Glucagon Receptor Antagonist I
Glucagon Receptor Antagonist I Basic information
- Product Name:
- Glucagon Receptor Antagonist I
- Synonyms:
-
- Glucagon Receptor Antagonist I
- N-[3-cyano-6-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-ethylbutanamide
- Butanamide, N-[3-cyano-6-(1,1-dimethylpropyl)-4,5,6,7-tetrahydrobenzo[b]thien-2-yl]-2-ethyl-
- hGCGR Antagonist
- CAS:
- 438618-32-7
- MF:
- C20H30N2OS
- MW:
- 346.53
- Mol File:
- 438618-32-7.mol
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Glucagon Receptor Antagonist I Chemical Properties
- Boiling point:
- 517.8±50.0 °C(Predicted)
- Density
- 1.07±0.1 g/cm3(Predicted)
- storage temp.
- Store at -20°C
- solubility
- DMSO: soluble
- form
- White crystalline solid.
- pka
- 13.46±0.40(Predicted)
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Glucagon Receptor Antagonist I Usage And Synthesis
Description
Glucagon receptor antagonist I is a competitive antagonist of the glucagon receptor (GCGR; IC50 = 181 nM). It blocks glucagon-induced glycogenolysis in primary human hepatocytes and isolated liver. Glucagon receptor antagonist I, at 50 mg/kg, reduces the increase in glucose levels observed after intraperitoneal administration of glucagon in humanized mice. Glucagon receptor antagonist inactive control does not prevent glucagon-mediated actions.
Glucagon Receptor Antagonist ISupplier
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