Basic information Safety Supplier Related

GITOXIGENIN

Basic information Safety Supplier Related

GITOXIGENIN Basic information

Product Name:
GITOXIGENIN
Synonyms:
  • 16β-Hydroxydigitoxigenin, 3β,14,16β-Trihydroxy-5β,20(22)-cardenolide, 5β,20(22)-Cardenolide-3β,14,16β-triol, 3β,14,16β,21-Tetrahydroxy-20(22)-norcholenic acid lactone
  • 3β,14,16β-Trihydroxy-5β,14β-card-20(22)-enolide
  • Gitoxigenin,98%
  • 3β,14,16β,21-Tetrahydroxy-20(22)-norcholenic acid lactone
  • 3β,14,16β-Trihydroxy-5β,20(22)-cardenolide
  • 5β,20(22)-Cardenolide-3β,14,16β-triol
  • 3,14,16-trihydroxy-,(3-beta,5-beta,16-beta)-card-20(22)-enolid
  • 3-beta,14,16-beta-trihydroxy-5-beta-card-20(22)-enolid
CAS:
545-26-6
MF:
C23H34O5
MW:
390.51
EINECS:
208-886-2
Mol File:
545-26-6.mol
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GITOXIGENIN Chemical Properties

Melting point:
~230 °C
Boiling point:
435.71°C (rough estimate)
Density 
1.0639 (rough estimate)
refractive index 
1.6120 (estimate)
storage temp. 
−20°C
pka
14.56±0.70(Predicted)
Merck 
13,4445
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Safety Information

Hazard Codes 
T
Risk Statements 
23/24/25
Safety Statements 
36/37/39-45
RIDADR 
UN 1544 6.1/PG 1
WGK Germany 
3
RTECS 
FH5391000
10
HazardClass 
6.1(b)
PackingGroup 
III

MSDS

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GITOXIGENIN Usage And Synthesis

Chemical Properties

light yellow flakes

Uses

Gitoxigenin is a related compound of Digitoxigenin, which has been used in a study to assess its stereochemical effects in cancer cytotoxicity. Digitoxigenin has also been used in a study to investigate the advantage of gold(I)-catalyzed glycosidation of glycosyl o-alkyl benzoates to assemble digitoxin.

Definition

ChEBI: Gitoxigenin is a 3beta-hydroxy steroid, a 14beta-hydroxy steroid and a 16beta-hydroxy steroid. It derives from a hydride of a 5beta-cardanolide.

Biochem/physiol Actions

Structure-activity relationships for 16β-substituted digitoxigenins as inhibitors of Na+/K+ ATPases.

Purification Methods

Recrystallisation of gitoxigenin from aqueous EtOH produces plates of the sesquihydrate which dehydrate on drying at 100o in vacuo. It also recrystallises from Me2CO/MeOH and from EtOAc (the crystals contain 1 mol of EtOAc) with [] D +24.8o (c 1, dioxane). It has UV with max at 310, 485 and 520nm in 96% H2SO4. On heating with ethanolic HCl it yields digitaligenin with loss of H2O. [Smith J Chem Soc 23 1931, Beilstein 8 IV 2456.]

GITOXIGENINSupplier

Meryer (Shanghai) Chemical Technology Co., Ltd.
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Shanghai Tauto Biotech Co., Ltd.
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Chengdu Push Bio-Technology Co., Ltd.
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028-85370565-229 18080489829
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Shenzhen Botel Biotechnology Co. Ltd.
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Hangzhou Synstar pharmaceutical Technology CO.,Ltd
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0571-85361029
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