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Agonist Inhibitors
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- Structure:
- Chemical Name:
- Afamelanotide acetate
- CAS:
- 1566590-77-9
- MF:
- C80H115N21O21
- Structure:
- Chemical Name:
- Saroglitazar (Magnesium)
- CAS:
- 1639792-20-3
- MF:
- C50H56MgN2O8S2
- Chemical Name:
- Eloralintide
- CAS:
- 2883634-40-8
- Structure:
- Chemical Name:
- (1R,3S)-5-[2-[(1R,3aR,7aS)-1-[(2R,5S)-5-hydroxy-6-methyl-heptan-2-yl]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-4-ylidene]ethylidene]-4-methylidene-cyclohexane-1,3-diol
- CAS:
- 93129-94-3
- MF:
- C27H46O4
- Structure:
- Chemical Name:
- 1 NM-PP1
- CAS:
- 221244-14-0
- MF:
- C20H21N5
- Structure:
- Chemical Name:
- (E)-1-[(1S)-1-(4-Fluorophenyl)ethyl]-3-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)benzylidene]piperidin-2-one
- CAS:
- 870843-42-8
- MF:
- C25H26FN3O2
- Structure:
- Chemical Name:
- LASOFOXIFENE HCL
- CAS:
- 190791-29-8
- MF:
- C32H37NO8
- Structure:
- Chemical Name:
- SAG
- CAS:
- 912545-86-9
- MF:
- C28H28ClN3OS
- Structure:
- Chemical Name:
- Coelenterazine
- CAS:
- 55779-48-1
- MF:
- C26H21N3O3
- Structure:
- Chemical Name:
- 5'-D(ATGAAAATCAGGGTTAGG)-3', SODIUM SALT
- CAS:
- 1047953-91-2
- MF:
- C19H17Cl3N4O3
- Structure:
- Chemical Name:
- H-ALA-TYR-PRO-GLY-LYS-PHE-NH2
- CAS:
- 352017-71-1
- MF:
- C34H48N8O7
- Structure:
- Chemical Name:
- ML-7 HYDROCHLORIDE
- CAS:
- 110448-33-4
- MF:
- C15H18ClIN2O2S
- Structure:
- Chemical Name:
- Sapropterin Hydrochloride
- CAS:
- 69056-38-8
- MF:
- C9H17Cl2N5O3
- Structure:
- Chemical Name:
- EFONIDIPINE
- CAS:
- 111011-63-3
- MF:
- C34H38N3O7P
- Structure:
- Chemical Name:
- MONASTROL
- CAS:
- 329689-23-8
- MF:
- C14H16N2O3S
- Structure:
- Chemical Name:
- 3-[3-[N-(2-CHLORO-3-TRIFLUOROMETHYLBENZYL)-(2,2-DIPHENYLETHYL)AMINO]PROPYLOXY]PHENYLACETIC ACID HYDROCHLORIDE
- CAS:
- 405911-09-3
- MF:
- C33H31ClF3NO3
- Structure:
- Chemical Name:
- ORITAVANCIN
- CAS:
- 171099-57-3
- MF:
- C86H97Cl3N10O26
- Structure:
- Chemical Name:
- OTAVA-BB 7070707015
- CAS:
- 934593-90-5
- MF:
- C26H29NO5
- Structure:
- Chemical Name:
- (2-METHOXY-5-[2-(2,4,6-TRIMETHOXY-PHENYL)-ETHENESULFONYLMETHYL]-PHENYLAMINO)-ACETIC ACID, SODIUM SALT
- CAS:
- 592542-59-1
- MF:
- C21H25NO8S
- Structure:
- Chemical Name:
- BIBF-1120
- CAS:
- 928326-83-4
- MF:
- C31H33N5O4
- Structure:
- Chemical Name:
- ONO-AE3-208
- CAS:
- 402473-54-5
- MF:
- C24H21FN2O3
- Structure:
- Chemical Name:
- (R)-5,6-Dihydro-5-(methylamino)-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (Z)-2-butenedioate
- CAS:
- 179386-44-8
- MF:
- C15H17N3O5
- Structure:
- Chemical Name:
- 3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyclopenta[c]pyrazole
- CAS:
- 851776-28-8
- MF:
- C7H8N6
- Structure:
- Chemical Name:
- LX-1606 Hippurate
- CAS:
- 1033805-22-9
- MF:
- C27H26ClF3N6O3
- Structure:
- Chemical Name:
- Doravirine
- CAS:
- 1338225-97-0
- MF:
- C17H11ClF3N5O3
- Structure:
- Chemical Name:
- AZ-23
- CAS:
- 915720-21-7
- MF:
- C17H19ClFN7O
- Structure:
- Chemical Name:
- 3--Phenyl-N-(2,2,2-trichloro-1-((((4-chlorophenyl)amino)carbonothioyl)amino)ethyl)acrylamide
- CAS:
- 1164470-53-4
- MF:
- C18H15Cl4N3OS
- Structure:
- Chemical Name:
- 2-[(1-Methylpropyl)dithio]-1H-imidazole
- CAS:
- 141400-58-0
- MF:
- C7H12N2S2
- Structure:
- Chemical Name:
- 4-(2,3-Dihydro-1,4-benzodioxin-6-yl)-2,4-dihydro-5-[(5-nitro-2-thiazolyl)thio]-3H-1,2,4-triazol-3-one
- CAS:
- 883065-90-5
- MF:
- C13H9N5O5S2
- Structure:
- Chemical Name:
- BMS-599626
- CAS:
- 873837-23-1
- MF:
- C27H28ClFN8O3
- Structure:
- Chemical Name:
- N-[2-Fluoro-5-[[3-[(1E)-2-(2-pyridinyl)ethenyl]-1H-indazol-6-yl]amino]phenyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
- CAS:
- 319460-94-1
- MF:
- C26H22FN7O
- Structure:
- Chemical Name:
- Saxagliptin hydrate
- CAS:
- 945667-22-1
- MF:
- C18H27N3O3
- Structure:
- Chemical Name:
- KX2-391
- CAS:
- 1038395-65-1
- MF:
- C20H21ClN4O
- Structure:
- Chemical Name:
- 5-Phenyl-1,2,5-thiadiazolidin-3-one 1,1-dioxide
- CAS:
- 612530-44-6
- MF:
- C8H8N2O3S
- Structure:
- Chemical Name:
- VU 0357017 hydrochloride
- CAS:
- 1135242-13-5
- MF:
- C18H28ClN3O3
- Structure:
- Chemical Name:
- N-[2-[[(2,3-Difluorophenyl)methyl]thio]-6-[[(1S,2R)-2,3-dihydroxy-1-methylpropyl]amino]-4-pyrimidinyl]-1-azetidinesulfonamide
- CAS:
- 1204707-73-2
- MF:
- C18H23F2N5O4S2
- Structure:
- Chemical Name:
- Azilsartan kaMedoxoMil
- CAS:
- 863031-24-7
- MF:
- C30H25KN4O8
- Structure:
- Chemical Name:
- Nortadalafil
- CAS:
- 171596-36-4
- MF:
- C21H17N3O4
- Structure:
- Chemical Name:
- (R)-XL518
- CAS:
- 934660-94-3
- MF:
- C21H21F3IN3O2
- Structure:
- Chemical Name:
- AM-679
- CAS:
- 1206880-66-1
- MF:
- C40H44N4O5S
- Structure:
- Chemical Name:
- SMER 28
- CAS:
- 307538-42-7
- MF:
- C11H10BrN3
- Structure:
- Chemical Name:
- (RS)-4-(3-MethylaMino-1-thiophen-2-yl-propyl)-naphthalen-1-ol
- CAS:
- 949095-98-1
- MF:
- C18H19NOS
- Structure:
- Chemical Name:
- NSC-348884
- CAS:
- 81624-55-7
- MF:
- C38H40N10
- Structure:
- Chemical Name:
- N-2-Biphenylyl-7-nitro-2,1,3-benzoxadiazol-4-aMine
- CAS:
- 413611-93-5
- MF:
- C18H12N4O3
- Structure:
- Chemical Name:
- (1,3-Benzothiazol-2-yl)[2-[[4-[(morpholin-4-yl)methyl]benzyl]oxy]pyrimidin-4-yl]acetonitrile
- CAS:
- 848344-36-5
- MF:
- C25H23N5O2S
- Structure:
- Chemical Name:
- 2-Methyl-5-(1-methylethyl)-2,5-cyclohexadiene-1,4-dione 1-[O-(2-methylbenzoyl)oxime]
- CAS:
- 321688-88-4
- MF:
- C18H19NO3
- Structure:
- Chemical Name:
- GAP 26
- CAS:
- 197250-15-0
- MF:
- C70H107N19O19S
- Structure:
- Chemical Name:
- GNE-490
- CAS:
- 1033739-92-2
- MF:
- C18H22N6O2S
- Structure:
- Chemical Name:
- BEZ235 (Tosylate)
- CAS:
- 1028385-32-1
- MF:
- C37H31N5O4S
- Structure:
- Chemical Name:
- Daun02
- CAS:
- 290304-24-4
- MF:
- C41H44N2O20
- Structure:
- Chemical Name:
- I2906
- CAS:
- 331963-29-2
- MF:
- C25H37N3O4
- Structure:
- Chemical Name:
- NBD-556
- CAS:
- 333353-44-9
- MF:
- C17H24ClN3O2
- Structure:
- Chemical Name:
- D3263 HCl salt
- CAS:
- 1008763-54-9
- MF:
- C21H32ClN3O3
- Structure:
- Chemical Name:
- Umeclidinium bromide
- CAS:
- 869113-09-7
- MF:
- C29H34BrNO2
- Structure:
- Chemical Name:
- 4-IsoxazolecarboxaMide, 3-(2-chlorophenyl)-N-(4-chlorophenyl)-N,5-diMethyl-
- CAS:
- 1197300-24-5
- MF:
- C18H14Cl2N2O2
- Structure:
- Chemical Name:
- A-443654
- CAS:
- 552325-16-3
- MF:
- C24H23N5O
- Structure:
- Chemical Name:
- LeterMovir
- CAS:
- 917389-32-3
- MF:
- C29H28F4N4O4
- Structure:
- Chemical Name:
- AP1903
- CAS:
- 195514-63-7
- MF:
- C78H98N4O20
- Structure:
- Chemical Name:
- Bavisant
- CAS:
- 929622-08-2
- MF:
- C19H27N3O2
- Structure:
- Chemical Name:
- CHR-6494
- CAS:
- 1333377-65-3
- MF:
- C16H16N6
- Structure:
- Chemical Name:
- DG 051 (HCl salt)
- CAS:
- 929915-58-2
- MF:
- C21H25Cl2NO4
- Structure:
- Chemical Name:
- Elagolix Sodium
- CAS:
- 832720-36-2
- MF:
- C32H29F5N3NaO5
- Structure:
- Chemical Name:
- EMD638683
- CAS:
- 1181770-72-8
- MF:
- C18H18F2N2O4
- Structure:
- Chemical Name:
- N6022
- CAS:
- 1208315-24-5
- MF:
- C24H22N4O3
- Structure:
- Chemical Name:
- SB-674042
- CAS:
- 483313-22-0
- MF:
- C24H21FN4O2S
- Structure:
- Chemical Name:
- SQ 109
- CAS:
- 502487-67-4
- MF:
- C22H38N2
- Structure:
- Chemical Name:
- UNC0321
- CAS:
- 1238673-32-9
- MF:
- C27H45N7O3
- Structure:
- Chemical Name:
- tiraseMtiv (CK-2017357)
- CAS:
- 1005491-05-3
- MF:
- C12H14N4O
- Structure:
- Chemical Name:
- ARRY-520 (R enantioMer)
- CAS:
- 885060-08-2
- MF:
- C20H22F2N4O2S
- Structure:
- Chemical Name:
- MK8245 Trifluoroacetate
- CAS:
- 1415559-41-9
- MF:
- C19H17BrF4N6O6
- Structure:
- Chemical Name:
- VUF11207
- CAS:
- 1378524-41-4
- MF:
- C27H35FN2O4
- Structure:
- Chemical Name:
- Bexagliflozin
- CAS:
- 1118567-05-7
- MF:
- C24H29ClO7
- Structure:
- Chemical Name:
- LY2801653
- CAS:
- 1206799-15-6
- MF:
- C30H22F2N6O3
- Structure:
- Chemical Name:
- LGD-4033
- CAS:
- 1165910-22-4
- MF:
- C14H12F6N2O
- Structure:
- Chemical Name:
- 1-(4-AMino-phenyl)-3-(4-tert-butyl-benzoyl)-thiourea
- CAS:
- 1011301-27-1
- MF:
- C18H21N3OS
- Structure:
- Chemical Name:
- RRX-001
- CAS:
- 925206-65-1
- MF:
- C5H6BrN3O5
- Structure:
- Chemical Name:
- PST2286
- CAS:
- 26629-41-4
- MF:
- C23H34O5
- Structure:
- Chemical Name:
- A 438079 (hydrochloride)
- CAS:
- 899431-18-6
- MF:
- C13H10Cl3N5
- Structure:
- Chemical Name:
- Bavisant (dihydrochloride)
- CAS:
- 929622-09-3
- MF:
- C19H28ClN3O2
- Structure:
- Chemical Name:
- (S)-2-(1-((2-aMino-9H-purin-6-yl)aMino)ethyl)-5-Methyl-3-(o-tolyl)quinazolin-4(3H)-one hydrochloride
- CAS:
- 1431697-78-7
- MF:
- C23H23ClN8O
- Structure:
- Chemical Name:
- Delafloxacin meglumine
- CAS:
- 352458-37-8
- MF:
- C18H12ClF3N4O4.C7H17NO5
- Structure:
- Chemical Name:
- GS9620
- CAS:
- 1228585-88-3
- MF:
- C22H30N6O2
- Structure:
- Chemical Name:
- Kalydeco hydrate
- CAS:
- 1134822-07-3
- MF:
- C24H30N2O4
- Structure:
- Chemical Name:
- MethylproaMine
- CAS:
- 188247-01-0
- MF:
- C28H31N7
- Structure:
- Chemical Name:
- MLN-120B
- CAS:
- 783348-36-7
- MF:
- C19H15ClN4O2
- Structure:
- Chemical Name:
- RAS-2410 hydrochloride
- CAS:
- 1187075-34-8
- MF:
- C16H20ClN3O4S
- Structure:
- Chemical Name:
- VcMMAD
- CAS:
- 1401963-17-4
- MF:
- C70H104N12O14S
- Structure:
- Chemical Name:
- ARN-2966
- CAS:
- 102212-26-0
- MF:
- C12H12N2O
- Structure:
- Chemical Name:
- Auristatin F
- CAS:
- 163768-50-1
- MF:
- C40H67N5O8
- Structure:
- Chemical Name:
- PF-4989216
- CAS:
- 1276553-09-3
- MF:
- C18H13FN6OS
- Structure:
- Chemical Name:
- PDK1 Inhibitor
- CAS:
- 850717-64-5
- MF:
- C15H14N4O2
- Structure:
- Chemical Name:
- 2-Naphthalenecarboxylic acid, 3-hydroxy-, 2-[(2,4,5-trihydroxyphenyl)Methylene]hydrazide
- CAS:
- 1256493-34-1
- MF:
- C18H14N2O5
- Structure:
- Chemical Name:
- CCT 244747
- CAS:
- 1404095-34-6
- MF:
- C20H24N8O2
- Structure:
- Chemical Name:
- Cort-108297
- CAS:
- 1018679-79-2
- MF:
- C26H25F4N3O3S
- Structure:
- Chemical Name:
- (S)-2-[4-(4-Chloro-phenyl)-2,3,9-triMethyl-6H-1-thia-5,7,8,9a-tetraaza-cyclopenta[e]azulen-6-yl]-acetaMide
- CAS:
- 202591-23-9
- MF:
- C19H18ClN5OS
- Structure:
- Chemical Name:
- NISOXETINE HYDROCHLORIDE
- CAS:
- 57754-86-6
- MF:
- C17H22ClNO2
- Structure:
- Chemical Name:
- N-((S)-1-(4-((S)-2-(2,4-dichlorophenylsulfonaMido)-3-hydroxypropanoyl)piperazin-1-yl)-4-Methyl-1-oxopentan-2-yl)benzo[b]thiophene-2-carboxaMide
- CAS:
- 942206-85-1
- MF:
- C28H32Cl2N4O6S2
- Structure:
- Chemical Name:
- K145
- CAS:
- 1309444-75-4
- MF:
- C18H24N2O3S
- Structure:
- Chemical Name:
- AP20187
- CAS:
- 195514-80-8
- MF:
- C82H107N5O20
- Structure:
- Chemical Name:
- 2 - (4 - Methylphenyl) - 1,2 - benzisothiazol - 3(2H)-one
- CAS:
- 2514-30-9
- MF:
- C14H11NOS