N-Acetyl Varenicline Chemical Properties

Boiling point:

481.2±45.0 °C(Predicted)

Density 

1.294±0.06 g/cm3(Predicted)

solubility 

Chloroform (Slightly), Methanol (Slightly)

form 

Solid

pka

1.56±0.20(Predicted)

color 

Light Orange to Orange

N-Acetyl Varenicline Usage And Synthesis

Uses

1-(6,7,9,10-Tetrahydro-6,10-methano-8H-pyrazino[2,3-h][3]benzazepin-8-yl)ethanone is related to its parent compound N-Formyl Varenicline (F701650), which is a metabolite of Varenicline and metabolite M5. Also, it is derived from Varenicline Tartrate (V098490), which is a nicotinic α4β2 acetylcholine receptor partial agonist and used to aid in smoking cessation (1,2,3,4).

N-Acetyl Varenicline(1213781-59-9)Related Product Information

• Varenicline Impurity 8
• Hydroxy Varenicline
• Varenicline Impurity 5
• (+/-)-2,2,2-trifluoro-1-(4-nitro-10-aza-tricyclo[6.3.1.02,7]dodeca-2(7),3,5-trien-10-yl)-ethanone
• Varenicline Impurity 17
• N-Methyl Varenicline
• 5,9-Methanoimidazo[4,5-h][3]benzazepine,1,5,6,7,8,9-hexahydro-(9CI)
• Varenicline-13C2,15N2
• 7,8,9,10-Tetrahydro-8-(trifluoroacetyl)-6,10-methano-6H-pyrazino[2,3-h][3]benzazepine (N-(Trifluoroacetyl)varenicline)
• Varenicline Impurity 13 HCl
• N-Formyl Varenicline
• Varenicline-d4
• 2,3,4,5-Tetrahydro-3-(trifluoroacetyl)-1,5-methano-1H-3-benzazepine-7,8-diamine
• 2,3,4,5-Tetrahydro-7,8-dinitro-3-(trifluoroacetyl)-1,5-methano-1H-3-benzazepine