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Erdosteine

Product Name
Erdosteine
CAS No.
84611-23-4
Chemical Name
Erdosteine
Synonyms
pv144;RV-144;KW-9144;Erdosten;Erdostiene;ERDOSTEINE;Dithiosteine;Erdosteine>ERDOSTEINE BP98;Erdosteine, ≥ 98.0%
CBNumber
CB0230173
Molecular Formula
C8H11NO4S2
Formula Weight
249.31
MOL File
84611-23-4.mol
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Erdosteine Property

Melting point:
156-160°C
Boiling point:
590.4±50.0 °C(Predicted)
Density 
1.48±0.1 g/cm3(Predicted)
storage temp. 
Sealed in dry,2-8°C
solubility 
Acetonitrile (Slightly), DMSO (Slightly), Methanol (Slightly)
pka
3.71(at 25℃)
form 
Solid
color 
White to Off-White
λmax
236nm(H2O)(lit.)
Merck 
14,3647
InChIKey
QGFORSXNKQLDNO-UHFFFAOYSA-N
CAS DataBase Reference
84611-23-4(CAS DataBase Reference)
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Safety

RTECS 
AJ1476200
HS Code 
2934.99.9001
Toxicity
LD50 in mice and rats (g/kg): >10 orally; >3.5 i.v. (Gonella)
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H320Causes eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

TCI Chemical
Product number
E1026
Product name
Erdosteine
Purity
>98.0%(GC)(T)
Packaging
1g
Price
$51
Updated
2024/03/01
TCI Chemical
Product number
E1026
Product name
Erdosteine
Purity
>98.0%(GC)(T)
Packaging
5g
Price
$153
Updated
2024/03/01
Cayman Chemical
Product number
29177
Product name
Erdosteine
Packaging
1g
Price
$121
Updated
2024/03/01
Cayman Chemical
Product number
29177
Product name
Erdosteine
Packaging
25g
Price
$1201
Updated
2024/03/01
Cayman Chemical
Product number
29177
Product name
Erdosteine
Packaging
5g
Price
$362
Updated
2024/03/01
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Erdosteine Chemical Properties,Usage,Production

Description

Erdosteine is a new expectorant introduced in France for the treatment of chronic bronchitis. Erdosteine possesses mucomodulator, mucolytic, mucokinetic and free radical scavenging properties. Its therapeutic efficacy has been demonstrated in patients affected by congestion and viscous mucus in higher and lower respiratory tracts as in acute and chronic bronchitis, sinusitis, otitis, tracheopharyngitis and coryza. Erdosteine acts through its active metabolites containing free sulfhydryl groups which are able to depolymerize the mucopolysaccharides of the excreatum by breaking the disulfide linkages (thereby lowing its viscosity). The prodrug approach provides unique characteristics to erdosteine by offering stable therapeutic efficacy and prevention of the gastric mucus from lythic phenomena. The agent was also reported to have local antiinflammatory and antielastase properties and enhances penetration of antibiotics into bronchial mucus.

Description

Erdosteine is a mucolytic agent and an antioxidant. It inhibits LPS-induced IκB kinase (IKK) activity, NF-κB-mediated transcription, and production of IL-6 and IL-1β in RAW 264.7 cells. Erdosteine (7.5 mg/kg) prevents depletion of renal catalase and glutathione peroxidase (GPX) and increases in renal malondialdehyde (MDA) and nitric oxide (NO) levels in a rat model of nephrotoxicity induced by cisplatin . It reduces spinal cord lipid peroxidation and destruction of spinal motor neurons in a rabbit model of spinal cord ischemia and reperfusion injury induced by thoracoabdominal aortic clamping. Erdosteine (150 mg/kg) reduces lung weight, MDA and protein carbonyl levels, and macrophage and neutrophil accumulation in a mouse model of acute lung injury induced by oleic acid (Item Nos. 90260 | 24659). Formulations containing erdosteine have been used in the treatment of chronic obstructive pulmonary disease (COPD).

Chemical Properties

Off-White Solid

Originator

Refarmed (Switzerland)

Uses

A mucolytic, developed for the treatment of chronic obstructive bronchitis.

Uses

Erdosteine is a mucolytic. Erdosteine was developed for the treatment of chronic obstructive bronchitis.

Definition

ChEBI: Erdosteine is a N-acyl-amino acid.

brand name

Edirel; Vectrine

Erdosteine Preparation Products And Raw materials

Raw materials

Preparation Products

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Erdosteine Suppliers

TCI Europe
Tel
320-37350700
Fax
+32 (0)37350701
Email
sales@tcieurope.eu
Country
Europe
ProdList
23671
Advantage
75
ecochem international chemical broker
Tel
--
Fax
--
Email
export@ecochem.dk
Country
Europe
ProdList
6371
Advantage
66
kemikalieimport
Tel
--
Fax
--
Email
Sales@kemikalieimport.dk
Country
Europe
ProdList
6685
Advantage
47
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View Lastest Price from Erdosteine manufacturers

BEIJING SJAR TECHNOLOGY DEVELOPMENT CO., LTD.
Product
Erdosteine 84611-23-4
Price
US $0.00/g
Min. Order
1g
Purity
More Than 99%
Supply Ability
100kg/Month
Release date
2024-09-06
Hangzhou Hyper Chemicals Limited
Product
Erdosteine 84611-23-4
Price
US $0.00-0.00/KG
Min. Order
1KG
Purity
99%, USP
Supply Ability
5,000KG
Release date
2024-08-30
XINGTAI XINGJIU NEW MATERIAL TECHNOLOGY CO., LTD
Product
Erdosteine 84611-23-4
Price
US $55.00/KG
Min. Order
1KG
Purity
99.9%
Supply Ability
500MT/month
Release date
2021-12-20

84611-23-4, ErdosteineRelated Search:


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  • SECRESOLV
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