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Rilmenidine

Product Name
Rilmenidine
CAS No.
54187-04-1
Chemical Name
Rilmenidine
Synonyms
s3341;Tenaxum;Hyperium;S-3341-3;RILMENIDINE;oxaminozoline;TENAXUM; HYPERIUM;Rilmenidine USP/EP/BP;Rilmenidinehemifuramate;RilMenidine heMifuMarate sa
CBNumber
CB0391076
Molecular Formula
C10H16N2O
Formula Weight
180.25
MOL File
54187-04-1.mol
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Rilmenidine Property

Melting point:
106-107°
Boiling point:
355.5±9.0 °C(Predicted)
Density 
1.45±0.1 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
H2O: 7.3 mg/mL
form 
solid
pka
7.88±0.50(Predicted)
color 
white
CAS DataBase Reference
54187-04-1(CAS DataBase Reference)
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Safety

Safety Statements 
22-24/25
WGK Germany 
3
RTECS 
RP7207400
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

American Custom Chemicals Corporation
Product number
API0004072
Product name
RILMENIDINE
Purity
95.00%
Packaging
10MG
Price
$284.55
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0004072
Product name
RILMENIDINE
Purity
95.00%
Packaging
50MG
Price
$1073.29
Updated
2021/12/16
AHH
Product number
MT-58447
Product name
Rilmenidine
Purity
98%
Packaging
0.1g
Price
$310
Updated
2021/12/16
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Rilmenidine Chemical Properties,Usage,Production

Description

Rilmenidine is a new antihypertensive agent with a selective alphaz-agonist/antagonist profile, reportedly useful in the management of mild to moderate hypertension. Its fmt-line indication is possible because of the clear dissociation of its antihypertensive activity from other neurophannacological effects.

Chemical Properties

water soluble

Originator

Servier (France)

Uses

I1-imidazoline binding site ligand and a2-adrenoceptor agonist, exhibits higher I1 vs. a2 selectivity than clonidine

Definition

ChEBI: Rilmenidine is an isourea.

brand name

Hyperium

Biological Activity

I 1 -imidazoline binding site selective ligand and α 2 -adrenoceptor agonist. Possesses greater I 1 vs α 2 selectivity than the prototypical compound, clonidine.

Metabolic pathway

In short-term rat hepatocyte cultures, oxaminozoline is metabolized and its four metabolites resulting from oxidation or hydrolysis are identified, three of which are identical to those reported in vivo. The presence of an additional minor metabolite in culture may be due to the higher metabolic rate of oxaminozoline in this model system.

Rilmenidine Preparation Products And Raw materials

Raw materials

Monoethanolamine Phenyl chloroformate 2-Chloroethyl isocyanate Thionyl chloride

Preparation Products

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Rilmenidine Suppliers

China 95 Czech 1 Europe 3 Germany 2 India 3 United Kingdom 5 United States 21 Global 130
3B Pharmachem (Wuhan) International Co.,Ltd.
Tel
821-50328103-801 18930552037
Fax
86-21-50328109
Email
3bsc@sina.com
Country
China
ProdList
15839
Advantage
69
JinYan Chemicals(ShangHai) Co.,Ltd.
Tel
13817811078
Fax
86-021-50426522,50426273
Email
sales@jingyan-chemical.com
Country
China
ProdList
9976
Advantage
60
LGM Pharma
Tel
1-(800)-881-8210
Fax
615-250-9817
Email
inquiries@lgmpharma.com
Country
United States
ProdList
2123
Advantage
70
XiaoGan ShenYuan ChemPharm co,ltd
Tel
15527768850
Email
1791901229@qq.com
Country
China
ProdList
8844
Advantage
52
Jinan Trio PharmaTech Co., Ltd.
Tel
+86 (531) 88811783
Fax
+86 (531) 55696010 QQ 1762738062
Email
sales@trio-pharmatech.com (International market)
Country
China
ProdList
1856
Advantage
62
BOC Sciences
Tel
1-631-485-4226; 16314854226
Email
info@bocsci.com
Country
United States
ProdList
14055
Advantage
65
Shanghai T&W Pharmaceutical Co., Ltd.
Tel
+86 21 61551611
Fax
+86 21 50676805
Country
China
ProdList
9891
Advantage
58
AdooQ BioScience, LLC
Tel
+1 (866) 930-6790
Fax
+1 (866) 333-9607
Email
info@adooq.com
Country
United States
ProdList
2782
Advantage
58
Shanghai Meishui Chemical Technology Co., Ltd
Tel
021-60549325 18616193163
Fax
021-33250306
Country
China
ProdList
4526
Advantage
56
Huainan Kedi Chemical Factory
Tel
0554-2106669
Fax
0554-2666215
Email
sales1@kedichem.com
Country
China
ProdList
4924
Advantage
55
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View Lastest Price from Rilmenidine manufacturers

Zhuozhou Wenxi import and Export Co., Ltd
Product
Rilmenidine 54187-04-1
Price
US $15.00-10.00/KG
Min. Order
1KG
Purity
99%+ HPLC
Supply Ability
Monthly supply of 1 ton
Release date
2021-08-11
Longyan Tianhua Biological Technology Co., Ltd
Product
Rilmenidine 54187-04-1
Price
US $5.00/KG
Min. Order
25KG
Purity
99
Supply Ability
999
Release date
2020-11-11
Shaanxi Dideu Medichem Co. Ltd
Product
Rilmenidine 54187-04-1
Price
US $0.00-0.00/Kg
Min. Order
1KG
Purity
99.0%
Supply Ability
500 MT
Release date
2020-05-09

54187-04-1, RilmenidineRelated Search:

3-Methyl-2-butanone Dihydromyrcenol N,N-Diisopropylethylamine Tolyltriazole 5-Methyl-1H-benzotriazole Chloromethyl isopropyl carbonate Cyclopropyl methyl ketone Allylamine Dicyclopropane methylamine (R)-1-(Cyclopropylethyl)amine (S)-1-CYCLOPROPYLETHYLAMINE RILMENIDINE DIHYDROGEN PHOSPHATE,rilmenidine phosphate O-METHYLISOUREA ACETATE RILMENIDINE FOR SYSTEM SUITABILITY Oxazoline RILMENIDINE DIHYDROGENOPHOSPHATE - REFERENCE SPECTRUM RILMENIDINE HEMIFUMARATE SALT CHEMBRDG-BB 4003538

  • n-(dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine
  • oxaminozoline
  • RILMENIDINE
  • 1,1-dicyclopropyl-n-(2-oxazolinyl)-methylamin
  • 2-((dicyclopropylmethyl)imino)-oxazolidin
  • 2-((dicyclopropylmethyl)imino)oxazolidine
  • 2-(dicyclopropylmethylamino)-2-oxazoline
  • 4,5-dihydro-n-(dicyclopropylmethyl)-2-oxazolamin
  • s3341
  • N-(dicyclopropylmethyl)-4,5-dihydrooxazol-2-amine
  • 2-(N-(Dicyclopropylmethyl)amino)oxazolinehemifuramate
  • Rilmenidinehemifuramate
  • Rilmenidine 2-[(Dicyclopropylmethyl)amino]-2-oxazoline
  • Hyperium
  • S-3341-3
  • RilMenidine heMifuMarate sa
  • 2-[N-(Dicyclopropylmethyl)amino]oxazoline fumarate (2:1) salt
  • N-(2-Oxazolin-2-yl)-α,α-dicyclopropylmethanamine
  • Oxaminozoline hemifumarate salt
  • Rilmenidene hemifumarate salt
  • Tenaxum
  • TENAXUM; HYPERIUM
  • 2-Oxazolamine, N-(dicyclopropylmethyl)-4,5-dihydro-
  • Rilmenidine USP/EP/BP
  • RilmenidineQ: What is Rilmenidine Q: What is the CAS Number of Rilmenidine Q: What is the storage condition of Rilmenidine
  • N-(dicyclopropyl methyl)-4, 5-dihydro2-oxazolamide
  • 54187-04-1
  • 54178-04-1
  • C10H16N2OC4H4O4
  • C10H16N2O05C4H4O4
  • C10H16N2O189C4H4O4
  • Antihypertensive
  • Imidazoline binding site