Altanserin
Altanserin Basic information
- Product Name:
- Altanserin
- Synonyms:
-
- 4(1H)-QUINAZOLINONE, 3-(2-(4-(4-FLUOROBENZOYL)-1-PIPERIDINYL)ETHYL)-2,3-DIHYDRO-2-THIOXO-
- ALTANSERIN
- ALTANSERIN HYDROCHLORIDE
- 3-[2-[4-(4-FLUOROBENZOYL)-1-PIPERIDINYL]ETHYL]-2,3-DIHYDRO-2-THIOXO-4(1H)-QUINAZOLINONE HYDROCHLORIDE
- 3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2,3-dihydro-2-thioxo-4(1H)-quinazolinone hydrate hydrochloride
- Altanserin hydrate hydrochloride
- 3-(2-(4-(4-Fluorobenzoyl)-1-piperidinyl)ethyl)-2,3-dihydro-2-thioxo-4(1H)-quinazolinonehydrochloride
- AltanserineHCl
- CAS:
- 76330-71-7
- MF:
- C22H22FN3O2S
- MW:
- 411.49
- EINECS:
- 278-422-1
- Product Categories:
-
- Serotonin receptor
- Mol File:
- 76330-71-7.mol
More
Less
Altanserin Chemical Properties
- storage temp.
- 2-8°C
- solubility
- DMSO: >5mg/mL
- form
- solid
- color
- White to light yellow
- InChI
- 1S/C22H22FN3O2S.ClH.H2O/c23-17-7-5-15(6-8-17)20(27)16-9-11-25(12-10-16)13-14-26-21(28)18-3-1-2-4-19(18)24-22(26)29;;/h1-8,16H,9-14H2,(H,24,29);1H;1H2
- InChIKey
- MFGBKMPKRJCLPK-UHFFFAOYSA-N
- SMILES
- O.Cl.Fc1ccc(cc1)C(=O)C2CCN(CC2)CCN3C(=S)Nc4ccccc4C3=O
More
Less
More
Less
Altanserin Usage And Synthesis
Chemical Properties
Yellowish solid
Uses
Serotonin antagonist.
Uses
Altanserin Hydrochloride is a useful intermediate for organic synthesis.
Definition
ChEBI: Altanserin is a member of quinazolines.
Biological Activity
Potent and selective 5-HT 2A receptor antagonist (K i values are 0.13, 4.55, 40, 62 and 1570 nM at 5-HT 2A , α 1 , 5-HT 2C , D 2 and 5-HT 1A respectively). Centrally active following systemic administration in vivo .
AltanserinSupplier
3B Pharmachem (Wuhan) International Co.,Ltd.
- Tel
- 821-50328103-801 18930552037
- 3bsc@sina.com
LGM Pharma
- Tel
- 1-(800)-881-8210
- inquiries@lgmpharma.com
Shanghai T&W Pharmaceutical Co., Ltd.
- Tel
- +86 21 61551611
Shanghai YuanYe Biotechnology Co., Ltd.
- Tel
- 021-61312847; 18021002903
- 3008007409@qq.com
Tianjin Kailiqi Biotechnology Co., Ltd.
- Tel
- 15076683720
- klq@cw-bio.com