MRS 1706 Chemical Properties

Density 

1.293±0.06 g/cm3(Predicted)

storage temp. 

Sealed in dry,2-8°C

solubility 

DMSO : 6.4 mg/mL (12.71 mM; Need ultrasonic and warming)H2O : < 0.1 mg/mL (insoluble)

form 

Powder

pka

8.25±0.70(Predicted)

color 

Off-white to yellow

MRS 1706 Usage And Synthesis

Description

MRS1706 is a selective adenosine A_2B receptor inverse agonist with K_i values of 1.39, 157, 112, and 230 nM for human A_2B, A₁, A_2A, and A₃ receptors, respectively.

Uses

MRS 1706 is a selective and potent Adenosine A2B-R inverse agonist Ki (binding affinity) values of 1.39, 157, 112, and 230 nM for human A2B, A1, A2A, and A3 receptors, respectively.

Biological Activity

Potent and selective adenosine A 2B receptor inverse agonist (K i values are 1.39, 157, 112 and 230 nM for human A 2B , A 1 , A 2A and A 3 receptors respectively).

MRS 1706(264622-53-9)Related Product Information

• 2-(4-ETHOXY-PHENYL)-1H-IMIDAZOLE
• 1,3-DIPROPYL-8-PHENYLXANTHINE
• 8-PHENYLTHEOPHYLLINE
• MRS 1706
• 1,3-DIETHYL-8-PHENYLXANTHINE