Uses
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Baloxavir

Uses
Product Name
Baloxavir
CAS No.
1985605-59-1
Chemical Name
Baloxavir
Synonyms
(R)-12-((S)-7,8-difluoro-6,11-dihydrodibenzo[b,e]thiepin-11-yl)-7-hydroxy-3,4,12,12a-tetrahydro-1H-[1,4]oxazino[3,4-c]pyrido[2,1-f][1,2,4]triazine-6,8-dione;S-033447;CPD2051;Baloxavir;Baloshavir;New Baloxavir;Baloxavir (Xofluza;Baloxavir USP/EP/BP;Baloxavir Impurity 10;BXA,endonuclease,S033447,Influenza Virus
CBNumber
CB04662930
Molecular Formula
C24H19F2N3O4S
Formula Weight
483.49
MOL File
1985605-59-1.mol
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Baloxavir Property

Boiling point:
644.7±65.0 °C(Predicted)
Density 
1.63±0.1 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
DMSO:41.67(Max Conc. mg/mL);86.19(Max Conc. mM)
form 
A solid
pka
4.50±1.00(Predicted)
color 
White to yellow
CAS DataBase Reference
1985605-59-1
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

ChemScene
Product number
CS-0039267
Product name
Baloxavir
Purity
98.92%
Packaging
5mg
Price
$350
Updated
2021/12/16
ChemScene
Product number
CS-0039267
Product name
Baloxavir
Purity
98.92%
Packaging
10mg
Price
$650
Updated
2021/12/16
ChemScene
Product number
CS-0039267
Product name
Baloxavir
Purity
98.92%
Packaging
25mg
Price
$1250
Updated
2021/12/16
ChemScene
Product number
CS-0039267
Product name
Baloxavir
Purity
98.92%
Packaging
50mg
Price
$1950
Updated
2021/12/16
ChemScene
Product number
CS-0039267
Product name
Baloxavir
Purity
98.92%
Packaging
100mg
Price
$3000
Updated
2021/12/16
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Baloxavir Chemical Properties,Usage,Production

Uses

Baloxavir is a drug employed in the treatment of influenza virus infection.
Baloxavir marboxil is a selective inhibitor of influenza cap-dependent endonuclease. It has shown therapeutic activity in preclinical models of influenza A and B virus infections, including strains resistant to current antiviral agents.

Uses

Baloxavir is a drug employed in the treatment of influenza virus infection.

Mechanism of action

Baloxavir marboxil is an influenza therapeutic agent, specifically, an enzyme inhibitor targeting the influenza virus' cap-dependent endonuclease activity, one of the activities of the virus polymerase complex. In particular, it inhibits a process known as cap snatching, by which the virus derives short, capped primers from host cell RNA transcripts, which it then uses for polymerase-catalyzed synthesis of its needed viral mRNAs. A polymerase subunit binds to the host pre-mRNAs at their 5' caps, then the polymerase's endonuclease activity catalyzes its cleavage "after 10–13 nucleotides". As such, its mechanism is distinct from neuraminidase inhibitors such as oseltamivir and zanamivir.

Side effects

Common side effects following the single dose administration of baloxavir marboxil include diarrhea, bronchitis, common cold, headache, and nausea. Adverse events were reported in 21% of people who received baloxavir, 25% of those receiving placebo, and 25% of oseltamivir.

Baloxavir Preparation Products And Raw materials

Raw materials

Preparation Products

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View Lastest Price from Baloxavir manufacturers

HangZhou RunYan Pharma Technology Co.,LTD.
Product
Baloxavir marboxil 1985605-59-1
Price
US $0.00-0.00/g
Min. Order
1g
Purity
99% HPLC
Supply Ability
10000
Release date
2024-09-19
Cangzhou Kangrui Pharma Tech Co. Ltd.,
Product
Baloxavir 1985605-59-1
Price
US $0.00-0.00/g
Min. Order
25g
Purity
99%
Supply Ability
10kgs
Release date
2024-10-18
Hebei Yanxi Chemical Co., Ltd.
Product
Baloxavir 1985605-59-1
Price
US $0.00-0.00/kg
Min. Order
1kg
Purity
99%
Supply Ability
100tons
Release date
2023-08-16

1985605-59-1, BaloxavirRelated Search:


  • Baloxavir
  • CPD2051
  • Baloxavir Impurity 10
  • S-033447
  • New Baloxavir
  • 1H-[1,4]Oxazino[3,4-c]pyrido[2,1-f][1,2,4]triazine-6,8-dione, 12-[(11S)-7,8-difluoro-6,11-dihydrodibenzo[b,e]thiepin-11-yl]-3,4,12,12a-tetrahydro-7-hydroxy-, (12aR)-
  • Baloxavir USP/EP/BP
  • (R)-12-((S)-7,8-difluoro-6,11-dihydrodibenzo[b,e]thiepin-11-yl)3,4,12,12a-tetrahydro-1H-[1,4]oxazino[3,4-c]pyrido[2,1-f][1,2’4]triazine-6,8- dione
  • Baloxavir (Xofluza
  • 1H-[1,4]Oxazino[3,4-c]pyrido[2,1-f][1,2,4]triazine-6,8-dione,12-[(11S)-7Chemicalbook,8-difluoro-6,11-dihydrodibenzo[b,e]thiepin-11-yl]-3,4,12,12a-tetrahydro-7-hydroxy-,(12aR)-
  • (R)-12-((S)-7,8-difluoro-6,11-dihydrodibenzo[b,e]thiepin-11-yl)-7-hydroxy-3,4,12,12a-tetrahydro-1H-[1,4]oxazino[3,4-c]pyrido[2,1-f][1,2,4]triazine-6,8-dione
  • (3R)-2-[(11S)-7,8-difluoro-6,11-dihydrobenzo[c][1]benzothiepin-11-yl]-11-hydroxy-5-oxa-1,2,8-triazatricyclo[8.4.0.03,8]tetradeca-10,13-diene-9,12-dione
  • BXA,endonuclease,S033447,Influenza Virus
  • influenza,RNA,inhibit,dolutegravir,Baloxavir,Inhibitor,cap-dependent,S 033447,CEN,transcription,replication
  • (3R)-2-[(11S)-7,8-difluoro-6,11-dihydrobenzo[c][1]benzothiepin-11-yl]-11-hydroxy-5-oxa-1,2,8-triazatricyclo[8.4.0.03?]tetradeca-10,13-diene-9,12-dione
  • Baloshavir
  • 1985605-59-1
  • 1985605-14-1
  • C24H19F2N3O4S
  • API
  • 1985605-59-1