GW 284543 hydrochloride - UNC 10225170 hydrochloride
GW 284543 hydrochloride - UNC 10225170 hydrochloride Basic information
- Product Name:
- GW 284543 hydrochloride - UNC 10225170 hydrochloride
- Synonyms:
-
- GW 284543 hydrochloride - UNC 10225170 hydrochloride
- GW 284543 hydrochloride
- 6,7-Dimethoxy-N-(3-phenoxyphenyl)quinolin-4-amine hydrochloride
- W 284543 hydrochloride
- CAS:
- 179246-08-3
- MF:
- C23H21ClN2O3
- MW:
- 408.88
- Mol File:
- 179246-08-3.mol
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GW 284543 hydrochloride - UNC 10225170 hydrochloride Chemical Properties
- storage temp.
- Sealed in dry,Room Temperature
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GW 284543 hydrochloride - UNC 10225170 hydrochloride Usage And Synthesis
Uses
GW284543 (UNC10225170) hydrochloride is a selective MEK5 inhibitor. GW284543 reduces pERK5, and decreases endogenous MYC protein[1].
IC 50
MEK5
References
[1] Vaseva AV, et al. KRAS Suppression-Induced Degradation of MYC Is Antagonized by a MEK5-ERK5 Compensatory Mechanism. Cancer Cell. 2018 Nov 12;34(5):807-822.e7. DOI:10.1016/j.ccell.2018.10.001
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