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Agonist Inhibitors

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Structure:
Chemical Name:
LEE011 (succinate)
CAS:
1374639-75-4
MF:
C27H36N8O5
Structure:
Chemical Name:
Cyclopentanone, 2,5-bis(2-thienylMethylene)-, (E,E)-
CAS:
176957-55-4
MF:
C15H12OS2
Structure:
Chemical Name:
Dihexa
CAS:
1401708-83-5
MF:
C27H44N4O5
Structure:
Chemical Name:
RPI-1
CAS:
269730-03-2
MF:
C17H15NO4
Structure:
Chemical Name:
Bedaquiline fumarate
CAS:
845533-86-0
MF:
C36H35BrN2O6
Structure:
Chemical Name:
DDR1-IN-1
CAS:
1449685-96-4
MF:
C30H31F3N4O3
Structure:
Chemical Name:
SM-164
CAS:
957135-43-2
MF:
C62H84N14O6
Structure:
Chemical Name:
Elamipretide
CAS:
736992-21-5
MF:
C32H49N9O5
Structure:
Chemical Name:
CASIN
CAS:
425399-05-9
MF:
C20H22N2O
Structure:
Chemical Name:
Eravacycline
CAS:
1207283-85-9
MF:
C27H31FN4O8
Structure:
Chemical Name:
Val-cit-PAB-OH
CAS:
159857-79-1
MF:
C18H29N5O4
Structure:
Chemical Name:
CP-640186 (hydrochloride)
CAS:
591778-70-0
MF:
C30H36ClN3O3
Structure:
Chemical Name:
HLM006474
CAS:
353519-63-8
MF:
C25H25N3O2
Structure:
Chemical Name:
ML365
CAS:
947914-18-3
MF:
C22H20N2O3
Structure:
Chemical Name:
NSC-41589
CAS:
6310-41-4
MF:
C9H11NOS
Structure:
Chemical Name:
VT-464 (raceMate)
CAS:
1375603-36-3
MF:
C18H17F4N3O3
Structure:
Chemical Name:
ACK1-B19
CAS:
1234480-46-6
MF:
C24H27N7O2
Structure:
Chemical Name:
CFI-400945
CAS:
1338806-73-7
MF:
C33H34N4O3
Structure:
Chemical Name:
SGI 7079
CAS:
1239875-86-5
MF:
C26H26FN7
Structure:
Chemical Name:
CB-839
CAS:
1439399-58-2
MF:
C26H24F3N7O3S
Structure:
Chemical Name:
GS-9820
CAS:
870281-34-8
MF:
C21H16FN7O
Structure:
Chemical Name:
PP2 analog
CAS:
309739-67-1
MF:
C16H17ClN4
Structure:
Chemical Name:
BET-BAY-002
CAS:
1588521-78-1
MF:
C22H18ClN5O
Structure:
Chemical Name:
ReModelin
CAS:
949912-58-7
MF:
C15H14N4S
Structure:
Chemical Name:
FMoc-Val-Cit-PAB-PNP
CAS:
863971-53-3
MF:
C40H42N6O10
Structure:
Chemical Name:
ASP-9521
CAS:
1126084-37-4
MF:
C19H26N2O3
Structure:
Chemical Name:
Y16
CAS:
429653-73-6
MF:
C24H20N2O3
Structure:
Chemical Name:
lifitegrast
CAS:
1025967-78-5
MF:
C29H24Cl2N2O7S
Structure:
Chemical Name:
Altiratinib
CAS:
1345847-93-9
MF:
C26H21F3N4O4
Structure:
Chemical Name:
AZD6738
CAS:
1352226-88-0
MF:
C20H24N6O2S
Structure:
Chemical Name:
N,N′-(Sulfonyldi-4,1-phenylene)bis[2,2,3,3-tetramethyl-cyclopropanecarboxamide
CAS:
329059-55-4
MF:
C28H36N2O4S
Structure:
Chemical Name:
CID-49830258
CAS:
1346527-98-7
MF:
C23H20N6O
Structure:
Chemical Name:
ONO-4059
CAS:
1351635-67-0
MF:
C25H24N6O3
Structure:
Chemical Name:
1-(2-Hydroxyethyl)imidazolidine-2-thione
CAS:
932-49-0
MF:
C5H10N2OS
Structure:
Chemical Name:
1-(2,4-DICHLOROPHENYL)-5-(4-IODOPHENYL)-4-METHYL-N-4-MORPHOLINYL-1H-PYRAZOLE-3-CARBOXAMIDE
CAS:
202463-68-1
MF:
C21H19Cl2IN4O2
Structure:
Chemical Name:
Tenapanor
CAS:
1234423-95-0
MF:
C50H66Cl4N8O10S2
Structure:
Chemical Name:
GDC-0810(ARN-810)
CAS:
1365888-06-7
MF:
C26H20ClFN2O2
Structure:
Chemical Name:
RQ-00203078
CAS:
1254205-52-1
MF:
C21H13ClF6N2O5S
Structure:
Chemical Name:
WEHI-345
CAS:
1354825-58-3
MF:
C22H23N7O
Structure:
Chemical Name:
TP-3654
CAS:
1361951-15-6
MF:
C22H25F3N4O
Structure:
Chemical Name:
LMI070
CAS:
1562338-42-4
MF:
C22H27N5O2
Structure:
Chemical Name:
Vps34-IN-1
CAS:
1383716-33-3
MF:
C21H24ClN7O
Structure:
Chemical Name:
ZA7371
CAS:
1494675-86-3
MF:
C18H21N5O3
Structure:
Chemical Name:
NSC59984
CAS:
803647-40-7
MF:
C12H15N3O4
Structure:
Chemical Name:
Larotrectinib Sulfate
CAS:
1223405-08-0
MF:
C21H24F2N6O6S
Structure:
Chemical Name:
BBT594
CAS:
882405-89-2
MF:
C28H30F3N7O3
Structure:
Chemical Name:
BP-1-102
CAS:
1334493-07-0
MF:
C29H27F5N2O6S
Structure:
Chemical Name:
BMS-986020
CAS:
1257213-50-5
MF:
C29H26N2O5
Structure:
Chemical Name:
ABT-639
CAS:
1235560-28-7
MF:
C20H20ClF2N3O3S
Structure:
Chemical Name:
Glesatinib (hydrochloride)
CAS:
1123838-51-6
MF:
C31H28ClF2N5O3S2
Structure:
Chemical Name:
AS1842856
CAS:
836620-48-5
MF:
C18H22FN3O3
Structure:
Chemical Name:
ALS-8176 (active form)
CAS:
1445379-92-9
MF:
C10H13ClFN3O4
Structure:
Chemical Name:
GDC-0084
CAS:
1382979-44-3
MF:
C18H22N8O2
Structure:
Chemical Name:
AZ6102
CAS:
1645286-75-4
MF:
C25H28N6O
Structure:
Chemical Name:
2-(1,3-DIMETHYL-2,6-DIOXO-1,2,3,6-TETRAHYDRO-7H-PURIN-7-YL)-N-(4-ISOPROPYLPHENYL)ACETAMIDE
CAS:
349085-38-7
MF:
C18H21N5O3
Structure:
Chemical Name:
BENZIMIDAVIR
CAS:
176161-24-3
MF:
C15H19Cl2N3O4
Structure:
Chemical Name:
(5-METHOXY-1H-INDOL-2-YL)PHENYLMETHANONE
CAS:
74588-78-6
MF:
C16H13NO2
Structure:
Chemical Name:
5,6-DIHYDRO-2,3-DIMETHOXY-6,6-DIMETHYLBENZ[7,8]INDOLIZINO[2,3-B]QUINOXALINE
CAS:
163769-88-8
MF:
C22H21N3O2
Structure:
Chemical Name:
TG 003
CAS:
719277-26-6
MF:
C13H15NO2S
Structure:
Chemical Name:
ONO-4059 (hydrochloride)
CAS:
1439901-97-9
MF:
C25H23ClN6O3
Structure:
Chemical Name:
CBR-5884
CAS:
681159-27-3
MF:
C14H12N2O4S2
Structure:
Chemical Name:
ARS-853
CAS:
1629268-00-3
MF:
C22H29ClN4O3
Structure:
Chemical Name:
IMR-1A
CAS:
331862-41-0
MF:
C13H11NO5S2
Structure:
Chemical Name:
NVP-BAW2881
CAS:
861875-60-7
MF:
C22H15F3N4O2
Structure:
Chemical Name:
CCT196969
CAS:
1163719-56-9
MF:
C27H24FN7O3
Structure:
Chemical Name:
LY-3177833
CAS:
1627696-51-8
MF:
C16H12FN5O
Structure:
Chemical Name:
HA-15
CAS:
1609402-14-3
MF:
C23H22N4O3S2
Structure:
Chemical Name:
PF-06282999
CAS:
1435467-37-0
MF:
C13H12ClN3O3S
Structure:
Chemical Name:
RR6
CAS:
1351758-37-6
MF:
C16H23NO4
Structure:
Chemical Name:
UNC3866
CAS:
1872382-47-2
MF:
C43H66N6O8
Structure:
Chemical Name:
SDZ285-428
CAS:
174262-13-6
MF:
C24H20ClN3O
Structure:
Chemical Name:
XMD16-5
CAS:
1345098-78-3
MF:
C23H24N6O2
Structure:
Chemical Name:
N-(3-((2-((3-Fluoro-4-(4-methylpiperazin-1-yl)phenyl)amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)phenyl)acrylamide maleate
CAS:
1557268-88-8
MF:
C30H30FN7O6
Structure:
Chemical Name:
TYRPHOSTIN B48
CAS:
133550-35-3
MF:
C16H12N2O3
Structure:
Chemical Name:
Adenosine 5'-monophosphate monohydrate
CAS:
18422-05-4
MF:
C10H16N5O8P
Structure:
Chemical Name:
Eprazinone dihydrochloride
CAS:
10402-53-6
MF:
C24H33ClN2O2
Structure:
Chemical Name:
4-AMINO-5-CHLORO-2-METHOXYBENZOIC ACID
CAS:
7206-70-4
MF:
C8H8ClNO3
Structure:
Chemical Name:
2-[1-BENZYL-4-PIPERIDYL]-2-PHENYLGLUTARIMIDE
CAS:
5633-14-7
MF:
C23H27ClN2O2
Structure:
Chemical Name:
2-Acetyl-4-butyramidophenol
CAS:
40188-45-2
MF:
C12H15NO3
Structure:
Chemical Name:
Nortropine
CAS:
538-09-0
MF:
C7H13NO
Structure:
Chemical Name:
(+/-)-BAY K 8644
CAS:
71145-03-4
MF:
C16H15F3N2O4
Structure:
Chemical Name:
SC-43
CAS:
1400989-25-4
MF:
C21H13ClF3N3O2
Structure:
Chemical Name:
PEN (human)
CAS:
597578-70-6
MF:
C97H159N27O32
Structure:
Chemical Name:
4-AMINO-N-(2-PHENYLETHYL)BENZENESULFONAMIDE
CAS:
587850-67-7
MF:
C14H16N2O2S
Structure:
Chemical Name:
CHK2 INHIBITOR II
CAS:
516480-79-8
MF:
C20H14ClN3O2
Structure:
Chemical Name:
TIZOXANIDE
CAS:
173903-47-4
MF:
C10H7N3O4S
Structure:
Chemical Name:
2-Methoxyphenothiazine
CAS:
1771-18-2
MF:
C13H11NOS
Structure:
Chemical Name:
TDZD-8
MF:
C10H10N2O2S
Structure:
Chemical Name:
H-SER-LEU-LEU-LYS-NH2
CAS:
464924-27-4
MF:
C21H41N5O6
Structure:
Chemical Name:
N-Phenylbenzylamine
CAS:
103-32-2
MF:
C13H13N
Structure:
Chemical Name:
1-(2,3-DIHYDRO-1,4-BENZODIOXIN-5-YL)-PIPERAZINE HYDROCHLORIDE
CAS:
98224-03-4
MF:
C12H16N2O2
Structure:
Chemical Name:
4-[(5,6,7,8-TETRAHYDRO-5,5,8,8-TETRAMETHYL-2-NAPHTHALENYL)CARBOXAMIDO]BENZOIC ACID
CAS:
102121-60-8
MF:
C22H25NO3
Structure:
Chemical Name:
N-(6-CHLORO-9H-PYRIDO[3,4-B]INDOL-8-YL)-3-PYRIDINECARBOXAMIDE DIHYDROCHLORIDE
CAS:
431898-65-6
MF:
C17H11ClN4O
Structure:
Chemical Name:
NS3861 >=98% (HPLC)
CAS:
216853-59-7
MF:
C12H14BrNS
Structure:
Chemical Name:
9-(2,3-DIDEOXY-2-FLUORO-ALPHA-D-THREOPENTOFURANOSYL)-ADENINE
CAS:
110143-10-7
MF:
C10H12FN5O2
Structure:
Chemical Name:
methyl N-ethyl-N-[4-[(5-nitro-2,1-benzisothiazol-3-yl)azo]phenyl]-beta-alaninate
CAS:
52239-04-0
MF:
C19H19N5O4S
Structure:
Chemical Name:
1,3-Benzenedicarboxylic acid, 5-[4,2':6',4''-terpyridin]-4'-yl-
CAS:
1610059-51-2
MF:
C23H15N3O4
Structure:
Chemical Name:
IKARISOSIDE F
CAS:
113558-14-8
MF:
C31H36O14
Structure:
Chemical Name:
Quinagolide hydrochloride
CAS:
94424-50-7
MF:
C20H34ClN3O3S
Chemical Name:
VX-745