Basic information Safety Supplier Related

CYS-TYR-ILE-THR-ASN-CYS-GLY-LEU-GLY-NH2

Basic information Safety Supplier Related

CYS-TYR-ILE-THR-ASN-CYS-GLY-LEU-GLY-NH2 Basic information

Product Name:
CYS-TYR-ILE-THR-ASN-CYS-GLY-LEU-GLY-NH2
Synonyms:
  • thr(4)-gly(7)-oxytoci
  • [THR4, GLY7] OT
  • [THR4, GLY7]-OXYTOCIN
  • CYS-TYR-ILE-THR-ASN-CYS-GLY-LEU-GLY-NH2
  • H-CYS-TYR-ILE-THR-ASN-CYS-GLY-LEU-GLY-NH2
  • H-CYS-TYR-ILE-THR-ASN-CYS-GLY-LEU-GLY-NH2, (DISULFIDE BOND)
  • 3,3-DiallylthiacarbocyanineBromide
  • Cys-Tyr-Ile-Thr-Asn-Cys-Gly-Leu-Gly-NH2 (Disulfide bridge Cys1-Cys6)
CAS:
60786-59-6
MF:
C39H61N11O12S2
MW:
940.1
Mol File:
60786-59-6.mol
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CYS-TYR-ILE-THR-ASN-CYS-GLY-LEU-GLY-NH2 Chemical Properties

Boiling point:
1489.4±65.0 °C(Predicted)
Density 
1.265±0.06 g/cm3(Predicted)
storage temp. 
−20°C
form 
Solid
pka
9.90±0.15(Predicted)
color 
White to off-white
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Safety Information

Hazard Codes 
Xn
Risk Statements 
20
Safety Statements 
36/37/39-45
WGK Germany 
3

MSDS

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CYS-TYR-ILE-THR-ASN-CYS-GLY-LEU-GLY-NH2 Usage And Synthesis

Uses

(Thr4,Gly7)-Oxytocin, an Oxytocin analogue, is a specific OT receptor agonist. (Thr4,Gly7)-Oxytocin also excites subicular neurons via activation of TRPV1 channels, and depression of K+ channels. [1][2].

in vivo

(Thr4,Gly7)-Oxytocin (1 μM, direct intra-PVT infusion for 1 min) evokes depolarization on TGOT-responsive neurons in mice[1].
(Thr4,Gly7)-Oxytocin (100 ng, intracerebroventrical injection) increases nitric oxide production in the paraventricular nucleus of the hypothalamus of male rats[3].

Animal Model:Swiss Webster mice [1]
Dosage:1 μM
Administration:Intratracheal administration for 24 h
Result:Excited 34.3% of aPVT neurons, 57.6% of mPVT neurons, and 60.0% of pPVT neurons.
Increased the firing rate of TGOT-responsive PVT neurons in all subregions.

References

[1] Lily R Barrett, et al. Oxytocin activation of paraventricular thalamic neurons promotes feeding motivation to attenuate stress-induced hypophagia. Neuropsychopharmacology. 2021 Apr;46(5):1045-1056. DOI:10.1038/s41386-021-00961-3
[2] Binqi Hu, et al. Activation of Oxytocin Receptors Excites Subicular Neurons by Multiple Signaling and Ionic Mechanisms. Cereb Cortex. 2021 Mar 31;31(5):2402-2415. DOI:10.1093/cercor/bhaa363
[3] M R Melis, et al. Oxytocin increases nitric oxide production in the paraventricular nucleus of the hypothalamus of male rats: correlation with penile erection and yawning. Regul Pept. 1997 Mar 26;69(2):105-11. DOI:10.1016/s0167-0115(97)00002-5

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