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ChemicalBook > CAS DataBase List > 5-BROMO-1H-INDOLE-3-CARBOXYLIC ACID METHYL ESTER

5-BROMO-1H-INDOLE-3-CARBOXYLIC ACID METHYL ESTER

Application
Product Name
5-BROMO-1H-INDOLE-3-CARBOXYLIC ACID METHYL ESTER
CAS No.
773873-77-1
Chemical Name
5-BROMO-1H-INDOLE-3-CARBOXYLIC ACID METHYL ESTER
Synonyms
RARECHEM AL BF 0374;Methyl 5-BroMoindole-3-carboxylate;METHYL 5-BROMO-1H-INDOLE-3-CARBOXYLATE;1H-Indole-3-carboxylicacid,5-broMo-,Methylester;5-BROMO-1H-INDOLE-3-CARBOXYLIC ACID METHYL ESTER;5-Bromo-1H-Indole-3-Carboxylic Acid Methyl Ester, 10 mM in DMSO
CBNumber
CB1191525
Molecular Formula
C10H8BrNO2
Formula Weight
254.08
MOL File
773873-77-1.mol
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5-BROMO-1H-INDOLE-3-CARBOXYLIC ACID METHYL ESTER Property

Melting point:
212-214 °C
Boiling point:
386.2±22.0 °C(Predicted)
Density 
1.629±0.06 g/cm3(Predicted)
storage temp. 
Sealed in dry,Room Temperature
pka
14.46±0.30(Predicted)
Appearance
White to off-white Solid
CAS DataBase Reference
773873-77-1
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Safety

HS Code 
2933998090
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

TRC
Product number
M295663
Product name
Methyl5-Bromoindole-3-carboxylate
Packaging
250mg
Price
$55
Updated
2021/12/16
AK Scientific
Product number
W8396
Product name
Methyl5-bromo-1H-indole-3-carboxylate
Packaging
1g
Price
$41
Updated
2021/12/16
Apolloscientific
Product number
OR962104
Product name
Methyl5-bromo-1H-indole-3-carboxylate
Purity
98%
Packaging
5g
Price
$65
Updated
2021/12/16
AK Scientific
Product number
J51148
Product name
Methyl5-bromo-1H-indole-3-carboxylate
Packaging
5g
Price
$80
Updated
2021/12/16
Matrix Scientific
Product number
073274
Product name
Methyl 5-bromo-1H-indole-3-carboxylate
Purity
95+%
Packaging
1g
Price
$82
Updated
2021/12/16
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5-BROMO-1H-INDOLE-3-CARBOXYLIC ACID METHYL ESTER Chemical Properties,Usage,Production

Application

Methyl 5-bromoindole-3-carboxylic acid can be used as an organic synthesis intermediate. It can be prepared in two steps from 5-bromo-1H-indole as a reactant, or it can be obtained by one-step esterification of 5-bromo-1H-indole-3-carboxylic acid.

Synthesis

67-56-1

10406-06-1

773873-77-1

GENERAL METHOD: 4.0 g of 5-bromo-1H-indole-3-carboxylic acid was dissolved in 40 times the volume (400 mL) of methanol and a catalytic amount of concentrated sulfuric acid was slowly added. The reaction mixture was heated to reflux for 5 hours, followed by slow cooling to room temperature. Ice-cold water was added to the cooled mixture and the yellow solid was collected by filtration. The solid was recrystallized from ethanol to give methyl 5-bromo-indole-3-carboxylate (12b) as a yellow solid in 62% yield. The product characterization data were as follows: melting point: 210-212 °C; IR (KBr, cm-1): 3213, 3114, 2929, 1745; 1H NMR (400 MHz, CDCl3): δ 3.93 (3H, s, -OCH3), 7.28 (1H, d, J = 8.8 Hz, Ar-H), 7.35 (1H, m, Ar-H ), 7.91 (1H, d, J = 2.8 Hz, Ar-H), 8.32 (1H, s, Ar-H), 8.67 (1H, s, -NH); 13C NMR (400 MHz, CDCl3 + DMSO-d6): δ 49.93, 105.91, 112.88, 113.75, 122.40, 124.26, 126.65, 131.89, 134.33, 164.13; HRMS (m/z): calculated value C10H9NO2Br [M]+: 253.98112, measured value: 253.98102.

References

[1] Chemical Papers, 2018, vol. 72, # 6, p. 1369 - 1378

5-BROMO-1H-INDOLE-3-CARBOXYLIC ACID METHYL ESTER Preparation Products And Raw materials

Raw materials

Preparation Products

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5-BROMO-1H-INDOLE-3-CARBOXYLIC ACID METHYL ESTER Suppliers

A.J Chemicals
Tel
--
Fax
--
Email
sales@ajchem.in
Country
India
ProdList
6100
Advantage
58
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View Lastest Price from 5-BROMO-1H-INDOLE-3-CARBOXYLIC ACID METHYL ESTER manufacturers

Career Henan Chemical Co
Product
5-BROMO-1H-INDOLE-3-CARBOXYLIC ACID METHYL ESTER 773873-77-1
Price
US $9.80/KG
Min. Order
1g
Purity
≥99%
Supply Ability
100kg
Release date
2020-01-08
Career Henan Chemical Co
Product
5-BROMO-1H-INDOLE-3-CARBOXYLIC ACID METHYL ESTER 773873-77-1
Price
US $1.00/KG
Min. Order
1KG
Purity
95-99%
Supply Ability
1ton
Release date
2020-01-08