Basic information Safety Supplier Related

4-HYDROXY-8-METHYLQUINOLINE-3-CARBOXYLIC ACID ETHYL ESTER

Basic information Safety Supplier Related

4-HYDROXY-8-METHYLQUINOLINE-3-CARBOXYLIC ACID ETHYL ESTER Basic information

Product Name:
4-HYDROXY-8-METHYLQUINOLINE-3-CARBOXYLIC ACID ETHYL ESTER
Synonyms:
  • ETHYL 4-HYDROXY-8-METHYL-3-QUINOLINECARBOXYLATE
  • ETHYL 4-HYDROXY-8-METHYLQUINOLINE-3-CARBOXYLATE
  • 4-HYDROXY-8-METHYLQUINOLINE-3-CARBOXYLIC
  • 4-HYDROXY-8-METHYLQUINOLINE-3-CARBOXYLIC ACID ETHYL ESTER
  • 4-HYDROXY-8-METHYLQUINOLINE-3-CARBOXYLIC ETHYL ESTER
  • 2-ethyl-8-methyl-4-oxo-1H-quinoline-3-carboxylate
  • 3-Quinolinecarboxylic acid, 4-hydroxy-8-methyl-, ethyl ester
  • Ethyl 8-methyl-4-oxo-1H-quinoline-3-carboxylate
CAS:
77156-75-3
MF:
C13H13NO3
MW:
231.25
Product Categories:
  • Quinoline&Isoquinoline
Mol File:
77156-75-3.mol
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4-HYDROXY-8-METHYLQUINOLINE-3-CARBOXYLIC ACID ETHYL ESTER Chemical Properties

Melting point:
271-274°(dec)
storage temp. 
Inert atmosphere,Room Temperature
CAS DataBase Reference
77156-75-3(CAS DataBase Reference)
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Safety Information

HazardClass 
IRRITANT
HS Code 
2933499090
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4-HYDROXY-8-METHYLQUINOLINE-3-CARBOXYLIC ACID ETHYL ESTER Usage And Synthesis

Synthesis

19146-73-7

77156-75-3

GENERAL METHOD: 2e-k (4 mmol) was dissolved in diphenyl ether with a catalytic amount of 2-chlorobenzoic acid and heated by microwave radiation at 250°C for 1-2 hours. After completion of the reaction, the reaction mixture was cooled, the precipitate 3e-k was collected by filtration and washed sequentially with hexane and water.

References

[1] Journal of Heterocyclic Chemistry, 2013, vol. 50, # SUPPL.1, p. E1-E8
[2] Nucleosides and Nucleotides, 1996, vol. 15, # 4, p. 889 - 898
[3] Medicinal Chemistry Research, 2016, vol. 25, # 9, p. 1861 - 1876
[4] Journal of Medicinal Chemistry, 2006, vol. 49, # 22, p. 6443 - 6450
[5] RSC Advances, 2014, vol. 4, # 12, p. 6254 - 6260

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