CJ 033466
CJ 033466 Basic information
- Product Name:
- CJ 033466
- Synonyms:
-
- CJ 033466
- 5-Amino-6-chloro-2-methyl-N-[[1-(2-methylpropyl)-4-piperidinyl]methyl]-imidazo[1,2-a]pyridine-8-carboxamide
- Imidazo[1,2-a]pyridine-8-carboxamide, 5-amino-6-chloro-2-methyl-N-[[1-(2-methylpropyl)-4-piperidinyl]methyl]-
- 5-HT Receptor,Inhibitor,inhibit,gastroprokinetic,CJ-033466,CJ033466,Serotonin Receptor,gastrointestinal dysfunction,CJ 033466,5-hydroxytryptamine Receptor
- 5-amino-6-chloro-2-methyl-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}imidazo[1,2-a]pyridine-8-carboxamide
- CJ 033466, 10 mM in DMSO
- CAS:
- 519148-48-2
- MF:
- C19H28ClN5O
- MW:
- 377.91
- Mol File:
- 519148-48-2.mol
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CJ 033466 Chemical Properties
- storage temp.
- Store at +4°C
- solubility
- Soluble to 100 mM in DMSO and to 100 mM in ethanol
- form
- Powder
- color
- Light yellow to light brown
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CJ 033466 Usage And Synthesis
Uses
CJ 033466 is a partial, potent, and selective SR-4 agonist.
Biological Activity
Potent and selective 5-HT 4 partial agonist (EC 50 = 0.927 nM). Displays > 1000-fold selectivity for 5-HT 4 over other 5-HT and D 2 receptors. Exhibits gastroprokinetic effects in vivo following oral administration. Weakly blocks hERG (IC 50 = 2.6 μ M).
IC 50
5-HT4 Receptor: 9 nM (EC50)
CJ 033466Supplier
3B Pharmachem (Wuhan) International Co.,Ltd.
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- 821-50328103-801 18930552037
- 3bsc@sina.com
BOC Sciences
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- 1-631-485-4226; 16314854226
- info@bocsci.com
Shanghai Lollane Biological Technology Co.,Ltd.
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- 021-52996696，15000506266 15000506266
EMMX Biotechnology LLC
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- 888-539-0666
- info@emmx.com
Shanghai YuanYe Biotechnology Co., Ltd.
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- 021-61312847; 18021002903
- 3008007409@qq.com