ChemicalBook > CAS DataBase List > macbecin I

macbecin I

Product Name
macbecin I
CAS No.
73341-72-7
Chemical Name
macbecin I
Synonyms
Macbecin;macbecin I;(15R)-6,17-Didemethoxy-15-methoxy-6-methyl-11-O-methyl-geldanamycin;(6S,15R)-6,17-Didemethoxy-15-methoxy-6-methyl-11-O-methylgeldanamycin;Geldanamycin, 6,17-didemethoxy-15-methoxy-6-methyl-11-O-methyl-, (15R)-
CBNumber
CB11346962
Molecular Formula
C30H42N2O8
Formula Weight
558.67
MOL File
73341-72-7.mol
More
Less

macbecin I Property

Melting point:
205-206 °C(Solv: ethanol (64-17-5); water (7732-18-5))
Boiling point:
736.2±60.0 °C(Predicted)
Density 
1.17±0.1 g/cm3(Predicted)
storage temp. 
Desiccate at -20°C
solubility 
Soluble in DMSO > 10 mM
form 
Powder
pka
8.62±0.70(Predicted)
More
Less

Hazard and Precautionary Statements (GHS)

More
Less

N-Bromosuccinimide Price

Cayman Chemical
Product number
22225
Product name
Macbecin I
Purity
≥95%
Packaging
1mg
Price
$291
Updated
2024/03/01
Tocris
Product number
3061
Product name
MacbecinI
Packaging
1
Price
$311
Updated
2021/12/16
Usbiological
Product number
255749
Product name
Macbecin I
Packaging
1mg
Price
$573
Updated
2021/12/16
TRC
Product number
M107525
Product name
MacbecinI
Packaging
0.5mg
Price
$1200
Updated
2021/12/16
ApexBio Technology
Product number
B7259
Product name
MacbecinI
Packaging
1mg
Price
$465
Updated
2021/12/16
More
Less

macbecin I Chemical Properties,Usage,Production

Uses

Macbecin I is an ansamycin antibiotic inhibitor of Hsp90 activity.

Biological Activity

Ansamycin antibiotic compound that inhibits Hsp90 activity (IC 50 = 2 μ M) by binding to the ATP-binding site. Exhibits antitumor and cytocidal activities (IC 50 ~ 0.4 μ M) by causing degradation of key oncogenic client proteins such as ErbB2 and cRaf1. Displays higher affinity and potency than geldanamycin (9,13-Dihydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-2-azabicyclo[16.3.1]docosa-4,6,10,18,21-pentaene-3,20,22-trione, 9-carbamate ).

macbecin I Preparation Products And Raw materials

Raw materials

Preparation Products

More
Less

macbecin I Suppliers

EMMX Biotechnology LLC
Tel
888-539-0666
Fax
888-539-0666
Email
info@emmx.com
Country
United States
ProdList
8447
Advantage
60
TargetMol Chemicals Inc.
Tel
+1-781-999-5354 +1-00000000000
Email
marketing@targetmol.com
Country
United States
ProdList
32161
Advantage
58
ApexBio Technology
Tel
--
Fax
--
Email
sales@apexbt.com
Country
United States
ProdList
6251
Advantage
58
BOC Sciences
Tel
16314854226
Email
info@bocsci.com
Country
United States
ProdList
9923
Advantage
65
Cayman Chemical Company
Tel
--
Fax
--
Email
cayman@caymanchem.com
Country
United States
ProdList
6213
Advantage
81
United States Biological
Tel
--
Fax
--
Email
chemicals@usbio.net
Country
United States
ProdList
6214
Advantage
80

73341-72-7, macbecin IRelated Search:


  • macbecin I
  • (6S,15R)-6,17-Didemethoxy-15-methoxy-6-methyl-11-O-methylgeldanamycin
  • (15R)-6,17-Didemethoxy-15-methoxy-6-methyl-11-O-methyl-geldanamycin
  • Geldanamycin, 6,17-didemethoxy-15-methoxy-6-methyl-11-O-methyl-, (15R)-
  • Macbecin
  • 73341-72-7