Basic information Safety Supplier Related

Metizolam

Basic information Safety Supplier Related

Metizolam Basic information

Product Name:
Metizolam
Synonyms:
  • Metizolam
  • 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine, 4-(2-chlorophenyl)-2-ethyl-
  • Metizolam (1.0 mg/mL in Methanol)
  • Metizolam 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine, 4-(2-chlorophenyl)-2-ethyl-
  • Metizolam, Desmethyletizolam
  • Metizolam solution
CAS:
40054-68-0
MF:
C16H13ClN4S
MW:
328.82
Mol File:
40054-68-0.mol
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Metizolam Chemical Properties

Melting point:
153-154 °C
Boiling point:
527.2±60.0 °C(Predicted)
Density 
1.46±0.1 g/cm3(Predicted)
storage temp. 
-10 to -25°C
solubility 
DMF: 15mg/mL; DMSO: 15mg/mL; DMSO:PBS (pH 7.2) (1:3): 0.25mg/mL
form 
A crystalline solid
pka
1.99±0.40(Predicted)
InChI
InChI=1S/C16H13ClN4S/c1-2-10-7-12-15(11-5-3-4-6-13(11)17)18-8-14-20-19-9-21(14)16(12)22-10/h3-7,9H,2,8H2,1H3
InChIKey
NQSSWDKQLVBUQN-UHFFFAOYSA-N
SMILES
N12C=NN=C1CN=C(C1=CC=CC=C1Cl)C1C=C(CC)SC=12
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Metizolam Usage And Synthesis

Uses

Metizolam can be used as reactant/reagent in in preparation of thienylazole and thienotriazolodiazepine compounds as cholecystokinin antagonists. It can also be used in biological study of platelet-activating factor antagonist.

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