3-MERCAPTO-3-METHYL-BUTYRYL-TYR(ME)-PHE-GLN-ASN-CYS-PRO-ARG-GLY-NH2 Chemical Properties

Density 

1.50±0.1 g/cm3(Predicted)

RTECS 

MB7547500

storage temp. 

−20°C

solubility 

H2O: soluble1mg/mL, clear, colorless

pka

12.85±0.70(Predicted)

form 

Solid

Water Solubility 

Soluble to 2 mg/ml in water

Sequence

{Pmp}-{Tyr(Me)}-Phe-Gln-Asn-Cys-Pro-Arg-Gly-NH2 (Disulfide bond: Pmp1-Cys6) (Pmp=β-Mercapto-β,β-cyclopentamethylene-propionic acid)

Safety Information

Hazard Codes 

Xn

Risk Statements 

20

Safety Statements 

36

WGK Germany 

3

MSDS

• Language:English Provider:SigmaAldrich

3-MERCAPTO-3-METHYL-BUTYRYL-TYR(ME)-PHE-GLN-ASN-CYS-PRO-ARG-GLY-NH2 Usage And Synthesis

Uses

(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin (SKF 100273) is a vasopressin V1 receptor selective antagonist[1].

storage

Store at -20°C

References

[1] Arai Y, et al. New topics in vasopressin receptors and approach to novel drugs: research and development of conivaptan hydrochloride (YM087), a drug for the treatment of hyponatremia. J Pharmacol Sci. 2009 Jan;109(1):53-9. DOI:10.1254/jphs.08r17fm

3-MERCAPTO-3-METHYL-BUTYRYL-TYR(ME)-PHE-GLN-ASN-CYS-PRO-ARG-GLY-NH2(73168-24-8)Related Product Information

• BETA-MERCAPTO-BETA,BETA-CYCLOPENTAMETHYLENE-PROPIONYL-TYR(ET)-PHE-VAL-ASN-CYS-PRO-ARG-OH
• BETA-MERCAPTO-BETA,BETA-CYCLOPENTAMETHYLENE-PROPIONYL-D-ILE-PHE-ILE-ASN-CYS-PRO-ARG-ALA-NH2
• BETA-MERCAPTO-BETA,BETA-CYCLOPENTAMETHYLENE-PROPIONYL-TYR(ET)-PHE-VAL-ASN-CYS-PRO-ARG-NH2
• BETA-MERCAPTO-BETA,BETA-CYCLOPENTAMETHYLENE-PROPIONYL-D-ILE-PHE-ILE-ASN-CYS-PRO-ARG-GLY-NH2
• (D(CH2)(5/1),D-TYR(ET)2,VAL4,ARG8,DES-GLY9)-VASOPRESSIN
• (d(CH?)?1,D-Phe2,Ile?,Ala-NH??)-Vasopressin
• METHYL PENTYL DISULPHIDE
• Cyclohexyl mercaptan
• 2-METHYL-2-PENTANETHIOL
• 3-(4-METHOXYPHENYL)PROPIONAMIDE
• 3-MERCAPTO-3-METHYL-BUTYRYL-TYR(ME)-PHE-GLN-ASN-CYS-PRO-ARG-GLY-NH2,3-Mercapto-3-methyl-butyryl-Tyr(Me)-Phe-Gln-Asn-Cys-Pro-Arg-Gly-NH2, (Disulfide bond)
• N-OCTYL-ETHYLENE-1,2-DIAMINE
• (ARG8)-VASOPRESSIN (4-9)
• 3-MERCAPTO-3-METHYL-BUTYRYL-TYR(ME)-PHE-GLN-ASN-CYS-PRO-ARG-GLY-NH2
• 3-ETHYL-3-PENTANETHIOL
• N-(4-Methoxyphenethyl)acetamide
• isopropyl propyl disulphide
• VASOPRESSIN, [PHENYLALANYL-3,4,5-3H]-D(CH-2-)-5-TYRME-[3H]-AVP