Varenicline-d4 Chemical Properties

storage temp. 

Store at -20°C

solubility 

Water: 0.0877 mg/mL

form 

A solid

Water Solubility 

Water: 0.0877 mg/mL

Varenicline-d4 Usage And Synthesis

Description

Varenicline-d₄ is intended for use as an internal standard for the quantification of varenicline by GC- or LC-MS. Varenicline is a full agonist of α7 subunit-containing neuronal nicotinic acetylcholine receptors (nAChRs; EC₅₀ = 18 μM) and a partial agonist of α4β2 subunit-containing nAChRs (EC₅₀ = 2.3 μM). Formulations containing varenicline have been used as aids in smoking cessation.

Varenicline-d4(2183239-01-0)Related Product Information

• Varenicline Impurity 18
• (+/-)-2,2,2-trifluoro-1-(4-nitro-10-aza-tricyclo[6.3.1.02,7]dodeca-2(7),3,5-trien-10-yl)-ethanone
• Hydroxy Varenicline
• Varenicline Impurity 8
• Varenicline Impurity 5
• Hydroxy Varenicline N-Trifluoroacetate
• Varenicline Impurity 3
• Varenicline Impurity 6
• Varenicline Impurity 17
• N-Methyl Varenicline
• 5,9-Methanoimidazo[4,5-h][3]benzazepine,1,5,6,7,8,9-hexahydro-(9CI)
• Varenicline-13C2,15N2
• 7,8,9,10-Tetrahydro-8-(trifluoroacetyl)-6,10-methano-6H-pyrazino[2,3-h][3]benzazepine (N-(Trifluoroacetyl)varenicline)
• Varenicline Impurity 13 HCl
• N-Acetyl Varenicline
• N-Formyl Varenicline
• 2,3,4,5-Tetrahydro-3-(trifluoroacetyl)-1,5-methano-1H-3-benzazepine-7,8-diamine
• 2,3,4,5-Tetrahydro-7,8-dinitro-3-(trifluoroacetyl)-1,5-methano-1H-3-benzazepine