ChemicalBook > Product Catalog > Biochemical Engineering > Biochemical Reagents > Agonist Inhibitors > BET-BAY-002
BET-BAY-002
BET-BAY-002 Basic information
- Product Name:
- BET-BAY-002
- Synonyms:
-
- BET-BAY 002
- BET-BAY-002
- (4R)-6-(4-Chlorophenyl)-1-methyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4H-[1,2,4]triazolo[4,3-a][1]benzazepine
- 4H-[1,2,4]Triazolo[4,3-a][1]benzazepine, 6-(4-chlorophenyl)-1-methyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-, (4R)-
- BET BAY 002,BETBAY 002
- CAS:
- 1588521-78-1
- MF:
- C22H18ClN5O
- MW:
- 403.86
- Mol File:
- 1588521-78-1.mol
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BET-BAY-002 Chemical Properties
- Boiling point:
- 635.7±65.0 °C(Predicted)
- Density
- 1.40±0.1 g/cm3(Predicted)
- storage temp.
- Store at -20°C
- solubility
- DMSO: ≥ 50 mg/mL (123.81 mM)
- pka
- 2.44±0.60(Predicted)
- form
- Powder
- color
- White to off-white
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BET-BAY-002 Usage And Synthesis
Uses
BET-BAY 002 is a potent BET inhibitor; shows efficacy in a multiple myeloma model.
References
[1] Evans DM,?et al. Exposure?time?versus?cytotoxicity?for?anticancer agents.Cancer Chemother Pharmacol.?2019 Aug;84(2):359-371. DOI:10.1007/s00280-019-03863-w
[2] Jung M,?et al. Targeting?BET?bromodomains?for?cancer?treatment. Epigenomics.?2015;7(3):487-501. DOI:10.2217/epi.14.91
BET-BAY-002Supplier
BOC Sciences
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- 1-631-485-4226; 16314854226
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Haoyuan Chemexpress Co., Ltd.
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- 021-58950125
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- +86-21-5821 5861
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