ChemicalBook > CAS DataBase List > BETAZOLE HYDROCHLORIDE

BETAZOLE HYDROCHLORIDE

Product Name
BETAZOLE HYDROCHLORIDE
CAS No.
138-92-1
Chemical Name
BETAZOLE HYDROCHLORIDE
Synonyms
histalog;Histimin;gastramine;Histalog (TN);betazolehydrochloride;betazoledihydrochloride;2-(3-Pyrazolyl)ethylamin;ametazoledihydrochloride;Betazole hydrochloride (JAN);BETAZOLE HYDROCHLORIDE (200 MG)
CBNumber
CB0501633
Molecular Formula
C5H11Cl2N3
Formula Weight
184.06694
MOL File
138-92-1.mol
More
Less

BETAZOLE HYDROCHLORIDE Property

Melting point:
224-226°
storage temp. 
Store at -20°C
solubility 
DMSO: 37 mg/mL (201.01 mM);Ethanol: 18 mg/mL (97.79 mM)
Water Solubility 
Water: 37 mg/mL (201.01 mM)
More
Less

Safety

HS Code 
2933199090
More
Less

Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

More
Less

N-Bromosuccinimide Price

TRC
Product number
B276680
Product name
BetazoleDihydrochloride
Packaging
2.5mg
Price
$160
Updated
2021/12/16
Biosynth Carbosynth
Product number
FP126823
Product name
Betazole dihydrochloride
Packaging
250mg
Price
$172.5
Updated
2021/12/16
Biosynth Carbosynth
Product number
FP126823
Product name
Betazole dihydrochloride
Packaging
2g
Price
$867
Updated
2021/12/16
Apolloscientific
Product number
OR471576
Product name
2-(3-Pyrazolyl)ethanaminedihydrochloride
Packaging
5g
Price
$1827
Updated
2021/12/16
Matrix Scientific
Product number
077451
Product name
[2-(1H-Pyrazol-3-yl)ethyl]amine dihydrochloride
Packaging
5g
Price
$2310
Updated
2021/12/16
More
Less

BETAZOLE HYDROCHLORIDE Chemical Properties,Usage,Production

Originator

Histalog,Lilly,US,1953

Uses

Betazole Hydrochloride is a histamine H2 receptor agonist that is used as a gastric stimulant for the investigation of gastric secretion activity.

Definition

ChEBI: The dihydrochloride salt of betazole.

Manufacturing Process

A solution of 55 grams (1.1 mol) of hydrazine hydrate in 100 ml of methanol was cooled in a water bath and stirred while a solution of 48 grams (0.50 mol) of pure γ-pyrone in 100 ml of methanol was added over a period of about 15 minutes. After the addition was complete, the solution was allowed to stand at room temperature for about 1 hour, and was placed in a 1 liter hydrogenation bomb. 25 ml of liquid ammonia were added cautiously with stirring, followed by about 15 cc of Raney nickel catalyst. The bomb was charged with hydrogen to 1,800 pounds pressure, heated to 90°C and agitated. The quantity of hydrogen required to convert the hydrazone into the desired aminoethylpyrazole was taken up in about 3 hours. The bomb was cooled and opened, and the contents filtered. The filtrate was evaporated under reduced pressure to remove the methanol and the residual liquid was distilled under reduced pressure, whereby there were obtained 44.5 grams (81% yield) of 3-β-aminoethylpyrazole boiling at 118°-123°C at a pressure of 0.5 mm of Hg.

brand name

Histalog (Lilly).

Therapeutic Function

Diagnostic aid (gastric secretion)

BETAZOLE HYDROCHLORIDE Preparation Products And Raw materials

Raw materials

Preparation Products

More
Less

BETAZOLE HYDROCHLORIDE Suppliers

Carbosynth
Tel
--
Fax
--
Email
sales@carbosynth.com
Country
United Kingdom
ProdList
6005
Advantage
58
Apollo Scientific Ltd.
Tel
--
Fax
--
Email
sales@apolloscientific.co.uk
Country
United Kingdom
ProdList
6084
Advantage
88
Whyte Chemicals
Tel
--
Fax
--
Email
sales@whytechemicals.co.uk
Country
United Kingdom
ProdList
3748
Advantage
50

138-92-1, BETAZOLE HYDROCHLORIDERelated Search:


  • 2-(1H-pyrazol-5-yl)ethan-1-amine dihydrochloride
  • betazolehydrochloride
  • gastramine
  • histalog
  • BETAZOLE HYDROCHLORIDE (200 MG)
  • Histimin
  • [2-(1H-Pyrazol-3-yl)ethyl]amine dihydrochloride
  • 2-(1H-pyrazol-3-yl)ethanamine dihydrochloride
  • 2-(3-Pyrazolyl)ethylamin
  • 2-(2H-pyrazol-3-yl)ethanamine dihydrochloride
  • 2-(2H-pyrazol-3-yl)ethylamine dihydrochloride
  • ametazoledihydrochloride
  • betazoledihydrochloride
  • 1h-pyrazole-3-ethanamine,dihydrochloride
  • 3-(2-aminoethyl)-pyrazoldihydrochloride
  • 3-(2-aminoethyl)pyrazole,dihydrochloride
  • 3,5-beta-pyrazoleethylaminedihydrochloride
  • 3-beta-aminoethylpyrazoledihydrochloride
  • Betazole hydrochloride (JAN)
  • Histalog (TN)
  • Pyrazole, 3-(2-aminoethyl)-, dihydrochloride
  • 2-(3-Pyrazolyl)ethanamine Dihydrochloride
  • BETAZOLE HYDROCHLORIDE USP/EP/BP
  • Betazole Hydrochloride (1070006)
  • secretion,bile,Betazole,gastric,acid,Histamine Receptor,inhibit,Betazole dihydrochloride,duct,secretory,histalog,Ametazole,capacity,pressure,Inhibitor
  • 138-92-1
  • Amine, Heterocycles, Pharmaceuticals, Intermediates & Fine Chemicals