-((R)-1-hydroxy-2-(((R)-4-phenylbutan-2-yl)aMino)ethyl)benzaMide
  • Benzamide, 2-hydroxy-5-(1-hydroxy-2-((1-methyl-3-phenylpropyl)amino)ethyl)-, (R-(R*,R*))-
  • Dilevalolum
  • Dilevalolum [latin]
  • 75659-07-3
  • Amines
  • Aromatics
  • Chiral Reagents
  • Intermediates & Fine Chemicals
  • Pharmaceuticals