1-BOC-5-METHOXYINDOLE Chemical Properties

Melting point:

75-79 °C

Boiling point:

357.3±34.0 °C(Predicted)

Density 

1.10±0.1 g/cm3(Predicted)

storage temp. 

Inert atmosphere,2-8°C

CAS DataBase Reference

99275-47-5(CAS DataBase Reference)

Safety Information

Hazard Codes 

Xi,Xn

Risk Statements 

22-36

Safety Statements 

26

RIDADR 

UN 2811 6.1/PG 3

WGK Germany 

3

Hazard Note 

Harmful/Irritant/Keep Cold

1-BOC-5-METHOXYINDOLE Usage And Synthesis

Uses

Reactant for preparation of:• ;Asymmetric intramolecular Friedel-Crafts alkylation reaction1• ;Palladium-catalyzed carboaminoxylations with arylboronic acids and TEMPO catalyst2• ;Fluorescent pyrimidopyrimidoindole nucleosides via Suzuki-Miyaura coupling reaction3• ;Novel conformationally restricted β- and γ-amino acids4• ;2-(Indolyl) borates, silanes, and silanols5• ;DNA minor groove alkylating agents as stable amine-based prodrugs designed for tumor-specific release6

Uses

Reactant for preparation of:

• Asymmetric intramolecular Friedel-Crafts alkylation reaction
• Palladium-catalyzed carboaminoxylations with arylboronic acids and TEMPO catalyst
• Fluorescent pyrimidopyrimidoindole nucleosides via Suzuki-Miyaura coupling reaction
• Novel conformationally restricted β- and γ-amino acids
• 2-(Indolyl) borates, silanes, and silanols
• DNA minor groove alkylating agents as stable amine-based prodrugs designed for tumor-specific release

1-BOC-5-METHOXYINDOLE(99275-47-5)Related Product Information

• 1-Boc-5-hydroxyindole
• 1-BOC-5-METHOXYINDOLE
• BOC-5-METHOXYINDOLE-3-CARBOXALDEHYDE
• 1-BOC-5-METHOXYINDOLE-2-BORONIC ACID,N-BOC-5-METHOXYINDOLE-2-BORONIC ACID
• 5-BENZYLOXY-1-BOC-INDOLE-2-BORONIC ACID
• N-BOC-6-METHOXYINDOLE-2-BORONIC ACID,1-BOC-6-METHOXYINDOLE-2-BORONIC ACID
• 1-BOC-7-methoxyindole-2-boronic acid
• 5-Methoxyindole
• 3-BROMO-5-METHOXYINDOLE-1-CARBOXYLIC ACID TERT-BUTYL ESTER
• TERT-BUTYL 3-(CYANOMETHYL)-5-METHOXY-1H-INDOLE-1-CARBOXYLATE
• 1-(TERT-BUTOXYCARBONYL)-5-(TRIFLUOROMETHOXY)INDOLE-2-BORONIC ACID
• 3-HYDROXYMETHYL-5-METHOXYINDOLE-1-CARBOXYLIC ACID TERT-BUTYL ESTER
• 3-IODO-5-METHOXYINDOLE-1-CARBOXYLIC ACID TERT-BUTYL ESTER
• 1-BOC-6-METHOXYINDOLE,N-BOC-6-METHOXYINDOLE
• N-BOC-5-METHOXYTRYPTOPHOL
• 5-BENZYLOXY-3-BROMOINDOLE-1-CARBOXYLIC ACID TERT-BUTYL ESTER
• 5-BENZYLOXY-3-FORMYLINDOLE-1-CARBOXYLIC ACID TERT-BUTYL ESTER
• 2-ETHYL-3-HYDROXYMETHYL-5-METHOXY-INDOLE-1-CARBOXYLIC ACID TERT-BUTYL ESTER