Basic information Safety Supplier Related

PALMITOYL-DL-CARNITINE CHLORIDE

Basic information Safety Supplier Related

PALMITOYL-DL-CARNITINE CHLORIDE Basic information

Product Name:
PALMITOYL-DL-CARNITINE CHLORIDE
Synonyms:
  • (+/-)-PALMITOYLCARNITINE CHLORIDE
  • PALMITOYL-DL-CARNITINE CHLORIDE
  • PALMITOYL-DL-CARNITINE HYDROCHLORIDE
  • PalMitoyl-DL-carnitine
  • DL-Palmitoylcarnitine chloride
  • 3-Carboxy-N,N,N-trimethyl-2-(palmitoyloxy)propan-1-aminium chloride
  • (+/-)-Palmitoylcarni
  • Palmitoyl-DL-carnitine chloride powder
CAS:
6865-14-1
MF:
C23H46ClNO4
MW:
436.07
Product Categories:
  • Lipid signaling
Mol File:
6865-14-1.mol
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PALMITOYL-DL-CARNITINE CHLORIDE Chemical Properties

storage temp. 
-20°C
solubility 
H2O: 25 mg/mL with heat or sonication
form 
powder
color 
white
biological source
synthetic (organic)
Water Solubility 
H2O: 25mg/mL (with he at or sonication)
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Safety Information

WGK Germany 
3
HS Code 
2923900090

MSDS

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PALMITOYL-DL-CARNITINE CHLORIDE Usage And Synthesis

Uses

DL-Palmitoylcarnitine (chloride) is a long-chain acylcarnitine with both intracellular and extracellular roles. Within the cell, palmitoylcarnitine is transported into mitochondria to deliver palmitate for fatty acid oxidation and energy production. Exogenously added DL-palmitoylcarnitine alters calcium mobilization in many cell types. It also affects endothelial and epithelial tight junctions, reducing resistance and increasing permeability while decreasing cell viability.

Uses

Palmitoyl-DL-carnitine chloride is a specific protein kinase C (PKC) inhibitor.

Uses

Palmitoyl-DL-carnitine chloride has been used to study its effect on inflammatory cytokines and calcium (Ca2+) influx, using in vitro models of prostate cancer.

Biochem/physiol Actions

Palmitoyl-DL-carnitine chloride is known to inhibit biofilm formation mediated by Pseudomonas aeruginosa and Escherichia coli. It is a phosphokinase C inhibitor.

in vivo

Palmitoylcarnitine (10 mg/kg, s.c., once daily for 28 days) induces insulin resistance and hyperinsulinemia, leading to glucose metabolism impairment in CD-1 mice[3]. Palmitoylcarnitine (50 mg/kg, s.c., single dose) reduces insulin sensitivity and induces glucose intolerance and metabolic dysfunction in CD-1 mice[3]. Palmitoylcarnitine (50 mg/kg, i.p., single dose) increases muscle long-chain acylcarnitine content and induces insulin resistance in CD-1 mice, characterized by hyperglycemia and reduced muscle glucose uptake[3].

Animal Model:Palmitoylcarnitine (HY-126357)-induced insulin resistance CD-1 mouse model[3]
Dosage:50 mg/kg (s.c. or i.p., single dose) or 10 mg/kg (s.c., long-term administration)
Administration:Intraperitoneal injection (i.p.), single dose; Continuously released for 24 hours via a subcutaneous osmotic minipump (s.c.)., single dose Subcutaneous osmotic minipump (s.c.), once daily for 28 days.
Result:Increased muscle long-chain acylcarnitine content, elevated blood glucose levels in both fasted and fed states, and decreased muscle glucose uptake (i.p.). Induced glucose intolerance, delayed energy metabolism shift, and reduced insulin sensitivity (s.c., single dose). induced insulin resistance and hyperinsulinemia, blocked insulin-mediated blood glucose reduction, increased blood lactate levels, and impaired glucose metabolism (s.c., long-term administration).

PALMITOYL-DL-CARNITINE CHLORIDESupplier

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