Basic information Safety Supplier Related

2-AMINO-6-CHLORO-9-(BETA-D-2-DEOXYRIBOFURANOSYL)PURINE

Basic information Safety Supplier Related

2-AMINO-6-CHLORO-9-(BETA-D-2-DEOXYRIBOFURANOSYL)PURINE Basic information

Product Name:
2-AMINO-6-CHLORO-9-(BETA-D-2-DEOXYRIBOFURANOSYL)PURINE
Synonyms:
  • 2-Amino-6-chloropurine-9-beta-D-(2'-deoxy)riboside
  • 2-AMINO-6-CHLOROPURINE-2'-DEOXYRIBOSIDE
  • 2-AMINO-6-CHLORO-9-(BETA-D-2-DEOXYRIBOFURANOSYL)PURINE
  • 2-AMINO-6-CHLOROPURINE-2'-DEOXY-D-RIBOFURANOSIDE
  • 2-Amino-6-chloro-9-(2'-deoxy-b-D-ribofuranosyl)purine
  • (2R,3S,5S)-5-(2-AMino-6-chloro-9H-purin-9-yl)-2-(hydroxyMethyl)tetrahydrofuran-3-ol
  • 2-Amino-6-chloro-9-(β-D-2-deoxyribofuranosyl)purine
  • 9H-Purin-2-amine, 6-chloro-9-(2-deoxy-β-D-erythro-pentofuranosyl)-
CAS:
120595-72-4
MF:
C10H12ClN5O3
MW:
285.69
Mol File:
120595-72-4.mol
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2-AMINO-6-CHLORO-9-(BETA-D-2-DEOXYRIBOFURANOSYL)PURINE Chemical Properties

storage temp. 
2-8°C
InChI
InChI=1/C10H12ClN5O3/c11-8-7-9(15-10(12)14-8)16(3-13-7)6-1-4(18)5(2-17)19-6/h3-6,17-18H,1-2H2,(H2,12,14,15)/t4-,5+,6+/s3
InChIKey
LEDIVMUMDVEFRG-FLEGHBDQNA-N
SMILES
N1(C=NC2C(Cl)=NC(N)=NC1=2)[C@H]1C[C@H](O)[C@@H](CO)O1 |&1:11,13,15,r|
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2-AMINO-6-CHLORO-9-(BETA-D-2-DEOXYRIBOFURANOSYL)PURINE Usage And Synthesis

Uses

2-Amino-6-chloropurine-9-beta-D-(2’-deoxy)riboside is a purine nucleoside analog. Purine nucleoside analogs have broad antitumor activity targeting indolent lymphoid malignancies. Anticancer mechanisms in this process rely on inhibition of DNA synthesis, induction of apoptosis, etc[1].

References

[1] Robak T, Robak P. Purine nucleoside analogs in the treatment of rarer chronic lymphoid leukemias. Curr Pharm Des. 2012;18(23):3373-88. DOI:10.2174/138161212801227005

2-AMINO-6-CHLORO-9-(BETA-D-2-DEOXYRIBOFURANOSYL)PURINESupplier

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