enalapril sodium salt
enalapril sodium salt Basic information
- Product Name:
- enalapril sodium salt
- Synonyms:
-
- Enalapril sodium
- enalapril sodium salt
- (-)-Enalapril sodium
- CAS:
- 149404-21-7
- MF:
- C20H29N2NaO5
- MW:
- 400.45
- Mol File:
- 149404-21-7.mol
enalapril sodium salt Usage And Synthesis
Uses
Enalapril (MK-421) sodium is an angiotensin-converting enzyme (ACE) inhibitor, can be used for hypertensive diseases research[1][2].
in vivo
Enalapril sodium (intraperitoneal injection, 0.03 mg/kg, once) reduces infarct volume due to middle cerebral artery occlusion and lower or higher doses are ineffective in Male NMRI mice[4].
| Animal Model: | Male NMRI mice 20-40 g[4] |
| Dosage: | 0.03 mg/kg |
| Administration: | Intraperitoneal injection; once |
| Result: | Reduced the area of middle cerebral artery infarction in mice at 0.03 mg/kg. |
References
[1] Serge Sicouri, et al. Antiarrhythmic effects of losartan and enalapril in canine pulmonary vein sleeve preparations. J Cardiovasc Electrophysiol. 2011 Jun;22(6):698-705. DOI:10.1111/j.1540-8167.2010.01972.x
[2] Rokhsareh Meamar, et al. Enalapril protects endothelial cells against induced apoptosis in Alzheimer's disease. J Res Med Sci. 2013 Mar;18(Suppl 1):S1-5. PMID:23961275
[3] Talita A Cunha, et al. Effect of stearic acid on enalapril stability and dissolution from multiparticulate solid dosage forms. AAPS PharmSciTech. 2013 Sep;14(3):1150-7. DOI:10.1208/s12249-013-0006-6
[4] A Ravati, et al. Enalapril and moexipril protect from free radical-induced neuronal damage in vitro and reduce ischemic brain injury in mice and rats. Eur J Pharmacol. 1999 May 28;373(1):21-33. DOI:10.1016/s0014-2999(99)00211-3
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