Napirimus Chemical Properties

Boiling point:

536.6±35.0 °C(Predicted)

Density 

1.25±0.1 g/cm3(Predicted)

solubility 

DMSO: Slightly soluble: 0.1-1 mg/ml

pka

3.83±0.41(Predicted)

Napirimus Usage And Synthesis

Description

Napirimus is an immunosuppressant.1 It is efficacious and preventative in a rat model of polyarthritis induced by complete Freund’s adjuvant when administered at doses of 200 and 100 mg/kg, respectively. Napirimus is 50 and 90% protective against experimental autoimmune encephalomyelitis (EAE), previously known as allergic encephalomyelitis, in rats when administered at doses of 100 and 400 mg/kg, respectively.WARNING This product is not for human or veterinary use.

References

[1] Peptides having immunostimulating properties and pharmaceutical compositions containing them[J]. Vaccine, 1983, 1 1: Page 52. DOI: 10.1016/0264-410x(83)90037-3

Napirimus(70696-66-1)Related Product Information

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• Napirimus
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