Basic information Safety Supplier Related

L371,257

Basic information Safety Supplier Related

L371,257 Basic information

Product Name:
L371,257
Synonyms:
  • L371,257
  • 1-[4-[(1-Acetyl-4-piperidinyl)oxy]-2-methoxybenzoyl]-4-(2-oxo-2H-3,1-benzoxazin-1(4H)-yl)piperidine
  • 1-[1-[4-(1-acetylpiperidin-4-yl)oxy-2-methoxybenzoyl]piperidin-4-yl]-4H-3,1-benzoxazin-2-one
  • 2H-3,1-Benzoxazin-2-one, 1-[1-[4-[(1-acetyl-4-piperidinyl)oxy]-2-methoxybenzoyl]-4-piperidinyl]-1,4-dihydro-
CAS:
162042-44-6
MF:
C28H33N3O6
MW:
507.58
Mol File:
162042-44-6.mol
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L371,257 Chemical Properties

Boiling point:
728.9±60.0 °C(Predicted)
Density 
1.282±0.06 g/cm3(Predicted)
storage temp. 
Store at RT
pka
0.73±0.20(Predicted)
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L371,257 Usage And Synthesis

Biological Activity

Potent, high affinity human oxytocin (OT) receptor antagonist (K i = 4.6 nM) that displays > 800-fold selectivity over human arginine vasopressin receptors V 1a and V 2 . Antagonizes oxytocin-induced contractions in isolated rat uterine tissue (pA 2 = 8.44) and in anesthetised rats following intravenous and intraduodenal administration. Orally active.

L371,257Supplier

3B Pharmachem (Wuhan) International Co.,Ltd.
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821-50328103-801
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3bsc@sina.com
BOC Sciences
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Email
info@bocsci.com
EMMX Biotechnology LLC
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888-539-0666
Email
info@emmx.com
Target Molecule Corp
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781-999-5354
Email
marketing@targetmol.com
Jiangsu yize medical technology co. LTD
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Email
23903480@qq.com